Collection
Special Issue in Honor of Professor Gary L. Grunewald
- Submission status
- Closed
A special issue honoring Professor Gary L. Grunewald for his many contributions and years of service to the field of medicinal chemistry.
Guest edited by Moorthy S. S. Palanki and Michael S. Wolfe
Editors
-
Moorthy S. S. Palanki
Director of the Undergraduate Degree Program in Biotechnology, Professor of Practice in Biotechnology, California State University San Marcos
-
Michael S. Wolfe
Mathias P. Mertes Professor of Medicinal Chemistry, School of Pharmacy, Department of Medicinal Chemistry, University of Kansas
Articles (15 in this collection)
-
-
Special issue of Medicinal Chemistry Research in honor of Professor Gary L. Grunewald
Authors
- Moorthy S. S. Palanki
- Michael S. Wolfe
- Longqin Hu
- Content type: Editorial
- Published: 18 June 2021
- Pages: 1317 - 1320
-
Analogs of the κ opioid receptor antagonist arodyn cyclized by ring-closing metathesis retain κ opioid receptor affinity, selectivity and κ opioid receptor antagonism
Authors
- Wei-Jie Fang
- Thomas F. Murray
- Jane V. Aldrich
- Content type: Original Research
- Published: 17 June 2021
- Pages: 1397 - 1407
-
Thiouracil SecA inhibitors: bypassing the effects of efflux pumps and attenuating virulence factor secretion in MRSA and Bacillus anthracis
Authors (first, second and last of 6)
- Jinshan Jin
- Arpana Chaudhary
- Phang C. Tai
- Content type: Original Research
- Published: 10 June 2021
- Pages: 1341 - 1347
-
Structure–activity relationship investigation of triazole-based kappa opioid receptor agonists
Authors (first, second and last of 6)
- Kevin J. Frankowski
- Tarsis Brust
- Jeffrey Aubé
- Content type: Original Research
- Published: 09 June 2021
- Pages: 1386 - 1396
-
Targeting γ-secretase for familial Alzheimer’s disease
Authors
- Michael S. Wolfe
- Content type: Review Article
- Published: 27 May 2021
- Pages: 1321 - 1327
-
Clathrolides A–B: previously undescribed macrocylic lactones from marine demosponge Clathria (Thalysias) vulpina (Lamarck, 1814) as potential antihypertensive leads attenuating angiotensin converting enzyme
Authors
- Prima Francis
- Kajal Chakraborty
- Content type: Original Research
- Published: 27 May 2021
- Pages: 1438 - 1451
-
Design, synthesis, and antidepressant/anticonvulsant activities of 3H-benzo[f]chromen chalcone derivatives
Authors (first, second and last of 8)
- Qiu-Wan Tan
- Li-Ya He
- Li-Ping Guan
- Content type: Original Research
- Published: 24 May 2021
- Pages: 1427 - 1437
-
Strong in vitro and in vivo cytotoxic effects of two platinum(II) complexes with cryptolepine derivatives
Authors (first, second and last of 7)
- Li-Qin Qin
- Zu-Zhuang Wei
- Hong Liang
- Content type: Original Research
- Published: 22 May 2021
- Pages: 1419 - 1426
-
Synthesis, structure-activity relationship studies and evaluation of a TLR 3/8/9 agonist and its analogues
Authors (first, second and last of 9)
- Anindya Sarkar
- Anushka C. Galasiti Kankanamalage
- Dale L. Boger
- Content type: Original Research
- Published: 18 May 2021
- Pages: 1377 - 1385
-
Synthesis and in vitro activity of oleanolic acid derivatives against Chlamydia trachomatis and Staphylococcus aureus
Authors (first, second and last of 9)
- Oxana Kazakova
- Liudmila Rubanik
- Elmira Khusnutdinova
- Content type: Original Research
- Published: 17 May 2021
- Pages: 1408 - 1418
-
Anti-TB evaluation of novel 2,3-dihydroquinazolin-4(1H)-ones and in silico studies of the active compounds
Authors (first, second and last of 6)
- Apurba Dutta
- Priyanka Trivedi
- Diganta Sarma
- Content type: Original Research
- Published: 15 May 2021
- Pages: 1366 - 1376
-
Design, synthesis, and evaluation of potential carbamate prodrugs of 5′-methylthioadenosine (MTA)
Authors
- Ashwini Sadanand Ranade
- Joseph R. Bertino
- Longqin Hu
- Content type: Original Research
- Published: 29 April 2021
- Pages: 1358 - 1365
-
Sulfamate-tethered aza-Wacker approach towards analogs of Bactobolin A
Authors
- Someshwar Nagamalla
- David K. Johnson
- Shyam Sathyamoorthi
- Content type: Original Research
- Published: 06 April 2021
- Pages: 1348 - 1357
-
Design, synthesis, and biological evaluation of pyrimidine analogs as SecA inhibitors
Authors (first, second and last of 5)
- Fante Bamba
- Jinshan Jin
- Binghe Wang
- Content type: Original Research
- Published: 12 March 2021
- Pages: 1334 - 1340