Collection
Anti-HIV activity
The following articles were selected by the editors as some of the best research recently published in Medicinal Chemistry Research on anti-HIV activity. This list is current to 1 October, 2023.
Articles (39 in this collection)
-
-
Isatin derivatives as broad-spectrum antiviral agents: the current landscape
Authors (first, second and last of 7)
-
Design, synthesis, in vitro evaluation, and docking studies on ibuprofen derived 1,3,4-oxadiazole derivatives as dual α-glucosidase and urease inhibitors
Authors (first, second and last of 13)
-
-
Synthesis and biological evaluation of pyrrolidine-functionalized nucleoside analogs
Authors (first, second and last of 8)
-
Phosphoramidate conjugates of 3′-azido-3′-deoxythymidine glycerolipid derivatives and amino acid esters: synthesis and anti-HIV activity
Authors (first, second and last of 5)
-
Microwave-assisted synthesis, molecular docking and anti-HIV activities of some drug-like quinolone derivatives
Authors (first, second and last of 4)
-
Synthesis and evaluation of antiviral activities of triterpenic conjugates with 2-aminobutan-1-ol as potent microbicidal agents
Authors (first, second and last of 6)
-
-
Combined topomer CoMFA and hologram QSAR studies of a series of pyrrole derivatives as potential HIV fusion inhibitors
Authors (first, second and last of 6)
-
Synthesis, crystal structure, anti-HIV, and antiproliferative activity of new pyrazolylthiazole derivatives
Authors (first, second and last of 6)
-
Ethyl phosphoramidates of acyclovir: design, synthesis, molecular docking (HN Protein), and evaluation of antiviral and antioxidant activities
Authors (first, second and last of 7)
-
Amino acid derivatives. Part 6. Synthesis, in vitro antiviral activity and molecular docking study of new N-α-amino acid derivatives conjugated spacer phthalimide backbone
Authors (first, second and last of 5)
-
Synthesis, crystal structure, anti-HIV, and antiproliferative activity of new oxadiazole and thiazole analogs
Authors (first, second and last of 7)
-
Synthesis of some new 2-amino-6-thiocyanato benzothiazole derivatives bearing 2,4-thiazolidinediones and screening of their in vitro antimicrobial, antitubercular and antiviral activities
Authors (first, second and last of 6)
-
Structural findings of quinolone carboxylic acids in cytotoxic, antiviral, and anti-HIV-1 integrase activity through validated comparative molecular modeling studies
Authors (first, second and last of 4)
-
Synthesis, molecular docking and antiviral screening of novel N′-substitutedbenzylidene-2-(4-methyl-5,5-dioxido-3-phenylbenzo[e]pyrazolo[4,3-c][1,2]thiazin-1(4H)-yl)acetohydrazides
Authors (first, second and last of 9)
-
Quantitative structure–activity relationship studies of diarylpyrimidine derivatives as anti-HIV drugs using new three-dimensional structure descriptors
Authors (first, second and last of 5)
-
Design, synthesis, and antiviral activity of new 1H-1,2,3-triazole nucleoside ribavirin analogs
Authors (first, second and last of 9)
-
Synthesis of novel biologically active methylene derivatives of sydnones
Authors (first, second and last of 5)
-
Syntheses and in vitro biological screening of 1-aryl-10H-[1,2,4]triazolo[3′,4′:3,4][1,2,4]triazino[5,6-b]indoles
Authors (first, second and last of 8)
-
Tautomeric origin of dual effects of N1-nicotinoyl-3-(4′-hydroxy-3′-methyl phenyl)-5-[(sub)phenyl]-2-pyrazolines on bacterial and viral strains: POM analyses as new efficient bioinformatics’ platform to predict and optimize bioactivity of drugs
Authors (first, second and last of 6)
-
Computational evaluation and experimental in vitro antibacterial, antifungal and antiviral activity of bis-Schiff bases of isatin and its derivatives
Authors (first, second and last of 5)
-
Molecular docking, QPLD, and ADME prediction studies on HIV-1 integrase leads
Authors (first, second and last of 4)
-
-
Synthesis, antimycobacterial, antiviral, antimicrobial activities, and QSAR studies of isonicotinic acid-1-(substituted phenyl)-ethylidene/cycloheptylidene hydrazides
Authors (first, second and last of 8)
-
Isonicotinic acid hydrazide derivatives: synthesis, antimicrobial activity, and QSAR studies
Authors (first, second and last of 8)
-
Synthesis and antiviral activity of benzimidazolyl- and triazolyl-1,3,5-triazines
Authors (first, second and last of 4)
-
-
-
Biological evaluation of novel 1,4-dithiine derivatives as potential antimicrobial agents
Authors (first, second and last of 7)
-
Quantitative structure activity relationship (QSAR) studies of a series of 2,5-disubstituted-1,3,4-oxadiazole derivatives as biologically potential compounds
Authors (first, second and last of 4)
-
Screening and evaluation of thiourea derivatives for their HIV capsid and human cyclophilin A inhibitory activity
Authors (first, second and last of 8)
-
Modification and biological evaluation of novel 4-hydroxy-pyrone derivatives as non-peptidic HIV-1 protease inhibitors
Authors (first, second and last of 5)
-
-
Synthesis and anti-HIV activity evaluation of novel N′-arylidene-2-[1-(naphthalen-1-yl)-1H-tetrazol-5-ylthio]acetohydrazides
Authors (first, second and last of 7)
-
Synthesis of some novel 2-substituted benzoxazoles as anticancer, antifungal, and antimicrobial agents
Authors (first, second and last of 5)
-
-
