Imidazole as an anti-epileptic: an overview Rahul MishraSwastika Ganguly Review Article 22 January 2012 Pages: 3929 - 3939
Isoniazid: the magic molecule Vikramjeet JudgeBalasubramanian NarasimhanMunish Ahuja Review Article 24 January 2012 Pages: 3940 - 3957
Modeling VEGFR kinase inhibition of aminopyrazolopyridine urea derivatives using topological and physicochemical descriptors: a quantitative structure activity analysis study Ashutosh Kumar PandeyOmprakash TanwarPiyush Trivedi Original Research 20 December 2011 Pages: 3958 - 3964
Synthesis and in vitro microbiological evaluation of novel 2,4-diaryl-3-azabicyclo[3.3.1]nonan-9,5′-spiro-1′,2′,4′-triazolidine-3′-thiones V. KanagarajanJ. ThanusuM. Gopalakrishnan Original Research 21 December 2011 Pages: 3965 - 3972
Synthesis and antimicrobial activity of novel derivatives of Biginelli pyrimidines Bita SedaghatiAfshin FassihiDaryoush Abedi Original Research 22 December 2011 Pages: 3973 - 3983
Two-dimensional quantitative structure–activity relationship study on polyphenols as inhibitors of α-glucosidase Vesna RastijaDrago BešloSonja Nikolić Original Research 22 December 2011 Pages: 3984 - 3993
Synthesis and in vitro anticancer activities of novel aryl-naphthalene lignans Jie HuiYu ZhaoLi Zhu Original Research 23 December 2011 Pages: 3994 - 4001
Synthesis, characterization and anticancer activity of 3-aza-analogues of DP-7 Jalpa J. BariwalManav MalhotraJitender B. Bariwal Original Research 24 December 2011 Pages: 4002 - 4009
Molecular dynamic and quantum mechanics study of drug recognition for the extremity of DNA G-quadruplex groove Jinlian LiJia FuXiaoqiang Jin Original Research 24 December 2011 Pages: 4010 - 4016
In vitro antibacterial, antifungal, and DNA cleavage studies of coumarin Schiff bases and their metal complexes: synthesis and spectral characterization Sangamesh A. PatilShrishila N. UnkiPrema S. Badami Original Research 24 December 2011 Pages: 4017 - 4027
Brain-targeting research of 10-O-nicotinate ginkgolide B: a new prodrug of ginkgolide B Ze-Yu WuJian PanXiao-Jian Zhou Original Research 24 December 2011 Pages: 4028 - 4036
Simultaneous determination of lisinopril and H2 antagonists in API, formulations and human serum by using two different HPLC systems Safila NaveedNajma SultanaM. Saeed Arayne Original Research 25 December 2011 Pages: 4037 - 4042
α,α-Dibromoacetophenones mediated synthesis of some new 7H-7-alkoxy-3-alkyl/phenyl-6-aryl-s-triazolo[3,4-b][1,3,4]thiadiazines and their antimicrobial evaluation Rashmi PundeerVijay KiranKamal R. Aneja Original Research 25 December 2011 Pages: 4043 - 4052
Amino acid and peptide esters of abacavir: synthesis and activity against human immunodeficiency virus type 1 in cell culture Ivanka StankovaKamelia StanoevaRadka Argirova Original Research 25 December 2011 Pages: 4053 - 4059
In silico screening of indinavir-based compounds targeting proteolytic activity in HIV PR: binding pocket fit approach Chandrabose SelvarajSanjeev Kumar SinghMurugappan Rama Original Research 27 December 2011 Pages: 4060 - 4068
Effects of inositol 1,2,6-triphosphate on human liver cancer SMMC-7721 cells Ya-Min ZhouMou-Cheng WuHong Jiang Original Research 28 December 2011 Pages: 4069 - 4073
Synthesis, DNA affinity, and antimicrobial activity of 4-substituted phenyl-2,2′-bichalcophenes and aza-analogues Magdy M. YoussefMohammed A. Al-OmairMohamed A. Ismail Original Research 29 December 2011 Pages: 4074 - 4082
