Synthesis and evaluation of thiopyrano[3,4-c]quinoline-9-carboxamide derivatives as inhibitors of poly(ADP-ribose) polymerase-1 (PARP-1) Chun-Ho ParkKwangwoo ChunMyung-Hwa Kim Original Research 25 May 2011 Pages: 1533 - 1543
Synthesis and local anaesthetic activities of 2-aminothiazole/thiadiazole analogues of lidocaine Naveen P. BadigerAshraf KhanI. M. Khazi Original Research 27 May 2011 Pages: 1544 - 1549
Microwave-assisted synthesis and antimicrobial activity of some imidazo[2,1-b][1,3,4]thiadiazole derivatives Sharad DhepeSujeet KumarSubhas S. Karki Original Research 27 May 2011 Pages: 1550 - 1556
Synthesis, antimycobacterial, antiviral, antimicrobial activities, and QSAR studies of nicotinic acid benzylidene hydrazide derivatives Rakesh NarangBalasubramanian NarasimhanJan Balzarini Original Research 28 May 2011 Pages: 1557 - 1576
A clubbed quinazolinone and 4-thiazolidinone as potential antimicrobial agents N. C. DesaiAmit M. DodiyaPrashant N. Shihora Original Research 28 May 2011 Pages: 1577 - 1586
Photodimerization of heteroaryl chalcones: comparative antimicrobial activities of chalcones and their photoproducts Rekha NagwanshiMeena BakhruShubha Jain Original Research 29 May 2011 Pages: 1587 - 1596
3D-QSAR and molecular docking studies of hydroxamic acids as peptide deformylase inhibitors Jian GaoYuanhua ChengMingjuan Ji Original Research 31 May 2011 Pages: 1597 - 1610
In vitro antimicrobial assessment of coumarin-based s-triazinyl piperazines Divyesh PatelRahul PatelNavin Patel Original Research 01 June 2011 Pages: 1611 - 1624
Analgesic study of novel pyrimidine derivatives linked with coumarin moiety Jitendra Kumar GuptaPramod K. SharmaShivjee Kashyap Original Research 03 June 2011 Pages: 1625 - 1632
Synthesis of new phenylcarbamoylbenzoic acid derivatives and evaluation of their in vitro antioxidant activity Waleed A. BayoumiMagda A. Elsayed Original Research 03 June 2011 Pages: 1633 - 1640
Synthesis of 9-O-glycosyl-berberine derivatives and bioavailability evaluation Zhu ChenXiaoli YeXuegang Li Original Research 03 June 2011 Pages: 1641 - 1646
Synthesis and antihypertensive activity evaluation in spontaneously hypertensive rats of lacidipine analogues Zeng-jun GuoKai ZhouSan-qi Zhang Original Research 03 June 2011 Pages: 1647 - 1651
Synthesis of 2-(aryl)-5-(arylidene)-4-thiazolidinone derivatives with potential analgesic and anti-inflammatory activity Aakash DeepSandeep JainManav Malhotra Original Research 04 June 2011 Pages: 1652 - 1659
Design, synthesis of some 2,6,9-trisubstituted purinyl thioureido derivatives and evaluation of antimicrobial activity Jigisha A. ModiK. C. Patel Original Research 04 June 2011 Pages: 1660 - 1664
QSAR and flexible docking studies of some aldose reductase inhibitors obtained from natural origin Shailesh V. JainKamlendra S. BhadoriyaSanjaykumar B. Bari Original Research 05 June 2011 Pages: 1665 - 1676
Molecular docking studies of potent inhibitors of tyrosinase and α-glucosidase Syed Sikander AzamReaz UddinZaheer-ul-Haq Original Research 05 June 2011 Pages: 1677 - 1683
Comparison of the constituents of Apocynum venetum and acidified Apocynum venetum by liquid chromatography–UV diode array detection–electrospray ionisation mass spectrometry Yuchi ZhangChunming LiuZhengkun Zhang Original Research 09 June 2011 Pages: 1684 - 1691
Synthesis and pharmacological properties of some novel pyrazolidine and pyrazole derivatives Bharat ParasharAbhilasha JainV. K. Sharma Original Research 09 June 2011 Pages: 1692 - 1699
