Kaempferia diterpenoids and flavonoids: an overview on phytochemistry, biosynthesis, synthesis, pharmacology, and pharmacokinetics Chu Anh VanDau Xuan DucNinh The Son Review Article 21 November 2023 Pages: 1 - 20
FTase inhibitors and cancer: prospects for use in targeted therapies Ming-tao XiaLing YuShuai Li Review Article 09 December 2023 Pages: 21 - 35
Pyrrolobenzodiazepines: natural sources, therapeutic uses, and future in neurological treatments Hadi ObajiAbbas G. ShilabinMohamed A. Ibrahim Review Article 18 December 2023 Pages: 36 - 46
A concise review on anti-breast cancer effectiveness of s-triazines through EGFR kinase inhibition Pooja TandelRachana UpadhyayAmit B. Patel Review Article 21 December 2023 Pages: 47 - 65
Design, synthesis, and in silico studies of novel di-(2-aryl hydrozonopropanal) arene derivatives as potent anticancer for targeting A2AR and LRP6 in HCT116 cell Tahani BakhshTamer S. SalehKhadijah M. Al-Zaydi Original Research Article 03 November 2023 Pages: 66 - 76
Design, synthesis and antimicrobial activities of 1,2,3-triazole hybrids with amine-ester functionality Jyoti SangwanC. P. KaushikManisha Chahal Original Research Article 04 November 2023 Pages: 77 - 88
Design and synthesis of novel cycloalkanecarboxamide parabanic acid hybrids as anticonvulsants Walaa Hamada Abd-AllahMohamed Samir Abd El-MaksoudRasha Mohamed Hassan Original Research Article Open access 15 November 2023 Pages: 89 - 106
Characterization of novel angiotensin-I converting enzyme inhibitory peptides derived from Taiwan red quinoa (Chenopodium formosanum Koidz.) seed proteins using two sequential bioassay-guided fractionations Dininurilmi Putri SulemanChristoper Caesar Yudho SutopoJue-Liang Hsu Original Research Article 23 November 2023 Pages: 107 - 116
One-pot synthesis and in vitro bioactivity of novel 4-aminopyrazolo[3,4-b]pyridine derivatives as potential antimicrobial compounds Ranjana AggarwalSuresh KumarDeepansh Sharma Original Research Article 23 November 2023 Pages: 117 - 126
Enantioselectivity of pinene against Leishmania amazonensis Ingrid S. AdãoAndreza R. GarciaIgor A. Rodrigues Original Research Article 25 November 2023 Pages: 127 - 135
Discovery of novel fatty acid amide hydrolase (FAAH) inhibitors as anti-Alzheimer’s agents through pharmacophore-based virtual screening, molecular docking and experimental validation Smita JainSwapnil SharmaJaiprakash Sharma Original Research Article 09 December 2023 Pages: 136 - 150
Computer-aided design, synthesis and evaluation of new SARS-CoV-2 Mpro inhibitors based on 1,5,6,7-tetrahydro-4H-indazol-4-one scaffold Yuri A. PivenVeronica G. ZinovichFedor A. Lakhvich Original Research Article 11 December 2023 Pages: 151 - 163
Indazole derivatives as novel inhibitors of monoamine oxidase and D-amino acid oxidase Chezélle StearAnél PetzerJacobus P. Petzer Original Research Article Open access 15 December 2023 Pages: 164 - 176
Design, synthesis, molecular docking, and biological activity of pyrazolo[3,4-b]pyridines as promising lead candidates against Mycobacterium tuberculosis H. Surya Prakash RaoR. GunasundariJayaraman Muthukumaran Original Research Article 19 December 2023 Pages: 177 - 200
Design, synthesis and evaluation of aurone and indanone derivatives as novel antitumor agents Baoxing XieGulmira TurduHaji Akber Aisa Original Research Article 20 December 2023 Pages: 201 - 220