Hypoglycemic herbs and their polyherbal formulations: a comprehensive review Deepti KatiyarVijender SinghAmita Vats Review Article 05 July 2014 Pages: 1 - 21
Comparative atom-based 3D QSAR study of 3-nitro-1H-1,2,4-triazole-based aliphatic and aromatic amines analogs for its anti-trypanosomal activities Suresh KumarRitesh AgrawalSandhya Bawa Original Research 03 July 2014 Pages: 22 - 31
Synthesis, structure elucidation, and anti-inflammatory/anti-cancer/anti-bacterial activities of novel (Z)-3-adamantyl-1-aryl-prop/but-2-en-1-ones Utpalparna KalitaShunan KapingJai Narain Vishwakarma Original Research 03 July 2014 Pages: 32 - 50
Design and microwave-assisted synthesis of tri- and dialkyltin(IV) hippurates, characterization, in vitro anti-cancer and in vivo anti-inflammatory activities Mala NathMonika VatsParta Roy Original Research 03 July 2014 Pages: 51 - 62
Synthesis, characterization, antibacterial, DNA cleavage and SOD activities of some 3d metal complexes of ethyl[2-(1H-indol-3-yl)methyleneamino]-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylate E. M. NiecyL. P. NithaK. Mohanan Original Research 03 July 2014 Pages: 63 - 77
Synthesis, bioassay studies, and molecular docking of novel 5-substituted 1H tetrazoles as cyclooxygenase-2 (COX-2) inhibitors Baker Jawabrah Al-HouraniSai Kiran SharmaFrank Wuest Original Research 03 July 2014 Pages: 78 - 85
Synthesis, antioxidant, and cytotoxic activities of bis(oxazolyl/thiazolyl/imidazolyl)amidomethanesulfonyl Acetamides Putta Ramachandra ReddyDandu SeenaiahNarra Siva Krishna Original Research 03 July 2014 Pages: 86 - 98
Design, synthesis, docking, and biological evaluation of some novel 5-chloro-2-substituted sulfanylbenzoxazole derivatives as anticonvulsant agents Mohamed-Kamal IbrahimKhaled El-AdlHazem A. Mahdy Original Research 03 July 2014 Pages: 99 - 114
Interaction of methotrexate, an anticancer agent, with copper(II) ions: coordination pattern, DNA-cleaving properties and cytotoxic studies Justyna NagajPaulina KołkowskaMałgorzata Jeżowska-Bojczuk Original Research Open access 04 July 2014 Pages: 115 - 123
γ-sitosterol a potent hypolipidemic agent: In silico docking analysis Rangachari BalamuruganAntony StalinJong-Hoon Kim Original Research 05 July 2014 Pages: 124 - 130
Heterocycles 26: synthesis, characterisation, and anticancer activity of some thiazolic chalcones Patrice K. AwoussongValentin ZahariaBonaventure T. Ngadjui Original Research 05 July 2014 Pages: 131 - 141
Synthesis and biological screening of pyrazole moiety containing analogs of podophyllotoxin Basavaiah UmeshaYeriyur Basavaiah BasavarajuChikkamadaiah Mahendra Original Research 05 July 2014 Pages: 142 - 151
Differential effect of 4′-phenylchalcones on acid and alkaline phosphatases Neera RaghavIndu Ravish Original Research 05 July 2014 Pages: 152 - 160
Design and applications of bifunctional cinnamide derivatives as potential antimycobacterial agents with few hepatotoxic effects Zheng-Rong WuDe-Juan ZhiHong-Yu Li Original Research 05 July 2014 Pages: 161 - 170
Green synthesis, antibacterial activity, and SAR of some novel naphthalimides and allylidenes Garima KumariRamendra K. Singh Original Research 05 July 2014 Pages: 171 - 181
Synthesis and biological evaluation of novel d-glucose-derived 1,2,3-triazoles as potential antibacterial and antifungal agents Hui-Zhen ZhangJin-Jian WeiCheng-He Zhou Original Research 05 July 2014 Pages: 182 - 196
Design, synthesis, molecular docking as histone deacetylase (HDAC8) inhibitors, cytotoxicity and antibacterial evaluation of novel 6-(4-(4-aminophenylsulfonyl)phenylamino)-5H-benzo[a]phenoxazin-5-one derivatives P. RavichandiranA. JeganS. Vasanthkumar Original Research 06 July 2014 Pages: 197 - 208
Didanosine phosphoramidates: synthesis, docking to viral NA, antibacterial and antiviral activity Kuruva Chandra SekharS. K. Thaslim BashaS. K. Ghosh Original Research 08 July 2014 Pages: 209 - 219
Structural modification of diarylpyrimidine derivatives as HIV-1 reverse transcriptase inhibitors Shuang-Xi GuYuan-Yuan ZhuChristophe Pannecouque Original Research 08 July 2014 Pages: 220 - 225
Virtual screening-based identification of lead molecules as selective TACE inhibitors Prashant R. MurumkarMayank Kumar SharmaMange Ram Yadav Original Research 10 July 2014 Pages: 226 - 244
