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Synthesis of peptide conjugates of mestranol by a 1,3-dipolar cycloaddition click reaction

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Chemistry of Heterocyclic Compounds Aims and scope

An efficient method is presented for the synthesis of a series of peptide conjugates of the ethynylestradiol 3-methyl ether and the corresponding azidopeptides by a copper(I)-catalyzed 1,3-di-polar cycloaddition click reaction.

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Authors and Affiliations

  1. M. V. Lomonosov Moscow State University, 1 Build. 3 Leninskie Gory, Moscow, 119991, Russia

    N. V. Sokolova & V. G. Nenajdenko

Authors
  1. N. V. Sokolova
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  2. V. G. Nenajdenko
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Correspondence to V. G. Nenajdenko.

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Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 6, pp. 972-976, June, 2012.

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Sokolova, N.V., Nenajdenko, V.G. Synthesis of peptide conjugates of mestranol by a 1,3-dipolar cycloaddition click reaction. Chem Heterocycl Comp 48, 903–906 (2012). https://doi.org/10.1007/s10593-012-1074-3

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  • DOI: https://doi.org/10.1007/s10593-012-1074-3

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