Volume 5, Issue 1

Search all Purinergic Signalling articles

March 2009

Medicinal Chemistry of Purines

Issue Editors:

Kenneth A. Jacobson,
Jeff Zablocki,
Shripad S. Bhagwat

11 articles in this issue

Preface: special issue on medicinal chemistry of purines
Kenneth A. Jacobson
Jeff Zablocki
Shripad Bhagwat
EditorialNotes Open access 05 July 2008 Pages: 1 - 1
Recent improvements in the development of A_2B adenosine receptor agonists
Pier Giovanni Baraldi
Mojgan Aghazadeh Tabrizi
Delia Preti
Review 31 January 2009 Pages: 3 - 19
Progress in the discovery of selective, high affinity A_2B adenosine receptor antagonists as clinical candidates
Rao V. Kalla
Jeff Zablocki
Review Open access 21 June 2008 Pages: 21 - 29
Synthesis and pharmacological characterization of [¹²⁵I]MRS1898, a high-affinity, selective radioligand for the rat A₃ adenosine receptor
Zhan-Guo Gao
Bao Teng
Kenneth A. Jacobson
Original Article Open access 05 June 2008 Pages: 31 - 37
Application of the functionalized congener approach to dendrimer-based signaling agents acting through A_2A adenosine receptors
Yoonkyung Kim
Athena M. Klutz
Kenneth A. Jacobson
Original Article Open access 04 July 2008 Pages: 39 - 50
Allosteric modulation of adenosine receptors
Anikó Göblyös
Ad P. IJzerman
Review Open access 10 July 2008 Pages: 51 - 61
Selective P2X₇ receptor antagonists for chronic inflammation and pain
William A. Carroll
Diana Donnelly-Roberts
Michael F. Jarvis
Review Open access 21 June 2008 Pages: 63 - 73
Development of selective agonists and antagonists of P2Y receptors
Kenneth A. Jacobson
Andrei A. Ivanov
Hyojin Ko
Review Open access 04 July 2008 Pages: 75 - 89
Structure-activity relationships of anthraquinone derivatives derived from bromaminic acid as inhibitors of ectonucleoside triphosphate diphosphohydrolases (E-NTPDases)
Younis Baqi
Stefanie Weyler
Christa E. Müller
Original Article Open access 05 June 2008 Pages: 91 - 106
Kinase inhibitors for the treatment of inflammatory and autoimmune disorders
Shripad S. Bhagwat
Review Open access 21 June 2008 Pages: 107 - 115
Protein and lipid kinase inhibitors as targeted anticancer agents of the Ras/Raf/MEK and PI3K/PKB pathways
Carlos García-Echeverría
Review Open access 04 June 2008 Pages: 117 - 125

Volume 5, Issue 1

Search

Navigation