Generic Anti-PEG Antibody Assay on ProterixBio’s (Formerly BioScale) ViBE Platform Shows Poor Reproducibility Shannon D. ChilewskiJulie ShieldsHeather Myler Brief/Technical Note 24 April 2018 Article: 65
Feasibility of Exposure-Response Analyses for Clinical Dose-Ranging Studies of Drug Combinations Theodoros PapathanasiouAnders StratheRune Viig Overgaard Research Article 23 April 2018 Article: 64
Investigation of the Mechanism of Therapeutic Protein-Drug Interaction Between Methotrexate and Golimumab, an Anti-TNFα Monoclonal Antibody Weirong WangJocelyn LeuHonghui Zhou Research Article 17 April 2018 Article: 63
Equivalence Testing of Complex Particle Size Distribution Profiles Based on Earth Mover’s Distance Meng HuXiaohui JiangRobert Lionberger Research Article 12 April 2018 Article: 62
Evaluation of 4β-Hydroxycholesterol and 25-Hydroxycholesterol as Endogenous Biomarkers of CYP3A4: Study with CYP3A-Humanized Mice Shin-ichiro NittaMari HashimotoKaoru Kobayashi Research Article 09 April 2018 Article: 61
Dissolution and Translational Modeling Strategies Enabling Patient-Centric Drug Product Development: the M-CERSI Workshop Summary Report Andreas AbendTycho HeimbachSandra Suarez-Sharp Meeting Report 09 April 2018 Article: 60
Computational Fragment-Based Drug Design: Current Trends, Strategies, and Applications Yuemin BianXiang-Qun (Sean) Xie Review Article 09 April 2018 Article: 59
Deep Learning for Drug Design: an Artificial Intelligence Paradigm for Drug Discovery in the Big Data Era Yankang JingYuemin BianXiang-Qun Sean Xie Review Article 30 March 2018 Article: 58
Measuring the Impact of Gastrointestinal Variables on the Systemic Outcome of Two Suspensions of Posaconazole by a PBPK Model Bart HensArjang TalattofGordon L. Amidon Research Article 29 March 2018 Article: 57
Comparison of Model Averaging and Model Selection in Dose Finding Trials Analyzed by Nonlinear Mixed Effect Models Simon BuatoisSebastian UeckertFrance Mentré Research Article 29 March 2018 Article: 56
Correction to: Model-Based Adaptive Optimal Design (MBAOD) Improves Combination Dose Finding Designs: an Example in Oncology Philippe B. PierrillasSylvain FouliardMats O. Karlsson Correction 27 March 2018 Article: 55
Improved Prediction of Blood–Brain Barrier Permeability Through Machine Learning with Combined Use of Molecular Property-Based Descriptors and Fingerprints Yaxia YuanFang ZhengChang-Guo Zhan Research Article 21 March 2018 Article: 54
Development of Fc-Fused Cocaine Hydrolase for Cocaine Addiction Treatment: Catalytic and Pharmacokinetic Properties Xiabin ChenJing DengFang Zheng Research Article 19 March 2018 Article: 53
PharmTeX: a LaTeX-Based Open-Source Platform for Automated Reporting Workflow Christian Hove RasmussenMike K. SmithTimothy Nicholas Research Article 16 March 2018 Article: 52
Detection of Memory B Activity Against a Therapeutic Protein in Treatment-Naïve Subjects Karen LiaoStacy DerbyshireGeorge R. Gunn Research Article 16 March 2018 Article: 51
Therapeutic Potential of Engineered Extracellular Vesicles Kyle I. MentkowskiJonathan D. SnitzerJennifer K. Lang Review Article Open access 15 March 2018 Article: 50
Selection of a Ligand-Binding Neutralizing Antibody Assay for Benralizumab: Comparison with an Antibody-Dependent Cell-Mediated Cytotoxicity (ADCC) Cell-Based Assay Yuling WuAhmad AkhgarLorin K. Roskos Research Article Open access 14 March 2018 Article: 49
A Minimal Physiologically Based Pharmacokinetic Model with a Nested Endosome Compartment for Novel Engineered Antibodies Dongfen YuanFrederik RodeYanguang Cao Research Article 14 March 2018 Article: 48
Towards Bridging Translational Gap in Cardiotoxicity Prediction: an Application of Progressive Cardiac Risk Assessment Strategy in TdP Risk Assessment of Moxifloxacin Nikunjkumar PatelOliver HatleySebastian Polak Research Article Open access 14 March 2018 Article: 47
Why Drugs Fail in Late Stages of Development: Case Study Analyses from the Last Decade and Recommendations Dolly A. ParasrampuriaLeslie Z. BenetAmarnath Sharma Commentary 13 March 2018 Article: 46
A Simple Approach to Determine a Curve Fitting Model with a Correct Weighting Function for Calibration Curves in Quantitative Ligand Binding Assays Yuhong XiangJean DonleyBoris Gorovits Research Article 13 March 2018 Article: 45