Plate-based diversity subset screening generation 2: an improved paradigm for high-throughput screening of large compound files Andrew S. BellJoseph BradleyHongyao Zhu Original Article Open access 08 September 2016 Pages: 789 - 803
Design and synthesis of novel protein kinase R (PKR) inhibitors Sagiv WeintraubTali YarnitzkyArie Gruzman Original Article 01 August 2016 Pages: 805 - 819
Synthesis of new quinazolin-2,4-diones as anti-Leishmania mexicana agents Eduardo EncisoJuan I. Sarmiento-SánchezEvangelina Beltrán-López Original Article 16 August 2016 Pages: 821 - 828
Skeletal modifications of \(\upbeta \)-carboline alkaloids and their antiviral activity profile Yan YangYuanqiong HuangQingmin Wang Original Article 18 April 2016 Pages: 829 - 835
Substituted N-aminothioglycolurils containing thiosemicarbazone moiety and their cytotoxic activity in vitro Galina A. GazievaLada V. AnikinaAngelina N. Kravchenko Original Article 23 May 2016 Pages: 837 - 846
Cerium oxide-catalyzed multicomponent condensation approach to spirooxindoles in water Rajeev ShresthaKavita SharmaYoung-Jung Wee Original Article 02 May 2016 Pages: 847 - 858
Synthesis of isoindolin-1-one derivatives via multicomponent reactions of methyl 2-formylbenzoate and intramolecular amidation Jie LeiZhi-Gang XuZhong-Zhu Chen Original Article 07 June 2016 Pages: 859 - 865
Multicomponent synthesis of diverse pyrano-fused benzophenazines using bifunctional thiourea-based organocatalyst in aqueous medium Ruchi BhartiTasneem Parvin Original Article 17 June 2016 Pages: 867 - 876
Microbial diversification of Diels–Alder cycloadducts by whole cells of Penicillium brasilianum Zia Ud DinTaicia P. FillE. Rodrigues-Filho Original Article 01 June 2016 Pages: 877 - 885
Synthesis of pyrazolo[1,5-a]pyrimidine derivatives and their antifungal activities against phytopathogenic fungi in vitro Jin ZhangJu-Fang PengZun-Ting Zhang Original Article 07 September 2016 Pages: 887 - 896
Synthesis and antifungal activity of dehydroabietic acid-based 1,3,4-thiadiazole-thiazolidinone compounds Naiyuan ChenWengui DuanDianpeng Li Original Article 01 August 2016 Pages: 897 - 905
Facile and efficient approach for the synthesis of spirocyclopropylbarbiturates and 3-substituted-1,1,2,2-tetracyanocyclopropanes using N-halosulfonamides Ramin Ghorbani-VagheiYaser MaghbooliJafar Mahmoodi Original Article 13 June 2016 Pages: 907 - 917
Design, synthesis, insecticidal activity, and structure-activity relationship (SAR): studies of novel triazone derivatives containing a urea bridge group based on transient receptor potential (TRP) channels Yan YangYuxiu LiuQingmin Wang Original Article 06 July 2016 Pages: 919 - 932
Identification of potential ACAT-2 selective inhibitors using pharmacophore, SVM and SVR from Chinese herbs Lian-sheng QiaoXian-bao ZhangGong-yu Li Original Article 21 June 2016 Pages: 933 - 944
Computational predictive models for P-glycoprotein inhibition of in-house chalcone derivatives and drug-bank compounds Trieu-Du NgoThanh-Dao TranKhac-Minh Thai Original Article 18 July 2016 Pages: 945 - 961
A new synthesis of \(\varvec{S}\)-aryl uracils from aryl thiols and 6-amino uracils in the presence of NCS Gholamhossein Khalili Short Communication 05 July 2016 Pages: 963 - 968
Ring opening of epoxides with C-nucleophiles Sadia FaizAmeer Fawad Zahoor Comprehensive Review 04 July 2016 Pages: 969 - 987
Advancements in tetronic acid chemistry. Part 2: Use as a simple precursor to privileged heterocyclic motifs Moaz M. AbdouRasha A. El-SaeedJohn Boukouvalas Short Review 27 June 2016 Pages: 989 - 999