Healthcare Systems and Artificial Intelligence: Focus on Challenges and the International Regulatory Framework Alessia RomagnoliFrancesco FerraraAndrea Zovi Perspectives 05 March 2024 Pages: 721 - 730
An Evaluation of Wet Granulation Process Selection for API Prone to Polymorphic Form Conversion in the Presence of Moisture and Heat Freddy ArceYue SchumanDivyakant Desai Original Research Article 21 February 2024 Pages: 595 - 607
Acetylcholine Analog-Modified Albumin Nanoparticles for the Enhanced and Synchronous Brain Delivery of Saponin Components of Panax Notoginseng Ying YuLi Yun WangCheng Xiao Wang Original Research Article 21 February 2024 Pages: 513 - 529
Research Landscape of Physiologically Based Pharmacokinetic Model Utilization in Different Fields: A Bibliometric Analysis (1999–2023) Xin WangJiangfan WuShenyin Zhu Original Research Article 21 February 2024 Pages: 609 - 622
Antibody-Drug Conjugate Overview: a State-of-the-art Manufacturing Process and Control Strategy Meng LiXueyu ZhaoLan Wang Review Article 17 February 2024 Pages: 419 - 440
Co-delivery of Brinzolamide and Timolol from Micelles-laden Contact Lenses: In vitro and In Vivo Evaluation Hongyu YangFaxing ZhangJi Li Original Research Article 16 February 2024 Pages: 531 - 546
Convolutional Neural Networks Guided Raman Spectroscopy as a Process Analytical Technology (PAT) Tool for Monitoring and Simultaneous Prediction of Monoclonal Antibody Charge Variants Nitika NitikaB. KeerthiveenaAnurag S. Rathore Original Research Article 16 February 2024 Pages: 463 - 479
Medicinal Polypharmacology in the Clinic – Translating the Polypharmacolome into Therapeutic Benefit Muhammad RafehiMarius MöllerSven Marcel Stefan Perspectives Open access 16 February 2024 Pages: 411 - 417
In Silico Study on the Contribution of the Follicular Route to Dermal Permeability of Small Molecules Daniel Sebastia-SaezGuoping LianTao Chen Original Research Article Open access 13 February 2024 Pages: 567 - 576
Physiologically Based Pharmacokinetic (PBPK) Model Predictions of Disease Mediated Changes in Drug Disposition in Patients with Nonalcoholic Fatty Liver Disease (NAFLD) Jeffry AdiwidjajaJessica SpiresKim L. R. Brouwer Original Research Article 13 February 2024 Pages: 441 - 462
Monte Carlo Optimization Method Based QSAR Modeling of Placental Barrier Permeability Predrag VukomanovićMilan StefanovićAleksandar M. Veselinović Original Research Article 09 February 2024 Pages: 493 - 500
Progress in the Application of Microneedles in Eye Disorders and the Proposal of the Upgraded Microneedle with Spinule Qiannan YangTingting ZhangXin Jin Review Article 09 February 2024 Pages: 203 - 222
Structure Based Machine Learning Prediction of Retention Times for LC Method Development of Pharmaceuticals Jonathan FineAmanda K. Peterson MannPankaj Aggarwal Original Research Article 08 February 2024 Pages: 365 - 374
Intradermal Vaccination with PLGA Nanoparticles via Dissolving Microneedles and Classical Injection Needles Jihui LeeMalene A. NeustrupKoen van der Maaden Original Research Article Open access 08 February 2024 Pages: 305 - 319
Unraveling Pre-filled Syringe Needle Clogging: Exploring a Fresh Outlook Through Innovative Techniques Guangli HuDaniel BonannoVladimir Novak Original Research Article 07 February 2024 Pages: 547 - 556
Characterization of mRNA Lipid Nanoparticles by Electron Density Mapping Reconstruction: X-ray Scattering with Density from Solution Scattering (DENSS) Algorithm Huy M. DaoKhaled AboulFotouhRobert O. Williams III Original Research Article 07 February 2024 Pages: 501 - 512
