Progress on biphenyl derivatives as PD-1/PD-L1 inhibitors Shurong WangYuli WangHong Yan Review Article 29 August 2023 Pages: 2089 - 2115
Design, synthesis and antitumor activity evaluation of 5-cyano-2,4,6-substituted pyrimidine derivatives containing acrylamide group Fuqiang YuLingling ChiQiurong Zhang Original Research 07 July 2023 Pages: 2116 - 2124
Design, synthesis and antitumor activity evaluation of pyrimidine derivatives containing 4-hydroxypiperidine group Lingling ChiHao WangQiurong Zhang Original Article 07 July 2023 Pages: 2125 - 2137
Design, synthesis and antitumor activity evaluation of tetrasubstituted pyrimidine derivatives containing methyl phenyl sulfone group Chao GaoFuqiang YuQiurong Zhang Original Research 12 July 2023 Pages: 2138 - 2155
Design, synthesis and antitumor activity evaluation of 4,6,7-trisubstituted quinazoline derivatives containing benzothiazole moiety Fuqiang YuYing XuQiurong Zhang Original Research Article 13 July 2023 Pages: 2156 - 2167
A new cadinane sesquiterpenoid from Eupatorium adenophorum and α-glycosidase and AChE inhibitory activities of a gossypetin acylglucoside Minh Giang PhanNgoc Phuc DongHideaki Otsuka Original Research Article 15 July 2023 Pages: 2168 - 2175
Design, synthesis and antitumor activity evaluation of 2,4,6-trisubstituted quinazoline derivatives containing piperidine moiety Honglin DaiFuqiang YuQiurong Zhang Original Research Article 15 July 2023 Pages: 2176 - 2195
Discovery of deguelin derivatives in combination with fluconazole against drug-resistant Candida albicans Biaoqi LiuYouwei WuRuihan Zhang Original Research Article 24 July 2023 Pages: 2196 - 2207
Using molecular networking and docking to explore arginase inhibitors among Drimys brasiliensis chemical constituents Léia da C. MendesThais B. Vieira DantasLorena R. F. de Sousa Original Research Article 24 July 2023 Pages: 2208 - 2218
Synthesis of amide warhead containing coumarin derivatives as potential pancreatic lipase inhibitors: in silico and in vitro evaluation for obesity treatment Nisha YadavAtish T. Paul Original Research Article 28 July 2023 Pages: 2219 - 2233
Synthesis of 2-amino-4H-chromenes catalyst-free via sequential Knoevenagel-Michael reaction and evaluation of biological activity in tumor cells Poliana Gomes de AbrantesPaloma Gomes de AbrantesJuliana Alves Vale Original Research Article 04 August 2023 Pages: 2234 - 2244
Structure activity relationship (SAR) driven design and discovery of WCK 5107 (Zidebactam): novel β-lactam enhancer, potent against multidrug-resistant gram-negative pathogens Satish BhavsarSanjeev JoshiMahesh Patel Original Research Article 09 August 2023 Pages: 2245 - 2255
Synthesis of indole-based ferulic acid derivatives and in vitro evaluation of antiviral activity against SARS-CoV-2 Marina Mol S. A. VerzolaDaisymara Priscila de Almeida MarquesRenata Barbosa de Oliveira Original Research Article 10 August 2023 Pages: 2256 - 2267
Correction: Stable isotope applications in drug development and the elucidation of mechanisms of drug metabolism Rheem A. TotahAllan E. Rettie Correction 16 September 2023 Pages: 2268 - 2268