Synthesis of new compounds derived from metronidazole and amino acids and their esters as antiparasitic agents Ahmed T. Al-MasriHaythem A. SaadehMohammad S. Mubarak Original Research 09 June 2011 Pages: 1700 - 1707
Synthesis, spectroscopic, thermal and antimicrobial studies of Co(II), Ni(II), Cu(II) and Zn(II) complexes with Schiff base derived from 4-amino-3-mercapto-6-methyl-5-oxo-1,2,4-triazine Kiran SinghYogender KumarK. R. Aneja Original Research 11 June 2011 Pages: 1708 - 1716
Antidiabetic and antioxidant activity of hydroxycinnamic acids from Calamintha Officinalis Moench. P. P. SinghS. JhaR. Irchhaiya Original Research 11 June 2011 Pages: 1717 - 1721
Synthesis and anti-inflammatory activity of some pyrazole derivatives Samir M. El-MoghazyFlora F. BarsoumAdel A. Marzouk Original Research 11 June 2011 Pages: 1722 - 1733
Synthesis and antibacterial activity of novel 7-haloanilino-8-nitrofluoroquinolone derivatives Yusuf M. Al-HiariAmjad M. QandilTariq M. Al-Qirim Original Research 11 June 2011 Pages: 1734 - 1740
Synthesis, evaluation of 6,8-dibromo-2-aryl-2,3-dihydroquinolin-4(1H)-ones in MCF-7 (breast cancer) cell lines and their docking studies Lakshmi Narayana BheemanapalliAmandeep KaurNarashima Murthy Javali Original Research 14 June 2011 Pages: 1741 - 1750
Synthesis, characterization and biological activity of some new carbostyril bearing 1H-pyrazole moiety Nilesh J. ThumarManish P. Patel Original Research 11 June 2011 Pages: 1751 - 1761
Synthesis and structure–activity relationships of serotonin derivatives effect on α-glucosidase inhibition Toshiyuki TakahashiMitsuo Miyazawa Original Research 18 June 2011 Pages: 1762 - 1770
Synthesis and pharmacological evaluation of some new naphthol derived aryloxy derivatives as cognition enhancers Poonam PiplaniRuchi MalikAnuradha Kaplish Original Research 22 June 2011 Pages: 1771 - 1779
Design, synthesis and biological evaluation of some novel 3-cinnamoyl-4-hydroxy-2H-chromen-2-ones as antimalarial agents Kuldeep PatelChandrabose KarthikeyanPiyush Trivedi Original Research 22 June 2011 Pages: 1780 - 1784
A facile and single pot strategy for the synthesis of novel naphthyridine derivatives under microwave irradiation conditions using ZnCl2 as catalyst, evaluation of AChE inhibitory activity, and molecular modeling studies C. KurumurthyP. Sambasiva RaoB. Narsaiah Original Research 22 June 2011 Pages: 1785 - 1795
Study of mangiferin-receptor affinity by cell membrane chromatography using rat pancreas Jian-Min ShenJin WangHai-Xia Zhang Original Research 22 June 2011 Pages: 1796 - 1802
Design and synthesis of new 2,4,5-triarylimidazole derivatives as selective cyclooxygenase (COX-2) inhibitors A. ZarghiS. ArfaeiR. Ghodsi Original Research 24 June 2011 Pages: 1803 - 1810
Synthesis, characterization and antimicrobial activities of some novel bis-chalcones Akbar MobinikhalediMehdi KalhorHossein Jamalifar Original Research 25 June 2011 Pages: 1811 - 1816
Investigation of myorelaxant activity of 9-aryl-3,4,6,7-tetrahydroacridine-1,8-(2H,5H,9H,10H)-diones in isolated rabbit gastric fundus Gökçe Sevim Öztürk FincanMiyase Gözde GündüzCihat Şafak Original Research 25 June 2011 Pages: 1817 - 1824
Synthesis, molecular docking, and cardioprotective activity of 2-methylthio-1,4-dihydropyrimidines Ramesh L. SawantVarsha I. SarodeJyoti B. Wadekar Original Research 25 June 2011 Pages: 1825 - 1832
