Abstract
N-(3-Thietanyl)-substituted heterocycles are formed in the alkylation of xanthine and benzimidazole derivatives with epithiochlorohydrin (ETCH) in an aqueous medium as a consequence of a thiirane—thietane rearrangement.
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Literature Cited
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Fifteenth Anniversary of the All-Union Lenin Young Communist League, Bashkir State Medical Institute, Ufa 450000. Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 4, pp. 516–518, April, 1991.
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Khaliuliin, F.A., Kataev, V.A. & Strokin, Y.V. Alkylation of xanthine and benzimidazole derivatives with epithiochlorohydrin. Chem Heterocycl Compd 27, 410–412 (1991). https://doi.org/10.1007/BF00480840
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DOI: https://doi.org/10.1007/BF00480840