Green Tea Catechins Decrease Solubility of Raloxifene In Vitro and Its Systemic Exposure in Mice Victoria O. OyannaBaron J. BechtoldJohn D. Clarke Original Research Article 01 February 2024 Pages: 557 - 566
Novel Pharmaceutical Cocrystals of Tegafur: Synthesis, Performance, and Theoretical Studies Haoran MeiNa WangHongxun Hao Original Research Article 30 January 2024 Pages: 577 - 593
The Effects of Excipients on Freeze-dried Monoclonal Antibody Formulation Degradation and Sub-Visible Particle Formation during Shaking Meng-Jia JinXin-Zhe GeWei-Jie Fang Original Research Article 30 January 2024 Pages: 321 - 334
Coupling Drug Dissolution with BCS Antony SimitopoulosAthanasios TsekourasPanos Macheras Original Research Article Open access 30 January 2024 Pages: 481 - 491
WANTED DEAD OR ALIVE: New Thinking to Incentivize Drug Development Michael S. Kinch Perspective 30 January 2024 Pages: 199 - 202
Keratinocyte Exosomes for Topical Delivery of Tofacitinib in Treatment of Psoriasis: an In Vitro/ In Vivo Study in Animal Model of Psoriasis Pouya DehghaniJaleh VarshosazMahdi Bodaghi Original Research Article Open access 23 January 2024 Pages: 263 - 279
Correction: Comparative Study of Dermal Pharmacokinetics Between Topical Drugs Using Open Flow Microperfusion in a Pig Model Manfred BodenlenzThean YeohThomas Birngruber Correction Open access 19 January 2024 Pages: 409 - 409
Time-Lapse Macro Imaging with Dissolution Tests for Exploring the Interrelationship Between Disintegration and Dissolution Behaviors of Solid Dosages Yichen YangJiajia GengjiLi Deng Original Research Article 19 January 2024 Pages: 387 - 400
Development of an Accelerated Rotator-based Drug Release Method for the Evaluation of Bupivacaine Multivesicular Liposomes Ziyun XiaMinzhi YuAnna Schwendeman Original Research Article 11 January 2024 Pages: 293 - 303
IVIVC Revised Nikolaos AlimpertisAntony SimitopoulosPanos Macheras Original Research Article 08 January 2024 Pages: 235 - 246
The Osmolality and Hemolysis of High-Concentration Monoclonal Antibody Formulations Meng-Juan PangMeng-Wen WangWei-Jie Fang Original Research Article 03 January 2024 Pages: 281 - 291
Correction: Effect of Buffer Salts on Physical Stability of Lyophilized and Spray-Dried Protein Formulations Containing Bovine Serum Albumin and Trehalose Tarun Tejasvi MutukuriJing LingQi Tony Zhou Correction 29 December 2023 Pages: 405 - 406
Comparative Study of Dermal Pharmacokinetics Between Topical Drugs Using Open Flow Microperfusion in a Pig Model Manfred BodenlenzThean YeohThomas Birngruber Original Research Article Open access 29 December 2023 Pages: 223 - 234
Retraction Note: Dual Blockade of PD-1 and LAG3 Immune Checkpoints Increases Dendritic Cell Vaccine Mediated T Cell Responses in Breast Cancer Model Asal BarshidiVahid KarpishehFarhad Jadidi-Niaragh Retraction Note 26 December 2023 Pages: 407 - 408
An In Silico Platform to Predict Cardiotoxicity Risk of Anti-tumor Drug Combination with hiPSC-CMs Based In Vitro Study Lan SangZhengying ZhouKun Hao Original Research Article Open access 26 December 2023 Pages: 247 - 262
Impact of Formulation and Microneedle Length on Transdermal Metronidazole Permeation through Microneedle-Treated Skin Krishna Kumar PatelNicole K. Brogden Original Research Article 22 December 2023 Pages: 355 - 363
Editorial: Improving Product Quality through Process and Materials Understanding Peter L. D. WildfongRahul V. HawareDavid A. Engers Preface 22 December 2023 Pages: 2759 - 2760
