Volume 21, Issue 6

Search all Medicinal Chemistry Research articles

June 2012

30 articles in this issue

QSAR analysis on PfPK7 inhibitors using HQSAR, CoMFA, and CoMSIA
Thirumurthy Madhavan
Gugan Kothandan
Seung Joo Cho
Original Research 01 February 2011 Pages: 681 - 693
Synthesis, characterization and antimicrobial activity of 4-amino-1-alkyl pyridinium salts
A. Ilangovan
P. Venkatesan
R. Rajesh Kumar
Original Research 02 February 2011 Pages: 694 - 702
Synthesis and antiviral activity of benzimidazolyl- and triazolyl-1,3,5-triazines
Azza R. Maarouf
Abdelbasset A. Farahat
Hassan M. Eisa
Original Research 04 February 2011 Pages: 703 - 710
Part of 1 collection:

Anti-HIV activity
Synthesis of a ligand–quencher conjugate for the ligand binding study of the aryl hydrocarbon receptor using a FRET assay
Yu Wang
Dazhou Yang
Liang Xue
Original Research 04 February 2011 Pages: 711 - 721
Skimmianine, a furoquinoline alkaloid from Zanthoxylum nitidum as a potential acetylcholinesterase inhibitor
Zhong-duo Yang
Dong-bo Zhang
Ming-jun Yang
Original Research 04 February 2011 Pages: 722 - 725
Synthesis of new piperidyl indanone derivatives as anticonvulsant agents
Nadeem Siddiqui
M. Faiz Arshad
Sharique Ahmed
Original Research 04 February 2011 Pages: 726 - 733
Acetylcholinesterase inhibitory activity of the total alkaloid from traditional Chinese herbal medicine for treating Alzheimer’s disease
Zhongduo Yang
Dongbo Zhang
Shuo Li
Original Research 05 February 2011 Pages: 734 - 738
QSAR and pharmacophore analysis of thiosemicarbazone derivatives as ribonucleotide reductase inhibitors
N. S. Hari Narayana Moorthy
Nuno M. F. S. A. Cerqueira
Pedro A. Fernandes
Original Research 05 February 2011 Pages: 739 - 746
Benzoxepin derivatives: design, synthesis, and pharmacological evaluation with sedative–hypnotic effect
Nagwa M. Abdel Gawad
Ghaneya S. Hassan
Hesham Y. El-Zorba
Original Research 06 February 2011 Pages: 747 - 759
Synthesis of antihyperglycemic, α-glucosidase inhibitory, and DPPH free radical scavenging furanochalcones
R. Ranga Rao
Ashok K. Tiwari
J. Madhusudana Rao
Original Research 08 February 2011 Pages: 760 - 774
Docking simulations, synthesis, and anti-inflammatory activity evaluation of 2-(N-alkyl)amino-3-nitroimidazo[1,2-a]pyridines
Yazmín K. Márquez-Flores
Ma. Elena Campos-Aldrete
Ma. Estela Meléndez-Camargo
Original Research 08 February 2011 Pages: 775 - 782
Nymphasterol, a new steroid from Nymphaea stellata
Amita Verma
Bahar Ahmed
Neetu Soni
Original Research 11 February 2011 Pages: 783 - 787
QSAR studies on substituted 3- or 4-phenyl-1,8-naphthyridine derivatives as antimicrobial agents
Ponnurengam Malliappan Sivakumar
Geetha Iyer
Mukesh Doble
Original Research 12 February 2011 Pages: 788 - 795
Synthesis and antibacterial evaluation of Cu(II) and Zn(II) complexes of the β-lactum antibiotic, cefdinir
Deepika Sharma
Pradeep Kumar
Balasubramanian Narasimhan
Original Research 13 February 2011 Pages: 796 - 803
Technetium-99m labeled Mebendazole and biodistribution in experimentally Trichinella spiralis-infected rats
Tonay Inceboz
Fatma Yurt Lambrecht
Ahmet Uner
Original Research 15 March 2011 Pages: 804 - 809
Novel antitubercular diallyl/dibenzylthiosemicarbazones endowed with high activity toward multi-drug-resistant tuberculosis
Dharmarajan Sriram
Debjani Banerjee
Perumal Yogeeswari
Original Research 07 April 2011 Pages: 810 - 815
New thiazolidinedione-5-acetic acid amide derivatives: synthesis, characterization and investigation of antimicrobial and cytotoxic properties
Shankar G. Alegaon
Kallanagouda R. Alagawadi
Original Research 17 February 2011 Pages: 816 - 824
Structure-based drug discovery of ApoE4 inhibitors from the plant compounds
Kh. Dhanachandra Singh
M. Karthikeyan
S. Nagamani
Original Research 17 February 2011 Pages: 825 - 833
Design, synthesis, and evaluation of novel indomethacin–antioxidant codrugs as gastrosparing NSAIDs
Shruti Sawraj
Tilak R. Bhardawaj
Pritam D. Sharma
Original Research 17 February 2011 Pages: 834 - 843
Comparative study of conventional and microwave-assisted synthesis of some Schiff bases and their potential as antimicrobial agents
Vikas Pandey
Viney Chawla
Shailendra K. Saraf
Original Research 17 February 2011 Pages: 844 - 852
QSAR and pharmacophore studies of telomerase inhibitors
Atefeh Hajiagha Bozorgi
Hamed Tabatabaei Ghomi
Abolghasem Jouyban
Original Research 18 February 2011 Pages: 853 - 866
Synthesis of novel 2-(3′-aryl-sydnon-4′-ylidene)-5′-substituted-[1,3,4]-thiadiazolylamines and [1,3,4]-thiadiazol-2′-yl-3-oxo-[1,2,4]-triazoles as antimicrobial agents
Soujanya Bansode
Ravindra Kamble
Original Research 17 February 2011 Pages: 867 - 873
Synthesis of curcumin and ethylcurcumin bioconjugates as potential antitumor agents
Reem I. Al-Wabli
Omaima M. AboulWafa
Khairia M. Youssef
Original Research 20 February 2011 Pages: 874 - 890
Common binding requirements of PPAR-α/δ/γ pan agonists: quantitative structure–activity relationship analysis of indanylacetic acid derivatives carrying 4-thiazolyl-phenoxy tail group
Sarvesh Paliwal
Divya Yadav
Shailendra Paliwal
Original Research 20 February 2011 Pages: 891 - 907
Synthesis of a New Series of 4-Aryl-1,4-Dihydropyridines with Calcium Channel Blocking and Vasodilatory Activity
Ranju Bansal
Priyanka Jain
Alan L. Harvey
Original Research 20 February 2011 Pages: 908 - 921
Chalcones as promising pesticidal agents against diamondback moth (Plutella xylostella): microwave-assisted synthesis and structure–activity relationship
Rakesh Kumar
Prabha Sharma
Arun Kumar Sinha
Original Research 20 February 2011 Pages: 922 - 931
Antibacterial and antifungal activities of some trimethoprim salts
Yağmur Tunalı
Hülya Karaca
Kadriye Benkli
Original Research 20 February 2011 Pages: 932 - 935
Erratum to: Antibacterial and antifungal activities of some trimethoprim salts
Yağmur Tunali
Hulya Karaca
Kadriye Benkli
Erratum 22 June 2011 Pages: 936 - 936
Protein–polysaccharides of Trametes versicolor: production and biological activities
José M. Santos Arteiro
M. Rosário Martins
A. Teresa Caldeira
Original Research 22 February 2011 Pages: 937 - 943
Synthesis of 2-R¹-2-(4-(2-fluoroethoxy)benzamido)acetate as potential PET imaging agents
Yong He
Jingli Xu
Ying Xie
Original Research 23 February 2011 Pages: 944 - 951

