Population Pharmacokinetic/Pharmacodynamic Analysis of the Glucokinase Activator PB201 in Healthy Volunteers and Patients with Type 2 Diabetes Mellitus: Facilitating the Clinical Development of PB201 in China Ling SongFangrui CaoDongyang Liu Original Research Article 20 November 2023 Pages: 93 - 108
How to Dose Vancomycin in Overweight and Obese Patients with Varying Renal (Dys)function in the Novel Era of AUC 400–600 mg·h/L-Targeted Dosing Tan ZhangElke H. J. KrekelsCatherijne A. J. Knibbe Original Research Article Open access 16 November 2023 Pages: 79 - 91
Preclinical Pharmacokinetic/Pharmacodynamic Studies and Clinical Trials in the Drug Development Process of EMA-Approved Antifungal Agents: A Review Theresa PechoMarkus Zeitlinger Review Article Open access 16 November 2023 Pages: 13 - 26
Development of a Generic Fetal Physiologically Based Pharmacokinetic Model and Prediction of Human Maternal and Fetal Organ Concentrations of Cefuroxime Xiaomei I. LiuDionna J. GreenAndré Dallmann Original Research Article 14 November 2023 Pages: 69 - 78
Pharmacokinetics, Safety, and Tolerability of Anti-SARS-CoV-2 Monoclonal Antibody, Sotrovimab, Delivered Intravenously or Intramuscularly in Japanese and Caucasian Healthy Volunteers Ahmed NaderElizabeth AlexanderDaren Austin Original Research Article Open access 13 November 2023 Pages: 57 - 68
Interplay of UDP-Glucuronosyltransferase and CYP2C8 for CYP2C8 Mediated Drug Oxidation and Its Impact on Drug–Drug Interaction Produced by Standardized CYP2C8 Inhibitors, Clopidogrel and Gemfibrozil Katsumi IgaAkiko Kiriyama Original Research Article 03 November 2023 Pages: 43 - 56
Evolution of Ritlecitinib Population Pharmacokinetic Models During Clinical Drug Development Jessica WojciechowskiVivek S PurohitTimothy Nicholas Original Research Article Open access 02 November 2023 Pages: 1765 - 1779
A Phase I, Open-Label, Fixed Sequence Study to Investigate the Effect of Cytochrome P450 2D6 Inhibition on the Pharmacokinetics of Ulotaront in Healthy Subjects Hironobu TsukadaYu-Luan ChenGerald R. Galluppi Original Research Article Open access 26 October 2023 Pages: 1755 - 1763
The Pharmacokinetics of the Nonsteroidal Mineralocorticoid Receptor Antagonist Finerenone Roland HeinigThomas Eissing Review Article Open access 24 October 2023 Pages: 1673 - 1693
Prognostic Value of Nivolumab Clearance in Non-Small Cell Lung Cancer Patients for Survival Early in Treatment Leila S. OttenBerber PietMichel M. van den Heuvel Original Research Article Open access 19 October 2023 Pages: 1749 - 1754
Safety, Pharmacokinetics, and Pharmacodynamics of SHR7280, a Non-peptide GnRH Antagonist in Premenopausal Women with Endometriosis: A Randomized, Double-Blind, Placebo-Controlled Phase 1 Study Yuan LiYing ZhengHongyan Guo Original Research Article 14 October 2023 Pages: 1739 - 1748
Plasma Pharmacokinetics of N-Acetylgalactosamine-Conjugated Small-Interfering Ribonucleic Acids (GalNAc-Conjugated siRNAs) Sebastian StenTim CardilinPeter Gennemark Leading Article Open access 12 October 2023 Pages: 1661 - 1672
Anti-coagulant Treatment of Cancer-Associated Thrombosis in Frail Patients: Impact of Frailties on the Management of Drug–Drug Interactions Claire GrangeCatherine RioufolSouad Assaad Review Article Open access 12 October 2023 Pages: 1523 - 1531
Population Pharmacokinetics of Total and Unbound Isavuconazole in Critically Ill Patients: Implications for Adaptive Dosing Strategies Anouk M. E. JansenBeatrijs MertensRoger J. M. Brüggemann Original Research Article Open access 11 October 2023 Pages: 1701 - 1711
High Variability in Isavuconazole Unbound Fraction in Clinical Practice: A Call to Reconsider Pharmacokinetic/Pharmacodynamic Targets and Breakpoints Anouk M. E. JansenRob ter HeineRoger J. M. Brüggemann Commentary Open access 11 October 2023 Pages: 1695 - 1699
