Synthesis of mono- and bis-spirooxindole derivatives “on water” using double salt of aluminum sulfate–sulfuric acid as a reusable catalyst Mohammad BashkarMasoumeh BavadiKhodabakhsh Niknam Original Article 30 April 2020 Pages: 2001 - 2015
Design and synthesis of novel (Z)-5-((1,3-diphenyl-1H-pyrazol-4-yl)methylene)-3-((1-substituted phenyl-1H-1,2,3-triazol-4-yl)methyl)thiazolidine-2,4-diones: a potential cytotoxic scaffolds and their molecular modeling studies N. J. P. SubhashiniKolluri Prashanth KumarManga Vijjulatha Original Article 02 May 2020 Pages: 2017 - 2033
Chemistry and anti-herpes simplex virus type 1 evaluation of 4-substituted-1H-1,2,3-triazole-nitroxyl-linked hybrids Anna C. CunhaVitor F. FerreiraAlessandro K. Jordão Original Article 06 May 2020 Pages: 2035 - 2043
Design, antihuman immunodeficiency activity and molecular docking studies of synthesized 2-aryl and 2-pyrimidinyl pyrrolidines Sahak P. GasparyanAshot H. MartirosyanRaymond F. Schinazi Original Article 05 May 2020 Pages: 2045 - 2052
A three-component cyclocondensation reaction for the synthesis of new triazolo[1,5-a]pyrimidine scaffolds using 3-aminotriazole, aldehydes and ketene N,S-acetal Solmaz KaramiMohammad BayatFaezeh Mirzaei Original Article 09 May 2020 Pages: 2053 - 2062
Synthesis of polycyclic N-heterocyclic compounds via one-pot three-component cyclization strategy Abdolali AlizadehElham SanjariMohammad Reza Halvagar Original Article 08 May 2020 Pages: 2063 - 2072
Synthesis and antimicrobial activities of some novel diastereoselective monocyclic cis-β-lactams using 2-ethoxy carbonyl DCPN as a carboxylic acid activator Mahesh Kumar MishraVedeshwar Narayan SinghSitaram Sharma Original Article 13 May 2020 Pages: 2073 - 2087
Novel 1,2,4-triazole analogues as mushroom tyrosinase inhibitors: synthesis, kinetic mechanism, cytotoxicity and computational studies Balasaheb D. VanjarePrasad G. MahajanKi Hwan Lee Original Article 12 May 2020 Pages: 2089 - 2106
Design and exploration of 5-nitro-3-trinitromethyl-1H-1,2,4-triazole and its derivatives as energetic materials Jian-ying ZhangGang-ling ChenXue-dong Gong Original Article 20 May 2020 Pages: 2107 - 2121
Synthesis of new curcumin-based aminocarbonitrile derivatives incorporating 4H-pyran and 1,4-dihydropyridine heterocycles Soheila Khajeh DangolaniFarhad PanahiAli Khalafi-Nezhad Original Article 17 May 2020 Pages: 2123 - 2135
Indole-fused spirochromenes as potential anti-tubercular agents: design, synthesis and in vitro evaluation Ashok DogamantiPamula ChiranjeeviMadderla Sarasija Original Article 30 May 2020 Pages: 2137 - 2148
Urease: a highly efficient biocatalyst for synthesis of polyhydroquinolines and polyhydroacridines from the ammonia formed in situ Gan ZhuYiqun Li Original Article 07 June 2020 Pages: 2149 - 2159
Synthesis of styryl-linked fused dihydropyridines by catalyst-free multicomponent reactions Rahul YadavTasneem ParvinLokman H. Choudhury Original Article 16 April 2021 Pages: 2161 - 2169
Production of benzazepine derivatives via four-component reaction of isatins: study of antioxidant activity Fathali Gholami OrimiBehrooz MirzaZinatossadat Hossaini Original Article 10 June 2020 Pages: 2171 - 2182
A facile green synthesis of MgCoFe2O4 nanomaterials with robust catalytic performance in the synthesis of pyrano[2,3-d]pyrimidinedione and their bis-derivatives Monireh AtarodJavad SafariAli Pourjavadi Original Article 27 July 2020 Pages: 2183 - 2200
Synthesis, antimicrobial evaluation, and in silico studies of quinoline—1H-1,2,3-triazole molecular hybrids Paul AwoladeNosipho CeleParvesh Singh Original Article 07 June 2020 Pages: 2201 - 2218
Planning new Trypanosoma cruzi CYP51 inhibitors using QSAR studies Pedro Igor Camara de OliveiraPaulo Henrique de Santana MirandaEuzebio Guimaraes Barbosa Original Article 16 June 2020 Pages: 2219 - 2235
Synthesis of tetracyclic pyrido-fused dibenzodiazepines via a catalyst-free cascade reaction Abdolali AlizadehAkram Bagherinejad Original Article 14 June 2020 Pages: 2237 - 2246
Head-to-head bisbenzazole derivatives as antiproliferative agents: design, synthesis, in vitro activity, and SAR analysis Ronak Haj ErsanMehmet Abdullah AlagozOztekin Algul Original Article 18 June 2020 Pages: 2247 - 2259
Design and in vitro analysis of SIRT2 inhibitor targeting Parkinson’s disease Amrendra Pratap SinghLokesh NigamSharmistha Dey Original Article 26 June 2020 Pages: 2261 - 2270
