1. Synthesis and biological evaluation of new 2-(6-alkyl-pyrazin-2-yl)-1H-benz[d]imidazoles as potent anti-inflammatory and antioxidant agents

   • Bhookya Shankar
   • Pochampally Jalapathi
   • Karunakar rao Kudle

   Original Research 17 April 2017 Pages: 1835 - 1846

   

2. Novel derivatives of substituted 6-fluorobenzothiazole diamides: synthesis, antifungal activity and cytotoxicity

   • Marcela Pejchalová
   • Radim Havelek
   • Vladimír Pejchal

   Original Research 17 April 2017 Pages: 1847 - 1862

   

3. A novel PTP1b inhibitor vanadium-flavone complex: synthesis and pharmacodynamic evaluation in streptozotocin-induced diabetic mice

   • Liying Duan
   • Junwei Ye
   • Guiling Ning

   Original Research 19 April 2017 Pages: 1863 - 1870

   

4. Synthesis and biological evaluation of α-methyl-chalcone for anti-cervical cancer activity

   • Bing-zhao Ren
   • Mourboul Ablise
   • Zheng Yang

   Original Research 22 April 2017 Pages: 1871 - 1883

   

5. In vitro and in silico evaluation of chromene based aroyl hydrazones as anticonvulsant agents

   • Violina T. Angelova
   • Yulian Voynikov
   • Jana Tchekalarova

   Original Research 22 April 2017 Pages: 1884 - 1896

   

6. Isolation and characterization of Streptomyces tauricus from Thajiwas glacier—a new source of actinomycin-D

   • Shabir Ahmad Rather
   • Aabid Manzoor Shah
   • Qazi Parvaiz Hassan

   Original Research 26 April 2017 Pages: 1897 - 1902

   

7. QSAR and pharmacophore modeling of anti-tubercular 6-Fluoroquinolone compounds utilizing calculated structural descriptors

   • Dipiksha
   • Mohd Salman
   • Sisir Nandi

   Original Research 26 April 2017 Pages: 1903 - 1914

   

8. Chemopreventive effect of saponin isolated from Gymnema sylevestre on prostate cancer through in silico and in vivo analysis

   • Rajamanickam Pon Nivedha
   • Venkatesan Suryanarayanan
   • Manikkam Rajalakshmi

   Original Research 26 April 2017 Pages: 1915 - 1925

   

9. Computational insights into HER3 gatekeeper T768I resistance mutation to bosutinib in HER3-related breast cancer

   • Chun-Ling Dong
   • Fang-Chun Guo
   • Jie Xue

   Original Research 26 April 2017 Pages: 1926 - 1934

   

10. Synthesis and evaluation of the anticonvulsant activities of 2,3-dihydrophthalazine-1,4-dione derivatives

    • Xiang-Jun Liu
    • Hong-Jian Zhang
    • Zhe-Shan Quan

    Original Research 27 April 2017 Pages: 1935 - 1946

    

11. (S,E)-2-hydroxy-N-(2-hydroxy-5-nitrobenzylidene) propane hydrazide as a quorum sensing inhibitor of Pseudomonas aeruginosa

    • Azam Heidari
    • Fakhri Haghi
    • Rahman Bikas

    Original Research 28 April 2017 Pages: 1947 - 1955

    

12. Novel arylazothiazoles and arylazo[1,3,4]thiadiazoles as potential antimicrobial and anticancer agents: synthesis, molecular modeling, and biological screening

    • Sayed M. Riyadh
    • Anwar A. Deawaly
    • Saleh Ihmaid

    Original Research 02 May 2017 Pages: 1956 - 1968

    

13. Design, synthesis and QSAR studies of 2-amino benzo[d]thiazolyl substituted pyrazol-5-ones: novel class of promising antibacterial agents

    • Mahesh B. Palkar
    • Aniket Patil
    • Rajshekhar V. Karpoormath

    Original Research 05 May 2017 Pages: 1969 - 1987

    

14. Development and application of novel molecular descriptors for predicting biological activity

    • R. Dutt
    • A. K. Madan

    Original Research 06 May 2017 Pages: 1988 - 2006

    

15. Replacing triazole with diazole to optimize physicochemical properties of a click-based lead compound

    • Yinping Tian
    • Wenhui Lv
    • Jie Shen

    Original Research 09 May 2017 Pages: 2007 - 2014

    

16. Synthesis and structure elucidation of 1-(2,5/3,5-difluorophenyl)-3-(2,3/2,4/2,5/3,4-dimethoxyphenyl)-2-propen-1-ones as anticancer agents

    • Cem Yamali
    • Dilan Ozmen Ozgun
    • Noriyuki Okudaira

    Original Research 09 May 2017 Pages: 2015 - 2023

    

17. Synthesis, antioxidative and antiproliferative activity of methoxy amidino substituted benzamides and benzimidazoles

    • Maja Cindrić
    • Irena Sović
    • Kristina Starčević

    Original Research 09 May 2017 Pages: 2024 - 2037

    

18. BIX-01294 inhibits oncoproteins NSD1, NSD2 and NSD3

    • Masayo Morishita
    • Damiaan E. H. F. Mevius
    • Eric di Luccio

    Original Research 09 May 2017 Pages: 2038 - 2047

    

19. Investigation on the effects of pomiferin from Maclura pomifera on indomethacin-induced gastric ulcer: An experimental study in rats

