Abstract
A convenient route to 9-(β-aminoethyl)isoalloxazines is offered, based on monoacetylethylenediamine. 6-Chloro-7-methyl-9-(β-aminoethyl)-isoalloxazine is used to synthesize some acyl derivatives and azomethines, among them some with the bis(β-chloroethyl)amino group, for biological testing.
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For Part II see [10].
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Petrova, L.F., Pushkareva, Z.V. & Vavilov, G.A. Research on isoalloxazine derivatives. Chem Heterocycl Compd 3, 734–736 (1967). https://doi.org/10.1007/BF00468362
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DOI: https://doi.org/10.1007/BF00468362