Application of PAT Probes in Aluminum Phosphate Adjuvant Manufacturing Przemyslaw KowalGinny FungMarina Kirkitadze Original Research Article 19 December 2023 Pages: 375 - 385
Exploiting Apical Sodium-Dependent Bile Acid Transporter (ASBT)-Mediated Endocytosis with Multi-Functional Deoxycholic Acid Grafted Alginate Amide Nanoparticles as an Oral Insulin Delivery System Maryam RazmjooeiSeyed Mohammad Hashem HosseiniMohammad Hadi Eskandari Original Research Article 19 December 2023 Pages: 335 - 353
PBPK/PD Modeling of Nifedipine for Precision Medicine in Pregnant Women: Enhancing Clinical Decision-Making for Optimal Drug Therapy Xinyang LiuWei WangDefang Ouyang Original Research Article 04 December 2023 Pages: 63 - 75
Impact of Processing Methods on the Physico-chemical Properties of Posaconazole Amorphous Solid Dispersions Ru HeMatthew S. LammYongjun Li Original Research Article 01 December 2023 Pages: 141 - 151
Professor David E. Smith: A Fearless Scientist and Devoted Mentor Brian ThompsonKim BrouwerMaria M. Posada EditorialNotes 29 November 2023 Pages: 2493 - 2497
General Commentary: A Tribute to Professor Kenneth R. Morris – Scientist, Teacher, Mentor, Friend…and Underappreciated Academic Arborist Peter L. D. Wildfong Tribute 28 November 2023 Pages: 2761 - 2767
Comparative Study of Sorption Phenomena Between Three Medications and Syringes Made of Cyclic Olefin Copolymer or Polypropylene Joëlle ClavesPhilip ChennellValérie Sautou Original Research Article 21 November 2023 Pages: 51 - 62
AgNPs-Modified Polylactic Acid Microneedles: Preparation and In Vivo/In Vitro Antimicrobial Studies Wenqin ZhangXiaozhen CaiJianmin Chen Original Research Article 20 November 2023 Pages: 93 - 104
Elucidating the Impact of Material Properties on Tablet Manufacturability for Binary Paracetamol Blends Lena MareczekCarolin RiehlStephan Reichl Original Research Article 17 November 2023 Pages: 185 - 197
Development of Sustained Release System Based on High Water-Absorbable Gel Formation Using Croscarmellose Sodium, Alkaline Excipients and HPMC (ACSH SR System); Novel Application of Croscarmellose Sodium as a Gel Former Masato GomiNaoya MizutaniKazutaka Higaki Original Research Article 14 November 2023 Pages: 3073 - 3086
LC–MS Approach to Decipher a Light Chain Chromatographic Peak Splitting of a Monoclonal Antibody Yanjun LiuZac VanAernumJennifer S. Chadwick Original Research Article 07 November 2023 Pages: 3087 - 3098
Use of Resonant Acoustic Mixing Technology for Ultra-Low-Dose Blending in a Single-Step Mixing Process Kyle A. FreyHelen BakerDavid A. Engers Original Research Article 07 November 2023 Pages: 165 - 183
Fabrication and Characterization of Dissolving Microneedles for Transdermal Drug Delivery of Apomorphine Hydrochloride in Parkinson’s Disease Daisuke AndoAisa OzawaKen-ichi Izutsu Original Research Article 03 November 2023 Pages: 153 - 163
Pharmaceutical and Immunological Evaluation of Cholera Toxin A1 Subunit as an Adjuvant of Hepatitis B Vaccine Microneedles Jong-Chan KimJung-ah ChoiJung-Hwan Park Original Research Article 01 November 2023 Pages: 3059 - 3071
A Stable Irinotecan Liposome with Enhanced Antitumor Activity in a Range of Tumor Models Zhengxing SuLi LiDong Zhao Original Research Article 01 November 2023 Pages: 3043 - 3058
Integrated Exposure–Response of Dupilumab in Children, Adolescents, and Adults With Atopic Dermatitis Using Categorical and Continuous Efficacy Assessments: A Population Analysis Emily BriggsMohamed A. KamalNidal Huniti Original Research Article Open access 11 December 2023 Pages: 2653 - 2666