Comparative biological study between quinazolinyl–triazinyl semicarbazide and thiosemicarbazide hybrid derivatives Janki J. PatelRahul P. ModhKishor H. Chikhalia Original Article 28 June 2020 Pages: 2271 - 2287
Antiproliferative activity of cardenolides on cell line A549: structure–activity relationship analysis Salvador Enrique Meneses-SagreroLuisa Alondra Rascón-ValenzuelaRamón Enrique Robles-Zepeda Original Article 05 July 2020 Pages: 2289 - 2305
Antiproliferative and antiinflammatory coxib–combretastatin hybrids suppress cell cycle progression and induce apoptosis of MCF7 breast cancer cells Quoc Anh NgoThuy Hang Nguyen ThiThi Thao Do Original Article 30 June 2020 Pages: 2307 - 2319
Revisit to the synthesis of 1,2,3,4-tetrasubstituted pyrrole derivatives in lactic acid media as a green solvent and catalyst Dilek AkbaslarE. Sultan GirayOztekin Algul Original Article 27 September 2020 Pages: 2321 - 2338
4H-benzochromene derivatives as novel tyrosinase inhibitors and radical scavengers: synthesis, biological evaluation, and molecular docking analysis Somaye KarimianSara RanjbarMehdi Khoshneviszadeh Original Article 18 July 2020 Pages: 2339 - 2349
A drug–biomarker interaction model to predict the key targets of Scutellaria barbata D. Don in adverse-risk acute myeloid leukaemia Teng WangChun-yi LyuRui-rong Xu Original Article 16 July 2020 Pages: 2351 - 2365
Ultrasound-assisted, low-solvent and acid/base-free synthesis of 5-substituted 1,3,4-oxadiazole-2-thiols as potent antimicrobial and antioxidant agents Elahe YarmohammadiHamid BeyzaeiAshraf Moradi Original Article 08 August 2020 Pages: 2367 - 2378
Synthesis of pyrazole-4-carboxamides as potential fungicide candidates Cuntao DongWei GaoLai Chen Original Article 30 July 2020 Pages: 2379 - 2388
Dehydroabietylamine-based thiazolidin-4-ones and 2-thioxoimidazolidin-4-ones as novel tyrosyl-DNA phosphodiesterase 1 inhibitors Kseniya KovalevaEvgeniya MamontovaNariman Salakhutdinov Original Article 24 August 2020 Pages: 2389 - 2397
Synthesis of 4-alkylaminoimidazo[1,2-a]pyridines linked to carbamate moiety as potent α-glucosidase inhibitors Mina SaeediMaryam Raeisi-NafchiTahmineh Akbarzadeh Original Article 12 October 2020 Pages: 2399 - 2409
Selection of antileishmanial sesquiterpene lactones from SistematX database using a combined ligand-/structure-based virtual screening approach Chonny Herrera-AcevedoMayara Dos Santos MaiaMarcus Tullius Scotti Original Article 09 September 2020 Pages: 2411 - 2427
Anticancer activity and evaluation of apoptotic genes expression of 2-azetidinones containing anthraquinone moiety Masoud MohamadzadehMaaroof Zarei Original Article 18 September 2020 Pages: 2429 - 2439
Facile synthesis of pyrrolo[2,1-a]isoquinolines by domino reaction of 1-aroyl-3,4-dihydroisoquinolines with conjugated ketones, nitroalkenes and nitriles Grigorii S. AstakhovRinat R. ShigaevMaria D. Matveeva Original Article 10 October 2020 Pages: 2441 - 2446
Construction of hybrid polycyclic quinolinobenzo[a]phenazinone architectures using solid-state melt reaction (SSMR) Manickam BakthadossVarathan Vinayagam Short Communication 04 May 2020 Pages: 2447 - 2458
gem-Difunctionalization of α-diazoarylketones with diaryldiselenides and N-halosuccinimides: facile synthesis of α-halo-α-arylseleno ketones Jiuling LiDong XingWenhao Hu Short Communication 14 May 2020 Pages: 2459 - 2466
Domino ring opening and selective O/S-alkylation of cyclic ethers and thioethers Manickam BakthadossVishal AgarwalMushaf Mohammad Short Communication 27 May 2020 Pages: 2467 - 2478
Visible-light-mediated one-pot efficient synthesis of 1-aryl-1H,3H-thiazolo[3,4-a]benzimidazoles: a metal-free photochemical approach in aqueous ethanol Mohd NazeefKm Neha ShivhareI. R. Siddiqui Short Communication 27 September 2020 Pages: 2479 - 2486
Recent synthetic strategies toward the synthesis of spirocyclic compounds comprising six-membered carbocyclic/heterocyclic ring systems Kashaf BabarAmeer Fawad ZahoorRabia Akhtar Comprehensive review 21 July 2020 Pages: 2487 - 2532
Vinylazides: versatile synthons and magical precursors for the construction of N-heterocycles Zahra TashrifiMohammad Mohammadi-KhanaposhtaniMohammad Mahdavi Short review 30 May 2020 Pages: 2533 - 2570
Recent strategies in the synthesis of thiophene derivatives: highlights from the 2012–2020 literature Fahimeh AbedinifarElham Babazadeh RezaeiMohammad Mahdavi Short review 30 July 2020 Pages: 2571 - 2604
