1. Medicinal chemistry insights into non-hydroxamate HDAC6 selective inhibitors

   • Faridoon
   • Yuqi Lavender Zha
   • Jie Jack Li

   Review Article 31 October 2022 Pages: 1 - 14

   

2. A study from structural insight to the antiamyloidogenic and antioxidant activities of flavonoids: scaffold for future therapeutics of Alzheimer’s disease

   • Madhu Sudan Dutta

   Review Article 09 November 2022 Pages: 15 - 31

   

3. Optimization of the dipeptide motifs in the PSMA ligands linker structure: synthesis and in vitro evaluation

   • Anastasiia A. Uspenskaya
   • Ekaterina A. Nimenko
   • Aleksei E. Machulkin

   Brief Report 21 December 2022 Pages: 32 - 37

   

4. Optimization of clofibrate with natural product sesamol for reducing liver injury induced by acetaminophen

   • Chuchu Han
   • Linyang Zhang
   • Ying Liu

   Original Research 01 November 2022 Pages: 38 - 46

   

5. Synthesis and in vitro antimicrobial evaluation of benzothiazolylindenopyrazoles

   • Satbir Mor
   • Mohini Khatri
   • Komal Jakhar

   Original Research 01 November 2022 Pages: 47 - 56

   

6. Novel Curcumin Monocarbonyl Analogue-Dithiocarbamate hybrid molecules target human DNA ligase I and show improved activity against colon cancer

   • Deependra K. Singh
   • Dhanaraju Mandalapu
   • Dibyendu Banerjee

   Original Research 05 November 2022 Pages: 57 - 75

   

7. Synthesis of myricetin derivatives and evaluation of their hypoglycemic activities

   • Feng Li
   • Chong Yang
   • Wenbao Li

   Original Research 10 November 2022 Pages: 76 - 84

   

8. Synthesis, antimicrobial, and antioxidant activities of disubstituted 1,2,3-triazoles with amide-hydroxyl functionality

   • Manisha Chahal
   • Chander Prakash Kaushik
   • Ashwani Kumar

   Original Research 17 November 2022 Pages: 85 - 98

   

9. Design, synthesis and anticancer activity studies of novel indole derivatives as Bcl-2/Mcl-1 dual inhibitors

   • Yingfei Liu
   • Jianjun Li
   • Tingting Liu

   Original Research 18 November 2022 Pages: 99 - 108

   

10. Design, synthesis, and biological evaluation of 2, 4-dichlorophenoxyacetamide chalcone hybrids as potential c-Met kinase inhibitors

    • Heena Bhojwani
    • Sanskruti Patil
    • Parul Bedi

    Original Research 24 November 2022 Pages: 109 - 127

    

11. Synthesis, pharmacological and molecular docking investigations of 1,3,4-oxadiazole-5-thionyl derivatives of extracted cis-clerodane diterpenoid from Cistus monspeliensis

    • Fatima I. Mahi
    • Mohammed A. Mehdid
    • Rachid Chahboun

    Original Research 01 December 2022 Pages: 128 - 143

    

12. Synthesis and cytotoxic/antimicrobial screening of 2-alkenylimidazo[1,2-a]pyrimidines

    • Ángel Ramírez-Trinidad
    • Karol Carrillo-Jaimes
    • Eduardo Hernández-Vázquez

    Original Research 09 December 2022 Pages: 144 - 157

    

13. 1,2,3-triazenes and 1,2,3-triazoles as antileishmanial, antitrypanosomal, and antiplasmodial agents

    • Insa Seck
    • Ismaïla Ciss
    • Matar Seck

    Original Research 10 December 2022 Pages: 158 - 164

    

14. Dipeptidyl Peptidase-IV Blockers Potently Inhibit Monoglyceride Lipase: Investigation By Docking Studies And In Vitro Bioassay

    • Dania Alkabbani
    • Lina A. Dahabiyeh
    • Mutasem O. Taha

    Original Research 14 December 2022 Pages: 165 - 175

    

15. 2,3-Diketopiperazine as potential scaffold to develop new anti-Chagasic agents

    • Urbano Osorio-Nieto
    • Cristian O. Salas
    • Christian Espinosa-Bustos

    Original Research 16 December 2022 Pages: 176 - 188

    

16. Tetra-substituted pyrazole analogues: synthesis, molecular docking, ADMET prediction, antioxidant and pancreatic lipase inhibitory activities

    • Adnan Cetin
    • Ali Donmez
    • Ishak Bildirici

    Original Research 22 December 2022 Pages: 189 - 204