Abstract
Methods for the synthesis of 2-ethynylaziridines by the cycloaddition of carbene to an α-ethynyl imine, cyclization of acetylenic β-amino alcohols in the presence of triphenylphosphine, and by means of the Gabriel reaction were developed.
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Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 2, pp. 184–187, February, 1984.
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Shubina, Y.V., Tikhomirov, D.A. & Eremeev, A.V. 2-Ethynylaziridines. Chem Heterocycl Compd 20, 147–150 (1984). https://doi.org/10.1007/BF00506283
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DOI: https://doi.org/10.1007/BF00506283