Towards the design of 3-aminopyrazole pharmacophore of pyrazolopyridine derivatives as novel antioxidants Apilak WorachartcheewanChanin NantasenamatVirapong Prachayasittikul Original Research 30 June 2017 Pages: 2699 - 2706
Discovery two potent and new inhibitors of 15-lipoxygenase: (E)-3-((3,4-dihydroxybenzylidene) amino)-7-hydroxy-2H-chromen-2-one and (E)-O-(4-(((7-hydroxy-2-oxo-2H-chromen-3-yl) imino)methine) phenyl)dimethylcarbamothioate Carolina NuñezNicole MoralesAngelica Fierro Original Research 07 July 2017 Pages: 2707 - 2717
Design, synthesis, and docking studies of new 2-benzoxazolinone derivatives as anti-HIV-1 agents Mahdieh SafakishZahra HajimahdiAfshin Zarghi Original Research 03 July 2017 Pages: 2718 - 2726
Involvement of reactive oxygen species in the oleoylethanolamide effects and its pyrazonilic analogue in melanoma cells Priscila Antiqueira-SantosDaiane S. dos SantosAna Paula S. Votto Original Research 01 July 2017 Pages: 2727 - 2736
Synthesis and evaluation of 2,3-indolotriterpenoids as new α-glucosidase inhibitors Elmira F. KhusnutdinovaIrina E. SmirnovaDo Quoc Viet Original Research 07 July 2017 Pages: 2737 - 2742
Phytochemical characterization and biological activity of secondary metabolites from three Limonium species Anastassiya V. GadetskayaShaymaa M. MohamedSamir A. Ross Original Research 12 July 2017 Pages: 2743 - 2750
RETRACTED ARTICLE: Rhodozepinone, a new antitrypanosomal azepino-diindole alkaloid from the marine sponge-derived bacterium Rhodococcus sp. UA13 Yasmin ElsayedJohn RefaatMostafa A. Fouad Original Research 15 July 2017 Pages: 2751 - 2760
Prenyl-flavonoids from Epimedium koreanum Nakai and their soluble epoxide hydrolase and tyrosinase inhibitory activities Xiang Dong SuWei LiYoung Ho Kim Original Research 31 August 2017 Pages: 2761 - 2767
Docking-based comparative intermolecular contacts analysis and in silico screening reveal new potent acetylcholinesterase inhibitors Maha HabashSawsan AbuhamdahMutasem O. Taha Original Research 11 July 2017 Pages: 2768 - 2784
Design, synthesis, estrogenic and antiestrogenic activities of some triarylpyrazole derivatives Mahmoud A. RagabHeba A. Abd El RazikNargues S. Habib Original Research 19 July 2017 Pages: 2785 - 2808
Choline kinase inhibition and docking studies of a series of 6-(benzylthio)-9H-purin-9-yl-pyridinium derivatives Belén Rubio-RuizPablo Ríos-MarcoAntonio Entrena Original Research 11 July 2017 Pages: 2809 - 2815
Liuweibuqi capsules suppress inflammation by affecting T cell polarization and survival in chronic obstructive pulmonary disease Chengyang WangHuanzhang DingLei Gan Original Research 13 July 2017 Pages: 2816 - 2823
Structure-based rational design of peptide inhibitors to disrupt the recognition and interaction between hepatitis B virus large envelope protein and human hepatocyte receptor γ2-adaptin Kuifeng WangChunying YangJiansheng Zhu Original Research 19 July 2017 Pages: 2824 - 2831
Design, synthesis, and biological evaluation of 4-H pyran derivatives as antimicrobial and anticancer agents Thatikonda Narendar ReddyMettu RavinderVaidya Jayathirtha Rao Original Research 17 July 2017 Pages: 2832 - 2844
Bioguided study of the in vitro parasitocidal effect on adult Hymenolepis nana of the Psidium sartorianum (O. Berg Nied.) fruit methanol extract Julio Montes-AvilaSylvia Páz Díaz-CamachoFrancisco Delgado-Vargas Original Research 19 July 2017 Pages: 2845 - 2852