Population Pharmacokinetics of Digoxin in Nonagenarian Patients: Optimization of the Dosing Regimen Angel Luis Salcedo-MingoarranzSusanna Edith Medellín-GaribayBenito García-Díaz Original Research Article 10 October 2023 Pages: 1725 - 1738
Pharmacokinetics and Tolerability of Zibotentan in Patients with Concurrent Moderate Renal and Moderate Hepatic Impairment Anne-Kristina MercierMikael SunnåkerJan Oscarsson Original Research Article Open access 06 October 2023 Pages: 1713 - 1724
Bridging the Worlds of Pharmacometrics and Machine Learning Kamilė StankevičiūtėJean-Baptiste WoillardMihaela van der Schaar Review Article 06 October 2023 Pages: 1551 - 1565
Clinical Pharmacokinetics of Ponesimod, a Selective S1P1 Receptor Modulator, in the Treatment of Multiple Sclerosis Terra M. KrugerBelén ValenzuelaJuan Jose Perez Ruixo Review Article 30 September 2023 Pages: 1533 - 1550
Escitalopram and Sertraline Population Pharmacokinetic Analysis in Pediatric Patients Ethan A. PoweleitZachary L. TaylorLaura B. Ramsey Original Research Article 27 September 2023 Pages: 1621 - 1637
Authors’ Reply to Ganijee et al.: “Comment on: Evaluation of the Influence of Sildenafil on Safety, Tolerability, Pharmacokinetics, and Pharmacodynamics of Vericiguat in Healthy Adults” Michael BoettcherCorina Becker Letter to the Editor Open access 26 September 2023 Pages: 1651 - 1653
Comment on: Evaluation of the Influence of Sildenafil on the Safety, Tolerability, Pharmacokinetics, and Pharmacodynamics of Vericiguat in Healthy Adults Mustafa GanijeeGaayen Ravii SahgalMalik Takreem Ahmad Letter to the Editor 26 September 2023 Pages: 1649 - 1650
Cannabidiol Exposure Through Maternal Marijuana Use: Predictions in Breastfed Infants Cindy H. T. YeungKerri A. BertrandAndrea N. Edginton Original Research Article 21 September 2023 Pages: 1611 - 1619
Mechanisms and Clinical Significance of Pharmacokinetic Drug Interactions Mediated by FDA and EMA-approved Hepatitis C Direct-Acting Antiviral Agents Michael Murray Review Article 20 September 2023 Pages: 1365 - 1392
Multivariate Exact Discrepancy: A New Tool for PK/PD Model Evaluation Sarah BakloutiEmmanuelle CometsDidier Concordet Original Research Article Open access 17 September 2023 Pages: 1599 - 1609
Irinotecan-Induced Toxicity: A Pharmacogenetic Study Beyond UGT1A1 Mirjam de WithLeni van DoornSander Bins Original Research Article Open access 16 September 2023 Pages: 1589 - 1597
Pharmacokinetics of Henagliflozin in Dialysis Patients with Diabetes Li DingShang LiuLeyi Gu Original Research Article 15 September 2023 Pages: 1581 - 1587
Imeglimin: A Clinical Pharmacology Review Clémence ChevalierPascale FouqueraySébastien Bolze Review Article 15 September 2023 Pages: 1393 - 1411
Assessing QTc Effects of Vericiguat Using Two Different Concentration-QTc Modeling Approaches Hauke RuehsAlexander SolmsMichaela Meyer Original Research Article Open access 06 September 2023 Pages: 1639 - 1648
Pharmacokinetics of Oral Vitamin D in Children with Obesity and Asthma Jason E. LangRodrigo Gonzalez RamirezLaura James Original Research Article Open access 30 August 2023 Pages: 1567 - 1579
Pharmacokinetics and Pharmacodynamics of Patisiran in Patients with hATTR Amyloidosis and with Polyneuropathy After Liver Transplantation Prajakta BadriBahru HabtemariamGabriel J. Robbie Original Research Article 28 August 2023 Pages: 1509 - 1522
Population Pharmacokinetic Analysis of Follicle-Stimulating Hormone During Ovarian Stimulation: Relation with Weight, Prolactin and Gene Polymorphism in THADA and ADIPOQ Xiaowei ZhangYu SuiYang Sui Original Research Article 26 August 2023 Pages: 1493 - 1507
Mirikizumab Pharmacokinetics in Patients with Moderately to Severely Active Ulcerative Colitis: Results from Phase III LUCENT Studies Laiyi ChuaStuart FriedrichXin Cindy Zhang Original Research Article Open access 23 August 2023 Pages: 1479 - 1491