    • İlyas Bozkurt
    • Esra Dilek
    • Mesut Bünyami Halici

    Original Research 12 May 2017 Pages: 2048 - 2056

    

20. The hepatoprotective activity of a new derivative kaempferol glycoside from the leaves of Vietnamese Phyllanthus acidus (L.) Skeels

    • Nguyen Cong Thuy Tram
    • Ninh The Son
    • Do Thi Thao

    Original Research 15 May 2017 Pages: 2057 - 2064

    

21. Cytotoxic activity evaluation and molecular docking study of phenolic derivatives from Achillea fragrantissima (Forssk.) growing in Egypt

    • Basma M. Awad
    • Eman S. Habib
    • Safwat A. Ahmed

    Original Research 16 May 2017 Pages: 2065 - 2073

    

22. Flavonoid rutinosides from Cinnamomum parthenoxylon leaves and their hepatoprotective and antioxidant activity

    • Antoni Pardede
    • Morina Adfa
    • Mamoru Koketsu

    Original Research 16 May 2017 Pages: 2074 - 2079

    

23. Synthesis and evaluation of novel urea and amide derivatives of 2-amino-4-phenylthiazole as potential antibacterial agents

    • Zhi-Hua Zhang
    • Yu Chen
    • Song You

    Original Research 17 May 2017 Pages: 2080 - 2087

    

24. Synthesis, biological evaluation and molecular docking studies of novel quinuclidinone derivatives as potential antimicrobial and anticonvulsant agents

    • Krzysztof Z. Łączkowski
    • Katarzyna Landowska
    • Anna Malm

    Original Research 19 May 2017 Pages: 2088 - 2104

    

25. The combination of Bleomycin with TRAIL agonists or PKC inhibitors sensitizes solid tumor cells to BLM-mediated apoptosis: new strategies to overcome chemotherapy resistance of tumors

    • Souhir Brahim
    • Sonia Aroui
    • Ali Bettaieb

    Original Research 19 May 2017 Pages: 2105 - 2111

    

26. Molecular screening and analysis of novel therapeutic inhibitors against c-Jun N-terminal kinase

    • Trinath Daggupati
    • Kumaraswamy Naidu Chitrala
    • Suneetha Yeguvapalli

    Original Research 19 May 2017 Pages: 2112 - 2118

    

27. Anti-HIV-1 and cytotoxicity of a new dimeric thiazepine alkaloid isolated from Ixora undulata Roxb. leaves

    • Magdy M. D. Mohammed
    • Khaled M. Mohamed

    Original Research 20 May 2017 Pages: 2119 - 2126

    

28. Design, synthesis and in vitro evaluation of some small molecules malonyl CoA decarboxylase inhibitors containing pyrazoline scaffold and study of their binding interactions with malonyl CoA decarboxylase via preliminary docking simulation

    • Deepali M. Jagdale
    • C. S. Ramaa

    Original Research 22 May 2017 Pages: 2127 - 2140

    

29. Synthesis, in vitro antimicrobial, antioxidant, and antidiabetic activities of thiazolidine–quinoxaline derivatives with amino acid side chains

    • Suhas A. Shintre
    • Deresh Ramjugernath
    • Neil A. Koorbanally

    Original Research 22 May 2017 Pages: 2141 - 2151

    

30. Synthesis and anti(myco)bacterial activity of novel 5,5-diphenylpyrrolidine N-aroylthiourea derivatives and a functionalized hexahydro-1H-pyrrolo[1,2-c]imidazole

    • Duygu Erşen
    • Mahmut Ülger
    • Yahya Nural

    Original Research 24 May 2017 Pages: 2152 - 2160

    

31. Synthesis and inhibitory effects of triarylpyrazoles on LPS-induced NO and PGE₂ productions in RAW 264.7 macrophages

    • Byung-Jun Park
    • Mohammed I. El-Gamal
    • Chang-Hyun Oh

    Original Research 29 May 2017 Pages: 2161 - 2171

    

32. (E)-2-Benzylidenecyclanones: part XIV. Study on interaction of some (E)-2-benzylidenebenzosuberone derivatives with calf thymus DNA by TLC and UV–Vis methods, a DNA cleavage study

    • Zsuzsanna Rozmer
    • Evelin Marton
    • Pál Perjési

    Original Research 29 May 2017 Pages: 2172 - 2179

    

33. Design, synthesis and cytotoxic evaluation of a novel series of benzo[d]thiazole-2-carboxamide derivatives as potential EGFR inhibitors

    • Lan Zhang
    • Xin-Shan Deng
    • Chun Hu

    Original Research 29 May 2017 Pages: 2180 - 2189

    

34. Regioselective synthesis of some new 1,4-disubstituted sulfonyl-1,2,3-triazoles and their antibacterial activity studies

    • Narasimha Swamy Thirukovela
    • Shravankumar Kankala
    • Ravinder Vadde

    Original Research 29 May 2017 Pages: 2190 - 2195

    

35. Efficacy of extracts and iridoid glucosides from Pentas lanceolata on humoral and cell-mediated immune response of viral vaccine

    • Howaida I. Abd-Alla
    • Heba-tollah M. Sweelam
    • Mohamed-Elamir F. Hegazy

    Original Research 29 May 2017 Pages: 2196 - 2204

    

36. Synthesis, characterization and biological evaluation of some new indomethacin analogs with a colon tumor cell growth inhibitory activity

    • Sally I. Eissa

    Original Research 01 June 2017 Pages: 2205 - 2220