Combined chemical feature-based assessment and Bayesian model studies to identify potential inhibitors for Factor Xa Meganathan ChandrasekaranSugunadevi SakkiahKeun Woo Lee Original Research 30 December 2011 Pages: 4083 - 4099
In silico and in vitro pharmacological investigations of a natural alkaloid Aimun A. E. AhmedArpad MarkiGeorge Falkay Original Research 30 December 2011 Pages: 4100 - 4107
In vitro antimicrobial and antitubercular studies of novel 6-substituted (pyrrolidin-1-yl)-2(1H)-pyridinones Navin B. PatelRakesh D. SharmaSmita D. Rajani Original Research 30 December 2011 Pages: 4108 - 4119
Coordination of 3-aminoquinoxaline-2-carbonitrile 1,4-dioxides to antimony(III) as a strategy for anti-Trypanosoma cruzi activity improvement Javier VarelaJosane Alves LessaMercedes González Original Research 30 December 2011 Pages: 4120 - 4128
Syntheses, spectral, crystallographic, antimicrobial, and antioxidant studies of few Mannich bases D. TamilvendanS. RajeswariG. Venkatesa Prabhu Original Research 31 December 2011 Pages: 4129 - 4138
Synthesis and antiviral activity of new 3-methyl-1,5-diphenyl-1H-pyrazole derivatives Atif S. TantawyMagda N. A. NasrSamar S. Tawfik Original Research 31 December 2011 Pages: 4139 - 4149
Design, synthesis and biological evaluation of 3-benzylideneflavanone derivatives as cytotoxic agents Shufang HuangYanmei ZhaoXiaowu Dong Original Research 01 January 2012 Pages: 4150 - 4157
Evaluation of antiasthmatic activity of 7,8,9,10-tetrahydroazepino[2,1-b]quinazolin-12(6H)-one in combination with ambroxol in Guinea pigs Mukunda BandeKunal NepaliKanaya Lal Dhar Original Research 01 January 2012 Pages: 4158 - 4167
Antituberculosis and antibacterial evaluations of some novel phenyl pyrazolone-substituted 1h-benzo[g]pyrazolo[3,4-b]quinoline-3-ylamine derivatives Nikhil M. ParekhKalpana C. Maheria Original Research 03 January 2012 Pages: 4168 - 4176
Discovery of 2-(4-cyano-3-trifluoromethylphenyl amino)-4-(4-quinazolinyloxy)-6-piperazinyl(piperidinyl)-s-triazines as potential antibacterial agents Rahul V. PatelPremlata KumariKishor H. Chikhalia Original Research 03 January 2012 Pages: 4177 - 4192
In vitro antimicrobial and molecular docking of dichloro substituted benzoxazole derivatives Rangadhol Vinayak-rao SatyendraKaragadi Anantha-adiga VishnumurthyAnantha-gowda Shruthi Original Research 03 January 2012 Pages: 4193 - 4199
Synthesis and antitumor activities of certain novel 2-amino-9-(4-halostyryl)-4H-pyrano[3,2-h]quinoline derivatives Ahmed M. El-AgrodyEssam Shawky A. E. H. KhattabAbdullah M. Al-Ghamdi Original Research 04 January 2012 Pages: 4200 - 4213
Synthesis and structure–activity relationship of acylthiourea derivatives as inhibitors of microsomal epoxide hydrolase Wei ShenYi FangQing Zhu Original Research 05 January 2012 Pages: 4214 - 4218
Neocryptolepine analogues containing N-substituted side-chains at C-11: synthesis and antischistosomicidal activity Ibrahim El SayedFatem RamzyMostafa M. Abd El-Sattar Original Research 07 January 2012 Pages: 4219 - 4229
Antiproliferative activity and synthesis of 8-prenylnaringenin derivatives by demethylation of 7-O- and 4′-O-substituted isoxanthohumols Mirosław AniołAnna ŚwiderskaAnna Katarzyna Żołnierczyk Original Research Open access 07 January 2012 Pages: 4230 - 4238
Molecular docking, QPLD, and ADME prediction studies on HIV-1 integrase leads Sunil Kumar TripathiChandrabose SelvarajKarnati Konda Reddy Original Research 08 January 2012 Pages: 4239 - 4251
The synthesis, anti-inflammatory and antimicrobial activity evaluation of novel thioanalogs of 3,4-dihydrothiopyrimidin-2(1H)-one derivatives of N-aryl urea Rajesh H. TaleAtish H. RodgeRajendra P. Pawar Original Research 10 January 2012 Pages: 4252 - 4260