Volume 21, Issue 6

QSAR analysis on PfPK7 inhibitors using HQSAR, CoMFA, and CoMSIA

Synthesis, characterization and antimicrobial activity of 4-amino-1-alkyl pyridinium salts

Synthesis and antiviral activity of benzimidazolyl- and triazolyl-1,3,5-triazines

Synthesis of a ligand–quencher conjugate for the ligand binding study of the aryl hydrocarbon receptor using a FRET assay

Skimmianine, a furoquinoline alkaloid from Zanthoxylum nitidum as a potential acetylcholinesterase inhibitor

Synthesis of new piperidyl indanone derivatives as anticonvulsant agents

Acetylcholinesterase inhibitory activity of the total alkaloid from traditional Chinese herbal medicine for treating Alzheimer’s disease

QSAR and pharmacophore analysis of thiosemicarbazone derivatives as ribonucleotide reductase inhibitors

Benzoxepin derivatives: design, synthesis, and pharmacological evaluation with sedative–hypnotic effect

Synthesis of antihyperglycemic, α-glucosidase inhibitory, and DPPH free radical scavenging furanochalcones

Docking simulations, synthesis, and anti-inflammatory activity evaluation of 2-(N-alkyl)amino-3-nitroimidazo[1,2-a]pyridines

Nymphasterol, a new steroid from Nymphaea stellata

QSAR studies on substituted 3- or 4-phenyl-1,8-naphthyridine derivatives as antimicrobial agents

Synthesis and antibacterial evaluation of Cu(II) and Zn(II) complexes of the β-lactum antibiotic, cefdinir

Technetium-99m labeled Mebendazole and biodistribution in experimentally Trichinella spiralis-infected rats

Novel antitubercular diallyl/dibenzylthiosemicarbazones endowed with high activity toward multi-drug-resistant tuberculosis

New thiazolidinedione-5-acetic acid amide derivatives: synthesis, characterization and investigation of antimicrobial and cytotoxic properties

Structure-based drug discovery of ApoE4 inhibitors from the plant compounds

Design, synthesis, and evaluation of novel indomethacin–antioxidant codrugs as gastrosparing NSAIDs

Comparative study of conventional and microwave-assisted synthesis of some Schiff bases and their potential as antimicrobial agents

QSAR and pharmacophore studies of telomerase inhibitors

Synthesis of novel 2-(3′-aryl-sydnon-4′-ylidene)-5′-substituted-[1,3,4]-thiadiazolylamines and [1,3,4]-thiadiazol-2′-yl-3-oxo-[1,2,4]-triazoles as antimicrobial agents

Synthesis of curcumin and ethylcurcumin bioconjugates as potential antitumor agents

Common binding requirements of PPAR-α/δ/γ pan agonists: quantitative structure–activity relationship analysis of indanylacetic acid derivatives carrying 4-thiazolyl-phenoxy tail group

Synthesis of a New Series of 4-Aryl-1,4-Dihydropyridines with Calcium Channel Blocking and Vasodilatory Activity

Chalcones as promising pesticidal agents against diamondback moth (Plutella xylostella): microwave-assisted synthesis and structure–activity relationship

Antibacterial and antifungal activities of some trimethoprim salts

Erratum to: Antibacterial and antifungal activities of some trimethoprim salts

Protein–polysaccharides of Trametes versicolor: production and biological activities

Synthesis of 2-R¹-2-(4-(2-fluoroethoxy)benzamido)acetate as potential PET imaging agents

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