Synthesis and antitumor activity of novel silibinin and 2,3-dehydrosilybin derivatives with carbamate groups Qiuchan WuJiang ZengJinfu Dong Original Research 15 February 2022 Pages: 533 - 544
Discriminative stimulus effects of an imidazolidine-derived appetite suppressant Richard Young Original Research 16 February 2022 Pages: 545 - 554
Design, synthesis, and LFA-1/ICAM-1 antagonist activity evaluation of Lifitegrast analogues Guoxin DuWeiwei DuDonglei Zhang Original Research 17 February 2022 Pages: 555 - 579
Synthesis and biological evaluations of novel pyrazinoic acid derivatives as anticancer agents Shiva AkhlaghiAzar MostoufiMasood Fereidoonnezhad Original Research 19 February 2022 Pages: 580 - 593
Design and synthesis of novel pyrazolopyrimidine-based derivatives as reversible BTK inhibitors with potent antiproliferative activity in mantle cell lymphoma Fansheng RanYang LiuGuisen Zhao Original Research 23 February 2022 Pages: 594 - 604
Synthesis and anticancer activity of Boc-Gly-Pro dipeptide-annonaceous acetogenin prodrugs targeting fibroblast activation protein or other hydrolytic enzymes Jing-Fang ShiPing WuZi-Hua Jiang Original Research 24 February 2022 Pages: 605 - 616
Synthesis and analgesic potential of 4-[4–chloro-3- (trifluoromethyl)-phenyl]-4-piperidinol analogues against pain model in mice Shazia HaiderZafar Saied SaifyNasreen Begum Original Research 24 February 2022 Pages: 617 - 627
Synthesis, antifungal activity, and molecular dynamics study of novel geranyl aromatic sulfonamide compounds as potential complex III inhibitors Xinning SongZhiyang JiangHongxia Duan Original Research 02 March 2022 Pages: 628 - 642
Review of 3D templates for in silico homology models of MATs: improved 3D model of hDAT Charles B. JonesMałgorzata Dukat Original Research 03 March 2022 Pages: 643 - 651
Design, synthesis and biological evaluation of 8-aminoquinoline-1,2,3-triazole hybrid derivatives as potential antimicrobial agents Fatma AlbayrakMustafa ÇiçekIrem Kulu Original Research 07 March 2022 Pages: 652 - 665
Anti-tumor metabolites from Synadenium grantii Hook F. Lujun LiQingya ZouPaul W. Paré Original Research 08 March 2022 Pages: 666 - 673
Correction to: Discriminative stimulus effects of an imidazolidine-derived appetite suppressant Richard Young Correction 15 March 2022 Pages: 674 - 675