The emerging role of proteolysis targeting chimeras (PROTACs) in the treatment of Alzheimer’s disease Namy GeorgeMd. Jawaid AkhtarShah Alam Khan Review Article 09 February 2023 Pages: 601 - 616
Recent advances on biologically active coumarin-based hybrid compounds Metin YildirimSamet PoyrazMehmet Ersatir Review Article 09 February 2023 Pages: 617 - 642
Baicalein—A review on its molecular mechanism against breast cancer and delivery strategies Shraddha SrivastavaJose MathewAvinash chandra Pandey Review Article 02 March 2023 Pages: 643 - 658
Recent updates on thienopyrimidine derivatives as anticancer agents Menna Tallah M. SayedRasha A. HassanAfaf K. El-Ansary Review Article Open access 02 March 2023 Pages: 659 - 681
Screening a small hydrazide-hydrazone combinatorial library for targeting the STAT3 in monocyte-macrophages with insulated reporter transposons Valeri V. MossineSteven P. KelleyThomas P. Mawhinney Original Research Open access 13 February 2023 Pages: 682 - 693
Synthesis of nitrogen-containing oleanolic acid derivatives as carbonic anhydrase and acetylcholinesterase inhibitors Halil ŞenolGurbet Çelik TurgutGülaçtı Topçu Original Research 13 February 2023 Pages: 694 - 704
Design, synthesis and anti-breast cancer properties of butyric ester tethered dihydroartemisinin-isatin hybrids Shijia ZhaoXiaoyan ZhangZhi Xu Original Research 14 February 2023 Pages: 705 - 712
Design, synthesis and α-glucosidase inhibition study of novel pyridazin-based derivatives Loghman FiroozpourFaraz Kazemzadeh ArasiAlireza Foroumadi Original Research 15 February 2023 Pages: 713 - 722
Synthesis, α-glucosidase inhibitory activity, and molecular docking of cinnamamides Nur Pasca AijijiyahFirst Ambar WatiMardi Santoso Original Research 16 February 2023 Pages: 723 - 735
Antibacterial, antifungal activities and toxicity of new synthetic fatty acid salicylate esters Monique B. EwonkemPascaline M. DeussomDuplex J. Wansi Original Research 20 February 2023 Pages: 736 - 748
Synthesis, antitumor activities and functional mechanism of purine derivatives harboring phenyl moieties through three carbon bridges Chao TianYifei ChenZhili Zhang Original Research 24 February 2023 Pages: 749 - 763
Novel imino-thiazoloquinoxaline derivatives against renal cell carcinoma: less radiation-damaging approach Nashwa H. ZaherReham M. M. El-HazekNoha A. Fadel Original Research Open access 24 February 2023 Pages: 764 - 776