Topomer-CoMFA-based predictive modelling on 2,3-diaryl-substituted-1,3-thiazolidin-4-ones as non-nucleoside reverse transcriptase inhibitors Surendra KumarMeena Tiwari Original Research 10 July 2014 Pages: 245 - 257
Synthesis, characterization, and antimicrobial activity of some novel thiazole clubbed 1,3,4-oxadiazoles N. C. DesaiNayan BhattHardik Somani Original Research 10 July 2014 Pages: 258 - 266
POM analyses of anti-kinase activity of thirteen peptide alkaloids extracted from Zizyphus species Moulay H. YoussoufiTaibi Ben HaddaAmmar Bader Original Research 10 July 2014 Pages: 267 - 274
TNFα-induced endothelial activation is counteracted by polyphenol extract from UV-stressed cyanobacterium Arthrospira platensis Pier Francesco FerrariDaniela PalmieriDomenico Palombo Original Research 10 July 2014 Pages: 275 - 282
QSAR models for 1,2,4-benzotriazines as Src inhibitors based on Monte Carlo method Andrey A. ToropovJovana B. VeselinovićAlla P. Toropova Original Research 10 July 2014 Pages: 283 - 290
Letter to the Editor: Quercetin and taxifolin completely break MDM2-p53 association: molecular dynamics simulation study by S. Verma, A. Singh, A. Mishra. Med Chem Res 2013, 22(6) 2778–2787 Anselm H. C. Horn Original Research 10 July 2014 Pages: 291 - 294
Effect of dehydroabietylamine in angiogenesis and GSK3-β inhibition during wound healing activity in rats Mahadevappa ParameshaChapeyil Kumaran RameshJoy Hoskerri Original Research 11 July 2014 Pages: 295 - 303
Synthesis, docking studies, and in silico ADMET predictions of some new derivatives of pyrimidine as potential KSP inhibitors Umer RashidSyed Fahad HassanFarzana Latif Ansari Original Research 11 July 2014 Pages: 304 - 315
Docking-based screening of natural product database in quest for dual site inhibitors of Trypanosoma cruzi trypanothione reductase (TcTR) Debasmita SahaAnuj Sharma Original Research 11 July 2014 Pages: 316 - 333
Synthesis of 3-chloro-4-fluorophenyl-3,4-dichlorophenyl substituted thiocarbamide derivatives as potential antitubercular agents M. Faiz ArshadSuresh KumarNeeraj Upmanyu Original Research 15 July 2014 Pages: 334 - 343
Synthesis, DNA-binding study, and antioxidant activity of 14-aryl-14H-dibenzo[a,j]xanthene derivatives Andivelu IlangovanKarnambaram AnandhanThilagar Sivasudha Original Research 15 July 2014 Pages: 344 - 355
Anti-inflammatory phenolic glycosides from Liparis odorata Yonghui XieSonghua YuBin Li Original Research 15 July 2014 Pages: 356 - 361
New antagonists of toll-like receptor 7 discovered through 3D ligand-based virtual screening Urban ŠvajgerŽiga HorvatStanislav Gobec Original Research 15 July 2014 Pages: 362 - 371
QSPR analysis of some agonists and antagonists of α-adrenergic receptors Piotr KawczakLeszek BoberTomasz Bączek Original Research Open access 15 July 2014 Pages: 372 - 382
Computational analysis of quinoline derivatives as potent topoisomerase-II inhibitors Ankur VaidyaShweta JainRam K. Agrawal Original Research 15 July 2014 Pages: 383 - 393
QSAR and docking analysis of A2B adenosine receptor antagonists based on non-xanthine scaffold Mahboubeh MansourianAfshin FassihiMaryam Abbasi Original Research 15 July 2014 Pages: 394 - 407
Synthesis and pharmacological investigations of novel 2-phenylquinazolin-4(3H)-one derivatives Govindaraj SaravananVeerachamy AlagarsamyPandurangan Dinesh Kumar Original Research 15 July 2014 Pages: 408 - 422
Design and synthesis of N-hydroxytriazole-4-carboxamides as HIV integrase inhibitors Yue-Xia BaiLong-Ji LiLi-Ming Hu Original Research 15 July 2014 Pages: 423 - 429
Long-chain alkyltriazoles as antitumor agents: synthesis, physicochemical properties, and biological and computational evaluation Vanessa Silva GontijoMichael Éder OliveiraRossimiriam Pereira Freitas Original Research 15 July 2014 Pages: 430 - 441
Design, synthesis, and antihypertensive evaluation of 2′-tetrazolyl and 2′-carboxy-biphenylylmethyl-pyrrolidine scaffolds substituted at their N1, C3, and C4 positions as potential angiotensin II AT1 receptor antagonists Mohamed A. H. IsmailMohamed Nabil Aboul-EneinNasser S. M. Ismail Original Research 16 July 2014 Pages: 442 - 458