Synthesis and biological evaluation of imidazo[1,2-\({{\varvec{b}}}\)]pyridazines as inhibitors of TNF-\({\varvec{\upalpha }}\) production Shivaji S. PanditMahesh R. KulkarniNitin P. Lad Original Article 02 December 2017 Pages: 545 - 560
Synthesis of functionalized dihydro-2-oxopyrroles using graphene oxide as heterogeneous catalyst Masoumeh BavadiKhodabakhsh Niknam Original Article 09 January 2018 Pages: 561 - 573
Structural insights of dipeptidyl peptidase-IV inhibitors through molecular dynamics-guided receptor-dependent 4D-QSAR studies Rajesh B. PatilEuzebio G. BarbosaSanjay D. Sawant Original Article 13 March 2018 Pages: 575 - 583
The influence of substituents on the reactivity and cytotoxicity of imidazothiazolotriazinones Galina A. GazievaAlexei N. Izmest’evAngelina N. Kravchenko Original Article 14 March 2018 Pages: 585 - 599
One-pot solvent-free three-component reaction between primary amines, carbon disulfide, and 5-alkylidene rhodanines: a convenient synthesis of asymmetric birhodanines Farough NasiriParisa Nazari Original Article 15 March 2018 Pages: 601 - 608
One-pot three-component synthesis and oxidation of functionalized tetrahydrobenzo[d]pyrrolo[2,1-b]thiazoles Gong JinJing SunChao-Guo Yan Original Article 19 March 2018 Pages: 609 - 626
High diastereoselective amine-catalyzed Knoevenagel–Michael-cyclization–ring-opening cascade between aldehydes, 3-arylisoxazol-5(4H)-ones and 3-aminocyclohex-2-en-1-ones Anatoly N. VereshchaginMichail N. ElinsonMikhail P. Egorov Original Article 20 March 2018 Pages: 627 - 636
Antibacterial and antiproliferative activity of novel 2-benzimidazolyl- and 2-benzothiazolyl-substituted benzo[b]thieno-2-carboxamides Maja CindrićMihaela PerićMarijana Hranjec Original Article 20 March 2018 Pages: 637 - 646
Insect growth regulatory activity of carvacrol-based 1,3,4-thiadiazoles and 1,3,4-oxadiazoles Suresh D. BagulJamatsing D. RajputRatnamala S. Bendre Original Article 23 March 2018 Pages: 647 - 655
Synthesis and antimicrobial evaluation of novel 1,2,4-triazole thioether derivatives bearing a quinazoline moiety Zhijiang FanJun ShiXiaoping Bao Original Article 24 March 2018 Pages: 657 - 667
Probing the opportunities for designing anthelmintic leads by sub-structural topology-based QSAR modelling Prabodh RanjanMohd AtharKari Vijaya Krishna Original Article 02 April 2018 Pages: 669 - 683
A practical multi-step synthesis of ethyl N-functionalized \(\varvec{\upbeta }\)-amino benzimidazole acrylate derivatives as promising cytotoxic agents Christelle N’Ta AmbeuRémy Le GuévelJean-Pierre Bazureau Original Article 05 April 2018 Pages: 685 - 708
An efficient protocol for the synthesis of highly sensitive indole imines utilizing green chemistry: optimization of reaction conditions Bushra NisarSyeda Laila RubabMuhammad Nawaz Tahir Original Article 11 April 2018 Pages: 709 - 722
Eco-friendly synthesis, in vitro anti-proliferative evaluation, and 3D-QSAR analysis of a novel series of monocationic 2-aryl/heteroaryl-substituted 6-(2-imidazolinyl)benzothiazole mesylates Livio RacanéLucija PtičekGrace Karminski-Zamola Original Article 17 April 2018 Pages: 723 - 741
Microwave-assisted green synthesis of 4,5-dihydro-1H-pyrazole-1-carbothioamides in water Hamid Reza FarmaniMohammad Hossein MossleminBahareh Sadeghi Short Communication 31 March 2018 Pages: 743 - 749
Current progress in asymmetric Biginelli reaction: an update Majid M. HeraviRazieh MoradiBorzou Moradi Comprehensive Review 23 June 2018 Pages: 751 - 767