3-Aryl-1-(3-nitrophenyl)triazenes were obtained in the cyclization reaction of diazotized 3-nitroaniline with arylamines in the presence of dimethyl sulfoxide and potassium carbonate to give 1-aryl-5-nitrobenzotriazoles.
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M. D. Mashkovskii, Drugs [in Russian], Novaya Volna, Moscow (2008).
B. D. Palmer, J. B. Smaill, M. Boyd, D. H. Boschelli, A. M. Doherty, J. M. Hamby, S. S. Khatana, J. B. Kramer, A. J. Kraker, R. L. Panek, G. H. Lu, T. K. Dahring, R. T. Winters, H. D. H. Showalter, and W. A. Denny, J. Med. Chem., 41, 5457 (1998).
N. Mishra, P. Arora, B. Kumar, L. C. Mishra, A. Bhattacharya, S. K. Awasthi, and V. K. Bhasin, Eur. J. Med. Chem., 43, 1530 (2008).
H. Wamhoff, in: A. R. Katritzky and C. W. Rees (editors), Comprehensive Heterocyclic Chemistry, Vol. 5, Pergamon Press, Oxford (1984), p. 722.
V. Zimmermann and S. Bräse, J. Comb. Chem., 9, 11 (2007).
L. M. Gornostaev and N. A. Bulgakova, Zh. Org. Khim., 37, 1416 (2001).
T. Čimbora-Zovko, A. Brozovic, I. Piantanida, G. Fritz, A. Virag, B. Alić, V. Majce, M. Kočevar, M. Polanc, and M. Osmak, Eur. J. Med. Chem., 46, 2971 (2011).
Weygand-Hilgetag, Experimental Methods in Organic Chemistry [Russian translation], Khimiya, Moscow (1968), p. 320.
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*A similar paper by the authors Z. Zhou, Q.-L. Liu, W. Li, and Y.-M. Zhu was published in Heterocycles, 83, 2057 (2011). The Editors decided to publish this paper by the Russian authors in Chemistry of Heterocyclic Compounds because it was submitted earlier.
Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 9, pp. 1375-1378, September, 2013.
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Gornostaev, L.M., Bulgakova, N.A. & Kalashnikova, I.V. Synthesis of 1-Aryl-5-Nitrobenzotriazoles*. Chem Heterocycl Comp 49, 1281–1284 (2013). https://doi.org/10.1007/s10593-013-1376-0
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DOI: https://doi.org/10.1007/s10593-013-1376-0