Investigation on the substitution effects of the flavonoids as potent anticancer agents: a structure–activity relationships study Xiao-Bing WangWei LiuLing-Yi Kong Original Research 25 June 2011 Pages: 1833 - 1849
Antioxidant potential and antimicrobial screening of some novel imidazole derivatives: greenway efficient one pot synthesis Jayaraman JayabharathiVenugopal ThanikachalamMarimuthu Venkatesh Perumal Original Research 25 June 2011 Pages: 1850 - 1860
Synthesis, preliminary cytotoxicity evaluation of new 3-formylchromone hydrazones and phosphorohydrazone derivatives of coumarin and chromone A. ŁazarenkowJ. Nawrot-ModrankaM. Różalski Original Research 25 June 2011 Pages: 1861 - 1868
Design and synthesis of new 1,2-diaryl-4,5,6,7-tetrahydro-1H-benzo[d] imidazoles as selective cyclooxygenase (COX-2) inhibitors A. ZarghiH. ReihanfardM. Hedayati Original Research 25 June 2011 Pages: 1869 - 1875
Synthesis of some novel triazoloquinazolines and triazinoquinazolines and their evaluation for anti-inflammatory activity Mohammed Abdalla Hussein Original Research 28 June 2011 Pages: 1876 - 1886
Synthesis and anti-tubercular evaluation of some novel pyrazolo[3,4-d]pyrimidine derivatives Amit R. TrivediBipin H. DholariyaViresh H. Shah Original Research 28 June 2011 Pages: 1887 - 1891
Molecular modeling study of HIV-1 gp120 attachment inhibitors Changdev G. GadheGugan KothandanSeung Joo Cho Original Research 30 June 2011 Pages: 1892 - 1904
Synthesis of N-hydroxycinnamoyl amino acid ester analogues and their free radical scavenging and antioxidative activities Qing-Yi WeiHong JiangHuan Wang Original Research 30 June 2011 Pages: 1905 - 1911
Docking and quantitative structure–activity relationship studies for imidazo[1,2-a]pyrazines as inhibitors of checkpoint kinase-1 Julio CaballeroSzymon ZilocchiSimona Collina Original Research 06 July 2011 Pages: 1912 - 1920
Structure–cytotoxicity relationship of a novel series of miconazole-like compounds Reza YousefiAli Khalafi-NezhadAli Akbar Moosavi-Movahedi Original Research 07 July 2011 Pages: 1921 - 1928
Substituted 2-[2-(pyridin-3-yl) phenyl] acetamides and ureas: design, synthesis, and anticonvulsant screening in mice A. V. ShindikarC. L. Viswanathan Original Research 07 July 2011 Pages: 1929 - 1934
Synthesis, antimycobacterial, antiviral, antimicrobial activities, and QSAR studies of isonicotinic acid-1-(substituted phenyl)-ethylidene/cycloheptylidene hydrazides Vikramjeet JudgeBalasubramanian NarasimhanJan Balzarini Original Research 09 July 2011 Pages: 1935 - 1952
Synthesis and QSAR analysis of chalcone derivatives as nitric oxide inhibitory agent Kok Wai LamReaz UddinNordin H. Lajis Original Research 09 July 2011 Pages: 1953 - 1966
Synthesis and evaluation of 4-(substituted)-acetylamino-3-mercapto-5-(4-substituted) phenyl-1,2,4-triazole derivatives as antimicrobial agents Neeraj UpmanyuSanjay KumarPradeep Mishra Original Research 09 July 2011 Pages: 1967 - 1976
Synthesis of 1-(4-((E)-3-arylacryloyl) phenyl)-3,4-dibromo-1H-pyrrole-2,5-diones and screening for anti-Candida and antituberculosis activity J. R. PatelB. Z. Dholakiya Original Research 09 July 2011 Pages: 1977 - 1983
Petra, Osiris and Molinspiration (POM) together as a successful support in drug design: antibacterial activity and biopharmaceutical characterization of some azo Schiff bases Aliasghar JarrahpourJihane FathiAli Parvez Original Research 09 July 2011 Pages: 1984 - 1990
