1. Phosphoryl prodrugs: characteristics to improve drug development

   • Samuel A. Kirby
   • Cynthia S. Dowd

   Review Article 23 July 2021 Pages: 207 - 216

   

2. A novel sight of the primary active compounds from Umbelliferae: focusing on mitochondria

   • Luping Yang
   • Ni Ni
   • Lan Shen

   Review Article 03 January 2022 Pages: 217 - 231

   

3. Review on molnupiravir as a promising oral drug for the treatment of COVID-19

   • Elham Zarenezhad
   • Mahrokh Marzi

   Review Article 03 January 2022 Pages: 232 - 243

   

4. Isatin derivatives as broad-spectrum antiviral agents: the current landscape

   • Tilal Elsaman
   • Malik Suliman Mohamed
   • Magdi Awadalla Mohamed

   Review Article 13 January 2022 Pages: 244 - 273

   

5. Design and discovery of a high affinity, selective and β-arrestin biased 5-HT₇ receptor agonist

   • Edem K. Onyameh
   • Edward Ofori
   • Seth Y. Ablordeppey

   Original Research 23 September 2021 Pages: 274 - 283

   

6. Antimicrobial action of arylsulfonamides bearing (aza)norbornane and related motifs: evaluation of new promising anti-MRSA agents

   • Vitalii Palchykov
   • Nazar Manko
   • Nazariy Pokhodylo

   Original Research 06 January 2022 Pages: 284 - 292

   

7. Structure related α-glucosidase inhibitory activity and molecular docking analyses of phenolic compounds from Paeonia suffruticosa

   • Po-Chun Chen
   • Bongani Sicelo Dlamini
   • Chi-I Chang

   Original Research 07 January 2022 Pages: 293 - 306

   

8. Design and synthesis of potential fungicidal compounds derived from natural products, (-)-menthol and (-)-borneol

   • Tianyuan Zhang
   • Shumin Zheng
   • Yong-Xian Cheng

   Original Research 07 January 2022 Pages: 307 - 315

   

9. Design, synthesis, in vitro evaluation, and docking studies on ibuprofen derived 1,3,4-oxadiazole derivatives as dual α-glucosidase and urease inhibitors

   • Saima Daud
   • Obaid-ur-Rahman Abid
   • Basit Niaz

   Original Research 08 January 2022 Pages: 316 - 336

   

10. Synthesis and evaluation of novel, selective, functionalized γ-butyrolactones as sigma-2 ligands

    • Benjamin E. Blass
    • Rong Gao
    • Daniel J. Canney

    Original Research 10 January 2022 Pages: 337 - 349

    

11. Synthesis and biological evaluation of (20S,24R)-epoxy-dammarane-3β,12β,25-triol derivatives as α-glucosidase and PTP1B inhibitors

    • Xiao-Tong Yang
    • Tian-Ze Li
    • Ji-Jun Chen

    Original Research 11 January 2022 Pages: 350 - 367

    

12. Synthesis and anticancer activity of novel hydrazone linkage-based aryl sulfonate derivatives as apoptosis inducers

    • Sevil Şenkardeş
    • M. İhsan Han
    • Ş. Güniz Küçükgüzel

    Original Research 12 January 2022 Pages: 368 - 379

    

13. Correction to: Design, synthesis and SAR of novel sulfonylurea derivatives for the treatment of diabetes mellitus in rats

    • Farid M. Sroor
    • Wahid M. Basyouni
    • Azza F. Arafa

    Correction 24 December 2021 Pages: 380 - 382