Prostaglandin analogues: current treatment option for glaucoma Poonam PiplaniDeepali AggarwalLovneet Saini Review Article 07 April 2016 Pages: 1031 - 1048
In silico structural prediction of human steroid 5α-reductase type II Wiranpat KarnsomwanThanyada RungrotmongkolSupakarn Chamni Original Research 09 March 2016 Pages: 1049 - 1056
Synthesis of novel triazolyl pyranochromen-2(1H)-ones and their antibacterial activity evaluation Shiv KumarSuchita PrasadSunil K. Sharma Original Research 12 March 2016 Pages: 1057 - 1073
Synthesis and biological evaluation of phenylpropanoid derivatives Sheng LiuYubin LiJingchen Wei Original Research 12 March 2016 Pages: 1074 - 1086
3-Epihydroxy lup-20(29)-en-19(28)-olide: partial synthesis, antitopoisomerase activity, and 3D molecular docking Amitava MandalAshim GhoshPranab Ghosh Original Research 14 March 2016 Pages: 1087 - 1095
Convenient synthesis, anticancer evaluation and QSAR studies of some thiazole tethered indenopyrazoles Satbir MorSavita NagoriaSandeep Lohan Original Research 16 March 2016 Pages: 1096 - 1114
Predicting potential antitumor targets of Aconitum alkaloids by molecular docking and protein–ligand interaction fingerprint Jing-wei LiangTing-jian ZhangFan-hao Meng Original Research 18 March 2016 Pages: 1115 - 1124
Synthesis, biological evaluation of 2,3-disubstituted-imidazolyl/benzimidazolyl-quinazolin-4(3H)-one derivatives Dilip A. PatilSanjay J. Surana Original Research 19 March 2016 Pages: 1125 - 1139
Pharmacophore modeling and 3D-QSAR studies of galloyl benzamides as potent P-gp inhibitors Shubham SrivastavaBhanwar Singh ChoudharyRuchi Malik Original Research 21 March 2016 Pages: 1140 - 1147
Design, synthesis, and in vitro antiplasmodial activity of 4-aminoquinolines containing modified amino acid conjugates Kondaparla SrinivasaraoPooja AgarwalS. B. Katti Original Research 25 March 2016 Pages: 1148 - 1162
Pyridine-catalyzed synthesis of quinoxalines as anticancer and anti-tubercular agents Atulkumar A. KambleRavindra R. KambleGireesh Tegginamath Original Research 28 March 2016 Pages: 1163 - 1174
Ferulic acid amide derivatives as anticancer and antioxidant agents: synthesis, thermal, biological and computational studies Naresh KumarSandeep KumarVikas Pruthi Original Research 29 March 2016 Pages: 1175 - 1192
Synthesis and evaluation of the trypanocidal activity of a series of 1,3,4-thiadiazoles derivatives of R-(+)-limonene benzaldehyde-thiosemicarbazones Solange C. MartinsVânia C. DesotiCelso V. Nakamura Original Research 31 March 2016 Pages: 1193 - 1203
Features of reversible P2Y12 receptor antagonists based on piperazinyl-glutamate-pyridines Zhen ZhangGuanzhong WuKejiang Lin Original Research 04 April 2016 Pages: 1204 - 1215
Synthesis, structure–activity relationship and antinociceptive activities of some 2-(2′-pyridyl) benzimidazole derivatives Arfa KamilShamim AkhtarUmar Farooq Original Research 04 April 2016 Pages: 1216 - 1228
Synthesis of several 4H-chromene derivatives of expected antitumor activity Ahmed M. Fouda Original Research 07 April 2016 Pages: 1229 - 1238
Synthesis and biological testing of (5Z)-2-aryl-5-arylmethylidene-3,5-dihydro-4H-imidazol-4-ones as antimitotic agents Anastasia A. BeloglazkinaBirgit WobithOlga N. Zefirova Original Research 07 April 2016 Pages: 1239 - 1249
Structural basis of DNA topoisomerase II-α (Top2-α) inhibition: a computational analysis of interactions between Top2-α and its inhibitors Farzaneh Mohamadi FarsaniMohamad Reza GanjalikhanySadeq Vallian Original Research 07 April 2016 Pages: 1250 - 1259
Synthesis of oxadiazoline and quinazolinone derivatives and their biological evaluation as nitric oxide synthase inhibitors M. José Pineda de las InfantasM. Dora CarriónM. Encarnación Camacho Original Research 08 April 2016 Pages: 1260 - 1273
Synthesis, antibacterial and antifungal activities of naphthoquinone derivatives: a structure–activity relationship study Juan M. Sánchez-CalvoGara R. BarberoFrancisco A. Macías Original Research 12 April 2016 Pages: 1274 - 1285