Towards Model-Informed Precision Dosing of Voriconazole: Challenging Published Voriconazole Nonlinear Mixed-Effects Models with Real-World Clinical Data Franziska KluweRobin MicheletCharlotte Kloft Original Research Article Open access 21 August 2023 Pages: 1461 - 1477
Population Pharmacokinetic Modeling of Dolutegravir to Optimize Pediatric Dosing in HIV-1-Infected Infants, Children, and Adolescents Hardik ChandasanaMita Thaparfor the IMPAACT P1093, ODYSSEY (PENTA 20) Study Teams Original Research Article Open access 21 August 2023 Pages: 1445 - 1459
Enigma of Intramuscular Triamcinolone Acetonide (Kenalog®) Efficacy Sheeva ShahinfarHoward Maibach Review Article 19 August 2023 Pages: 1189 - 1199
Population Pharmacokinetic Analysis Supports Initiation Treatment and Bridging from Sublingual Buprenorphine to Subcutaneous Administration of a Buprenorphine Depot (CAM2038) in the Treatment of Opioid Use Disorder Marcus BjörnssonChayan AcharyaFredrik Tiberg Original Research Article Open access 16 August 2023 Pages: 1427 - 1443
Therapeutic Drug Monitoring of Kinase Inhibitors in Oncology Maud B. A. van der KleijNiels A. D. GuchelaarNeeltje Steeghs Review Article Open access 16 August 2023 Pages: 1333 - 1364
Pharmacokinetics of Antiretroviral Drugs in Older People Living with HIV: A Systematic Review Thainá ToledoThales CastroRita Estrela Systematic Review 10 August 2023 Pages: 1219 - 1230
Correction to: Pharmacokinetics of Nasal Esketamine in Patients with Allergic Rhinitis with and Without Nasal Decongestant Pretreatment and in Healthy Subjects with and Without Nasal Corticosteroid Pretreatment Peter ZannikosBhavna SolankiJaskaran Singh Correction 05 August 2023 Pages: 1329 - 1330
Correction: A Review of Population Pharmacokinetic Analyses of Linezolid Enrique Bandín-VilarLaura García-QuintanillaAnxo Fernández-Ferreiro Correction 03 August 2023 Pages: 1331 - 1331
Population Pharmacokinetic Analysis of Dorzagliatin in Healthy Subjects and Patients with Type 2 Diabetes Mellitus Kun WangLingge FengLi Chen Original Research Article Open access 03 August 2023 Pages: 1413 - 1425
CYP3A and CYP2C19 Activity Determined by Microdosed Probe Drugs Accurately Predict Voriconazole Clearance in Healthy Adults Amin MuharebAntje BlankGerd Mikus Original Research Article Open access 28 July 2023 Pages: 1305 - 1314
Significant Effects of Renal Function on Mycophenolic Acid Total Clearance in Pediatric Kidney Transplant Recipients with Population Pharmacokinetic Modeling Yan RongJenny WichartTony K. L. Kiang Original Research Article 26 July 2023 Pages: 1289 - 1303
Clinical Pharmacology of Brigatinib: A Next-Generation Anaplastic Lymphoma Kinase Inhibitor Neeraj GuptaMichael J. HanleyVikram Sinha Review Article Open access 26 July 2023 Pages: 1063 - 1079
Status and Quality of Guidelines for Therapeutic Drug Monitoring Based on AGREE II Instrument Zhan-Miao YiXinya LiRongsheng Zhao Systematic Review 25 July 2023 Pages: 1201 - 1217
Clinical Pharmacokinetics and Pharmacodynamics of the Next Generation Androgen Receptor Inhibitor—Darolutamide Eva PodgoršekNiven MehraNielka P. van Erp Review Article Open access 17 July 2023 Pages: 1049 - 1061
Population Target-Mediated Pharmacokinetic/Pharmacodynamic Modeling to Evaluate SPI-62 Exposure and Hepatic 11β-Hydroxysteroid Dehydrogenase Type 1 (HSD-1) Inhibition in Healthy Adults Nan WuDavid A. KatzGuohua An Original Research Article Open access 15 July 2023 Pages: 1275 - 1288
Relationship Between Cetuximab Target-Mediated Pharmacokinetics and Progression-Free Survival in Metastatic Colorectal Cancer Patients Sarah LobetGilles PaintaudDavid Ternant Original Research Article 13 July 2023 Pages: 1263 - 1274
Population Pharmacokinetic Model of Intravenous Busulfan in Hematopoietic Cell Transplantation: Systematic Review and Comparative Simulations Takuto TakahashiMutaz M. JaberMahmoud Al-Kofahi Systematic Review 06 July 2023 Pages: 955 - 968