One-pot organocatalytic/multicomponent approach for the preparation of novel enantioenriched non-natural selenium-based peptoids and peptide–peptoid conjugates Alexander F. de la TorreAkbar AliMárcio W. Paixão Original Article 18 February 2019 Pages: 1 - 10
Substituent effect on inter-ring interaction in paracyclophanes Irena MajerzTeresa Dziembowska Original Article Open access 19 February 2019 Pages: 11 - 20
Lupenone is a good anti-inflammatory compound based on the network pharmacology Feng XuLiubo YangHongmei Wu Original Article 22 February 2019 Pages: 21 - 30
The periodic table of urea derivative: small molecules of zinc(II) and nickel(II) of diverse antimicrobial and antiproliferative applications Christina N. BantiMehmet PoyrazSotiris K. Hadjikakou Original Article 23 February 2019 Pages: 31 - 43
Combining ligand- and structure-based in silico methods for the identification of natural product-based inhibitors of Akt1 Priya MahajanBhumika WadhwaAmit Nargotra Original Article 23 February 2019 Pages: 45 - 60
Single-stage synthesis of heterocyclic alkaloid-like compounds from (+)-camphoric acid and their antiviral activity Vladimir V. ChernyshovOlga I. YarovayaNariman F. Salakhutdinov Original Article 28 February 2019 Pages: 61 - 67
Design and synthesis of new imidazo[1,2-b]pyrazole derivatives, in vitro α-glucosidase inhibition, kinetic and docking studies Fariba PeytamMehdi AdibBagher Larijani Original Article 02 March 2019 Pages: 69 - 80
Four-component green synthesis of benzochromene derivatives using nano-KF/clinoptilolite as basic catalyst: study of antioxidant activity Elham EzzatzadehZinatossadat Hossaini Original Article 04 March 2019 Pages: 81 - 91
A quick accelerating microwave-assisted sustainable technique: permutated spiro-casing for imaging experiment Animesh MondalBarnali NaskarChhanda Mukhopadhyay Original Article 06 March 2019 Pages: 93 - 106
Regioselective synthesis of pyrimidine-fused tetrahydropyridines and pyridines by microwave-assisted one-pot reaction Pooja KumariRahul YadavTasneem Parvin Original Article 07 March 2019 Pages: 107 - 117
Synthesis and plant growth regulatory activities of 2′,3′-PhABA and iso-2′,3′-PhABA esters Chuan WanJiaqi LiZhaohai Qin Original Article 09 March 2019 Pages: 119 - 130
Iodine/potassium iodide catalyst for the synthesis of trifluoromethylated quinazolines via intramolecular cyclization of 2,2,2-trifluoro-N-benzyl-N′-arylacetimidamides Ali DarehkordiElham Kazemi Original Article 13 March 2019 Pages: 131 - 139
Two- and three-dimensional QSAR studies on hURAT1 inhibitors with flexible linkers: topomer CoMFA and HQSAR Tingting ZhaoZean ZhaoYuanxin Tian Original Article 13 March 2019 Pages: 141 - 154
Synthesis and process optimization of symmetric and unsymmetric barbiturates C5-coupled with 2,1-benzisoxazoles João L. SerranoPedro F. SoeiroPaulo Almeida Original Article 14 March 2019 Pages: 155 - 166
Application of 2,4-bis(halomethyl)quinoline: synthesis and biological activities of 2,4-bis(benzofuran-2-yl)- and 2,4-bis(aroxymethyl)quinolines Yang LiQiqi XuYu Chen Original Article 20 March 2019 Pages: 167 - 178
Novel fused 1,2,3-triazolo-benzodiazepine derivatives as potent anticonvulsant agents: design, synthesis, in vivo, and in silico evaluations Arefeh ShafieMaryam Mohammadi-KhanaposhtaniAhmad Reza Dehpour Original Article 20 March 2019 Pages: 179 - 189
DBU-mediated annulation of 2-aryl-3-nitro-2H-chromenes with 1,3-cyclohexanediones for the synthesis of benzofuro[2,3-c]chromenone derivatives Chenlu DaiZengyang XieCunde Wang Original Article 23 March 2019 Pages: 191 - 200
Preparation and characterization of a novel spherical cellulose–copper(II) oxide composite particles: as a heterogeneous catalyst for the click reaction Seyedeh Fazileh HamzaviSanaz GerivaniGholamhossein Shahverdizadeh Original Article 26 March 2019 Pages: 201 - 209
Design, synthesis, in vivo and in vitro studies of 1,2,3,4-tetrahydro-9H-carbazole derivatives, highly selective and potent butyrylcholinesterase inhibitors Roshanak GhobadianRoghaieh EsfandyariMohsen Amini Original Article 29 March 2019 Pages: 211 - 223
A novel protocol for catalyst-free synthesis of fused six-member rings to triazole and pyrazole Sedigheh AkramiBahador KaramiMahnaz Farahi Original Article 01 April 2019 Pages: 225 - 231
Identification of pyrrolo-pyridine derivatives as novel class of antibacterials Mark S. VeselovYan A. IvanenkovOlga A. Dontsova Original Article 04 April 2019 Pages: 233 - 239
Facile, efficient and one-pot access to diverse new functionalized aminoalkyl and amidoalkyl naphthol scaffolds via green multicomponent reaction using triethylammonium hydrogen sulfate ([Et3NH][HSO4]) as an acidic ionic liquid under solvent-free conditions Elahe HadadianpourBehjat Pouramiri Original Article 05 April 2019 Pages: 241 - 252
Adamantyl pyran-4-one derivatives and their in vitro antiproliferative activity Vesna Petrović PerokovićŽeljka CarSrđanka Tomić Original Article 05 April 2019 Pages: 253 - 263
Synthesis, anti-proliferative activity, theoretical and 1H NMR experimental studies of Morita–Baylis–Hillman adducts from isatin derivatives Vinicius B. M. BritoGilmar F. SantosEdilson B. Alencar-Filho Original Article 06 April 2019 Pages: 265 - 281
Amine-functionalized graphene oxide nanosheets (AFGONs): an efficient bifunctional catalyst for selective formation of 1,4-dihydropyridines, acridinediones and polyhydroquinolines Prasun ChoudhuryPranab GhoshBasudeb Basu Short Communication 06 April 2019 Pages: 283 - 294
5-Endo-dig cyclizations in organic syntheses Muhammad Aamir SajidZulfiqar Ali KhanMuhammad Usman Comprehensive Review 05 March 2019 Pages: 295 - 317