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Synthesis of 2-arylpyrrolidines by reaction of γ-ureidoacetals with benzene-1,3,5-triol

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Abstract

New 2,2′-(2,4,6-trihydroxybenzene-1,3-diyl)dipyrrolidine derivatives have been synthesized by reaction of benzene-1,3,5-triol (phloroglucinol) with γ-ureidoacetals in the presence of trifluoroacetic acid as catalyst.

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Authors and Affiliations

  1. Arbuzov Institute of Organic and Physical Chemistry, Kazan Scientific Center, Russian Academy of Sciences, ul. Arbuzova 8, Kazan, Tatarstan, 420088, Russia

    A. V. Smolobochkin, A. S. Gazizov, A. R. Burilov & M. A. Pudovik

  2. Kazan Federal University, ul. Kremlevskaya 18, Kazan, Tatarstan, 420008, Russia

    D. G. Khuzyasheva & R. R. Amirov

Authors
  1. A. V. Smolobochkin
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  2. A. S. Gazizov
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  3. A. R. Burilov
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  4. M. A. Pudovik
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  5. D. G. Khuzyasheva
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  6. R. R. Amirov
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Corresponding author

Correspondence to A. S. Gazizov.

Additional information

Original Russian Text © A.V. Smolobochkin, A.S. Gazizov, A.R. Burilov, M.A. Pudovik, D.G. Khuzyasheva, R.R. Amirov, 2016, published in Zhurnal Organicheskoi Khimii, 2016, Vol. 52, No. 4, pp. 552–554.

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Smolobochkin, A.V., Gazizov, A.S., Burilov, A.R. et al. Synthesis of 2-arylpyrrolidines by reaction of γ-ureidoacetals with benzene-1,3,5-triol. Russ J Org Chem 52, 538–540 (2016). https://doi.org/10.1134/S1070428016040102

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  • DOI: https://doi.org/10.1134/S1070428016040102

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