GdCl3 promoted synthesis of novel pyrimidine fused indazole derivatives and their anticancer activity T. YakaiahC. KurumurthyB. Sridhar Original Research 11 January 2012 Pages: 4261 - 4273
CytochromeP450 isoenzyme specificity in the metabolism of anti-malarial biguanides: molecular docking and molecular dynamics analyses Dhilon S. PatelM. RameshPrasad V. Bharatam Original Research 11 January 2012 Pages: 4274 - 4289
Two new halocuprates complexes [CuII(1,4,8,11-tetraazacyclotetradecane)][CuICl3] and [H4(1,4,8,11-tetrazacyclotetradecane)][Cu 2 I Cl6]: synthesis, characterizations and biological studies Mohammed LachkarIlham HalimeM. Iqbal Choudhary Original Research 13 January 2012 Pages: 4290 - 4300
Synthesis, anti-microbial evaluation, and QSAR studies of 4-amino-3-hydroxy-naphthalene-1-sulfonic acid derivatives Rajesh KumarPradeep KumarBalasubramanian Narasimhan Original Research 17 January 2012 Pages: 4301 - 4310
Microwave-assisted synthesis, pharmacological evaluation, and QSAR studies of 1,3-diaryl-2-propen-1-ones Shalaka S. VaidyaH. VinayaSupriya S. Mahajan Original Research 18 January 2012 Pages: 4311 - 4323
Antioxidant and α-glucosidase inhibitory compounds from Pimpinella candolleana Wight et Arn. Xing ChangWenyi Kang Original Research 18 January 2012 Pages: 4324 - 4329
Anti-microbial benzimidazole derivatives: synthesis and in vitro biological evaluation Love Kumar SoniTamanna NarsinghaniAnand Sethi Original Research 18 January 2012 Pages: 4330 - 4334
Synthesis, antibacterial, and antitubercular studies of some novel isatin derivatives K. MuraliR. AvinashScott G. Franzblau Original Research 15 January 2012 Pages: 4335 - 4340
Virtual screening of phenylsulfonamido-3-morpholinopropan-2-yl dihydrogen phosphate derivatives as novel inhibitors of MurC–MurF ligases from Mycobacterium leprae Anusuya ShanmugamVenkattappan AnbazhaganJeyakumar Natarajan Original Research 22 January 2012 Pages: 4341 - 4351
Synthesis and blood glucose lowering activity of some novel benzenesulfonylurea derivatives substituted with 6-aryl-4,5-dihyropyridazin-3(2H)-ones Rafia BashirSyed OvaisKalim Javed Original Research 22 January 2012 Pages: 4352 - 4356
Advanced QSRR models of toxicological screening of basic drugs in whole blood by UPLC-TOF–MS Hadi NoorizadehMehrab NoorizadehAbbas Farmany Original Research 26 January 2012 Pages: 4357 - 4368
Synthesis, molecular modeling and anti-inflammatory screening of new 1,2,3-benzotriazinone derivatives Tarek S. IbrahimAdel A. RashadWaleed Barakat Original Research 28 January 2012 Pages: 4369 - 4380
Synthesis, characterization and biological evaluation of some pyridine and quinoline fused chromenone derivatives Mehul A. PatelVarun G. BhilaDinker I. Brahmbhatt Original Research 28 January 2012 Pages: 4381 - 4388
Analysis of carbamazepine serum by differential pulse voltammetry (DPV) and comparison with fluorescence polarization immunoassay (FPIA): an animal study W. Y. LinM. L. PanP. W. Huang Original Research 31 January 2012 Pages: 4389 - 4394
Synthesis and evaluation of some new 4-aminopyridine derivatives as a potent antiamnesic and cognition enhancing drugs Saurabh K. SinhaSushant K. Shrivastava Original Research 02 February 2012 Pages: 4395 - 4402
Synthesis, pharmacological evaluation and molecular docking studies of indanone derivatives Ankur PatelD. GilesAvani Patel Original Research 01 February 2012 Pages: 4403 - 4411