A New Approach to the Synthesis of Anti-Reverse Cap Analog (ARCA) 2mGpppG A. L. KayushinK. V. AntonovI. D. Konstantinova OriginalPaper 13 February 2024 Pages: 1 - 7
Pyrazinamide Analogs Designed for Rational Drug Designing Strategies Against Resistant Tuberculosis (A Review) Xinyu WangHongshang HuJuan Xu ReviewPaper 13 February 2024 Pages: 8 - 27
Synthesis, Characterization, and Study of Anticancer Activities of New Schiff Bases and 1,3-Oxazepine Containing Drug Rana Abid AliLuma S. AhamedShaima Ibraheem Chyad AL-Khazraji OriginalPaper 13 February 2024 Pages: 28 - 33
Synthesis of Novel 2-((3-(Benzofuran-2-yl)-1-phenyl-1H-pyrazol-4-yl)methylene)hydrazinyl-4-phenylthiazole: Potent EGFR Targeting Anticancer Agents Sateesh AmudalaRambabu PalabindelaJyothi Mandala OriginalPaper 13 February 2024 Pages: 34 - 44
Surfactants as a Means of Delivering a Reporter Genetic Construct Based on Binase Suicide Gene to Tumor Cells E. V. DudkinaE. A. VasilievaO. N. Ilinskaya OriginalPaper 13 February 2024 Pages: 45 - 55
Participation of the Transcription Factor CREB1 in the Regulation of the Mdh2 Gene Encoding Malate Dehydrogenase in the Liver of Rats with Alloxan-Induced Diabetes A. T. EprintsevK. R. RomanenkoN. V. Selivanova OriginalPaper 13 February 2024 Pages: 56 - 63
Assessing the Potential of Vitamin Drug Conjugate for Its Activity against Infectious Disease R. P. BholeP. C. BhondaveR. V. Chikhale OriginalPaper 13 February 2024 Pages: 64 - 75
Synthesis of Novel N-Acylhydrazones Derived from 3,5-Dinitrobenzohydrazide and Evaluation of Their Anticholinesterase and Antioxidant Activities Reşit ÇakmakErcan ÇınarMehmet Boğa OriginalPaper 13 February 2024 Pages: 76 - 85
Synthesis, Characterization of Formazan Derivatives from Isoniazid and Study Their Antioxidant Activity and Molecular Docking W. K. DamdoomO. H. R. Al-Jeilawi OriginalPaper 13 February 2024 Pages: 86 - 94
Isolation, Physico-Chemical Characteristics, and Acute Toxicity Evaluation of Water-Soluble Polysaccharide from Basidial Raw Material Ganoderma lucidum S. B. KhaytmetovaA. S. TuraevB. I. Muhitdinov OriginalPaper 13 February 2024 Pages: 95 - 105
Tetrahedral Boronate Ester as Regulators of Inflammation and Adhesion in ox-LDL Induced Atherosclerotic Model U. DegirmenciA. KilicM. Yildirim OriginalPaper 13 February 2024 Pages: 106 - 115
Synthesis of Steroid Tracers by an Oxime Ligation Method and Their Use in Fluorescent Polarisation Immunoassay I. A. ProkhorenkoD. A. GlushchenkoS. A. Eremin OriginalPaper 13 February 2024 Pages: 116 - 127
Benzothiophene Schiff Bases Disrupt Cytoplasmic Membrane Integrity of Gram-Positive and -Negative Bacteria Cells Bengü ErgüdenHatice Büşra LüleciYasemin Ünver OriginalPaper 13 February 2024 Pages: 128 - 137
Synthesis, Spectral Identification of Some New Schiff Bases, and Evaluation of Their Antibacterial Activity and Inhibitory Effect on Proinflammatory Cytokines (IL-1β, TNF), and DNA Ligase Israa A. Alhasan HamdanAlaa Abd Alhasan HamdanRasha A. Abidalmutalib Aljabawi OriginalPaper 13 February 2024 Pages: 138 - 146
Synthesis and Anti-Mycobacterium Activity of Some New N-Rich Heterocyclic Derivatives and Their Molecular Docking, and DFT Studies Raghavendra HegdeItte PushpavathiS. Ravi Kumar OriginalPaper 13 February 2024 Pages: 147 - 161
Design and Synthesis of Benzo-Spirocyclic Derivatives as Potent PARP-1 Inhibitors Shu JiaLing YuXin He OriginalPaper 13 February 2024 Pages: 162 - 169
Synthesis, Identification, Antioxidant, Molecular Docking, and In Silico ADME Study for Some New Derivatives Containing Thiourea Moiety Asmaa Abdulbaqi MaryooshOday H. R. Al-Jeilawi OriginalPaper 13 February 2024 Pages: 170 - 180
Synthesis of Chromeno[2,3-d]pyrimidine-2,4(3H)-dion Derivatives Fused with Indole Moiety as Potent Biological Agents P. V. NavaneethgowdaY. D. BodkeN. B. Nippu OriginalPaper 13 February 2024 Pages: 181 - 190
Synthesis and Biological Evaluation of Coumarin-Amino Acid-Benzotriazole Conjugates Emre MenteşeNedime ÇalışkanGülay Akyüz OriginalPaper 13 February 2024 Pages: 191 - 200
New Coumarin-Metronidazole Composites: Synthesis, Biocompatibility, and Anti-anaerobic Bacterial Activity Yasser Fakri Mustafa OriginalPaper 13 February 2024 Pages: 201 - 210
Acetylcholine Inhibitory Study of Novel Thio Linked Coumarin-Benzimidazole Derivatives: Design, Synthesis, Computational, and In Silico Molecular Docking Studies T. H. Maruthi NayakaItte PushpavathiY. R. Nagesh OriginalPaper 13 February 2024 Pages: 211 - 226
Novel Bipyrazole Targeting Dual CDK-2 and VEGFR-2 Kinases: Synthesis, Anticancer Evaluation, and In Silico Studies E. S. NossierN. M. KhalifaM. M. Ali OriginalPaper 13 February 2024 Pages: 227 - 238
Effective Microwave-Assisted Synthesis of 2-Chloro-5,6-dimethyl-3-(((substituted-benzylidene)hydrazono)methyl)-quinoline and Its Biological Assessment N. K. VegalT. D. BhattH. S. Joshi OriginalPaper 13 February 2024 Pages: 239 - 250
2,5-Dimethoxy-Benzylidene-Rhodanine and Its Acyclic Analogues as Selective Fluorogenic Dyes for Lipid Droplets of Living Cells S. A. KrasnovaYu. A. BogdanovaM. S. Baranov BriefCommunication 13 February 2024 Pages: 251 - 259
Aminocoumaranones as Chemiluminescence Indicators of the Urease Activity and Hydrogen Peroxide A. Yu. SmirnovN. S. BaleevaM. S. Baranov BriefCommunication 13 February 2024 Pages: 260 - 266
Aryliden-Imidazolones as Fluorogens of NanoLuc Protein E. R. ZaitsevaYu. A. BogdanovaM. S. Baranov BriefCommunication 13 February 2024 Pages: 267 - 272