Design, synthesis, and evaluation of the anticonvulsant and antidepressant activities of pyrido[2,3-d]pyrimidine derivatives Hong-Jian ZhangShi-Ben WangZhe-Shan Quan Original Research 13 May 2016 Pages: 1287 - 1298
Synthesis, characterization and evaluation of antiproliferative activity of diisopropylphenyl esters of fatty acids from selected oils Sathyam Reddy YasaShiva Shanker KakiVijayalakshmi Penumarthy Original Research 13 April 2016 Pages: 1299 - 1307
Synthesis, in vitro and in silico anti-proliferative activity of 4-aryl-4H-chromene derivatives A. ParthibanM. KumaravelH. Surya Prakash Rao Original Research 15 April 2016 Pages: 1308 - 1315
HQSAR and molecular docking studies of furanyl derivatives as adenosine A2A receptor antagonists Camila Muñoz-GutiérrezJulio CaballeroAlejandro Morales-Bayuelo Original Research 15 April 2016 Pages: 1316 - 1328
QSAR studies for some thiazolidine-2,4-dione derivatives as PIM-2 kinase inhibitors Vivek AsatiSanjay K. Bharti Original Research 16 April 2016 Pages: 1329 - 1339
Binding mode of conformations and structure-based pharmacophore development for farnesyltransferase inhibitors N. S. Hari Narayana MoorthySergio F. SousaPedro A. Fernandes Original Research 16 April 2016 Pages: 1340 - 1357
Design, synthesis and anti-acetylcholinesterase evaluation of some new pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine derivatives Anis RomdhaneAbderrahim Ben SaidHichem Ben Jannet Original Research 18 April 2016 Pages: 1358 - 1368
Discovery of highly potent analgesic activity of isopulegol-derived (2R,4aR,7R,8aR)-4,7-dimethyl-2-(thiophen-2-yl)octahydro-2H-chromen-4-ol Ekaterina NazimovaAlla PavlovaNariman Salakhutdinov Original Research 18 April 2016 Pages: 1369 - 1383
Inhibitory effect of 4,4′-[ethane-1,2-diylbis(sulfandiylmethanediyl)]bis(3,5-dimethyl-1H-pyrazole) and its derivatives on alpha-amylase activity Vadim MaksimovRadik ZaynullinAnna Ilyina Original Research 18 April 2016 Pages: 1384 - 1389
Synthesis of new benzimidazole and phenylhydrazinecarbothiomide hybrids and their anticonvulsant activity Nadeem SiddiquiMd. Shamsher AlamOzair Alam Original Research 19 April 2016 Pages: 1390 - 1402
A facile synthesis and neuroprotective role of novel quinoxaline-2,3-bis hydrazones in ethidium bromide-induced demyelinated rats Gayathri RajamanickamJubie SelvarajThirumurthy Rajendran Original Research 19 April 2016 Pages: 1403 - 1410
In silico molecular docking of niloticin with acetylcholinesterase 1 (AChE1) of Aedes aegypti L. (Diptera: Culicidae): a promising molecular target Appadurai Daniel ReeganAntony StalinNaif Abdullah Al-Dhabi Original Research 19 April 2016 Pages: 1411 - 1419
Synthesis and anticonvulsant activities of functionalized 5-(isoindole-1,3-dione)-pyrimidinones Rashmi SharmaDinesh Y. GawandeRajesh Kumar Goel Original Research 19 April 2016 Pages: 1420 - 1424
Synthesis and potential anticonvulsant activity of new aryl sulfonyl semicarbazide derivatives Yousong NieMin ZhongXianran He Original Research 21 April 2016 Pages: 1425 - 1432
Formylchromone derivatives as novel and selective PTP-1B inhibitors: a drug design aspect using molecular docking-based self-organizing molecular field analysis Sant K. VermaSuresh Thareja Original Research 22 April 2016 Pages: 1433 - 1467
Piroxicam sulfonates biology-oriented drug synthesis (BIODS), characterization and anti-nociceptive screening Safi UllahMuhammad SaeedShahnaz Perveen Original Research 25 April 2016 Pages: 1468 - 1475
Identification and antioxidant of polyhydroxylated naphthoquinone pigments from sea urchin pigments of Echinometra mathaei Soolmaz SoleimaniMorteza YousefzadiNarges Amrollahi Bioki Original Research 27 April 2016 Pages: 1476 - 1483
Synthesis and characterization of novel conjugates of 4-[3-(aryl/heteroaryl)-3-oxo-propenyl]-benzaldehyde with thiazole and thiazolidinones as possible voltage-gated sodium channel blockers Sundeep PandeyPankaj K. SonarShailendra K. Saraf Original Research 27 April 2016 Pages: 1484 - 1496
Design, synthesis of new chiral fluorine-containing β-hydroxysulfonamides from natural amino acids and study of their anti-inflammatory and analgesic activities Monia GloulouJamil KraïemMohamed Kallel Original Research 30 April 2016 Pages: 1497 - 1506
Design, synthesis and evaluation of acridin-9-yl hydrazide derivatives as BACE-1 inhibitors Priti JainPankaj K. WadhwaHemant R. Jadhav Original Research 30 April 2016 Pages: 1507 - 1513