Antiproliferative effect of apocynin in cervical epithelial cells infected by HPV 16 involves change of ROS production and cell cycle Natália Alves LimaNatália de Carvalho Scharf SantanaSueli de Oliveira Silva Original Research 19 July 2017 Pages: 2853 - 2860
Synthesis, cytotoxicity and pro-apoptosis activity of isoquinoline quinones Hua NiChao XiaYu Zhao Original Research 19 July 2017 Pages: 2861 - 2869
PTP1B inhibitory and cytotoxic activities of triterpenoids from the aerial parts of Agrimonia pilosa Bing Tian ZhaoDuc Hung NguyenMi Hee Woo Original Research 20 July 2017 Pages: 2870 - 2878
Design, synthesis and biological evaluation of urea-based benzamides derivatives as HDAC inhibitors Yong ZhuXin ChenWeifang Tang Original Research 26 July 2017 Pages: 2879 - 2888
Synthesis, antimycobacterial screening and molecular docking studies of 4-aryl-4′-methyl-2′-aryl-2,5′-bisthiazole derivatives Yogita K. AbhaleAbhijit D. ShindePravin C. Mhaske Original Research 21 July 2017 Pages: 2889 - 2899
Isolation of three new metabolites and intervention of diazomethane led to separation of compound 1 & 2 from an endophytic fungus, Cryptosporiopsis sp. depicting cytotoxic activity Sunil KumarYedukondalu NalliAsif Ali Original Research 28 July 2017 Pages: 2900 - 2908
Synthesis and biological evaluation of pyrazolo[1,5-a]pyrimidine-3-carboxamide as antimicrobial agents Ashraf S. HassanDoaa M. MasoudAhmed A. Askar Original Research 21 July 2017 Pages: 2909 - 2919
The effects of flavonoid compound from Agrimonia pilosa Ledeb on promotting 3T3-L1 preadipocytes differentiation by activating PPARγ partially Liancai ZhuJun TanBochu Wang Original Research 05 August 2017 Pages: 2920 - 2928
Imatinib derivatives as inhibitors of K562 cells in chronic myeloid leukemia Liviane D. AzevedoMônica M. BastosNubia Boechat Original Research 04 September 2017 Pages: 2929 - 2941
Antiacetylcholinesterase activity and docking studies with chlorogenic acid, cynarin and arzanol from Helichrysum stoechas (Lamiaceae) Letícia SilvaAna Margarida RodriguesMaria Luísa Marques Serralheiro Original Research 29 July 2017 Pages: 2942 - 2950
Design, synthesis and CoMFA studies of OEA derivatives as FAAH inhibitors Daxiong HanBiyan WangMeimei Chen Original Research 31 July 2017 Pages: 2951 - 2966
Quinoxalin-2(1H)-one derived AMPA-receptor antagonists: Design, synthesis, molecular docking and anticonvulsant activity Abdel-Ghany A. El-HelbyRezk R. A. AyyadAlaa Elwan Original Research 04 August 2017 Pages: 2967 - 2984
Design and synthesis of novel triazole linked pyrrole derivatives as potent Mycobacterium tuberculosis inhibitors M. Lakshmi DeviP. Lakshmi ReddyR. Narender Original Research 05 September 2017 Pages: 2985 - 2999
Identification of potential type 4 cAMP phosphodiesterase inhibitors via 3D pharmacophore modeling, virtual screening, DFT and structural bioisostere design Dhrubajyoti GogoiAmrita K. ChalihaAlak K. Buragohain Original Research 09 August 2017 Pages: 3000 - 3014
Novel L-arginine derivatives as aminopeptidase N inhibitors: design, chemistry, and pharmacological evaluation Jiajia MouYepeng LuanQiang Wang Original Research 16 August 2017 Pages: 3015 - 3025
Analgesic, anti-inflammatory, and antimicrobial activities of novel isoxazole/pyrimidine/pyrazole substituted benzimidazole analogs Krishna Veni ChikkulaRaja Sundararajan Original Research 09 August 2017 Pages: 3026 - 3037
Synthesis and preliminary assessment of the anticancer and Wnt/β-catenin inhibitory activity of small amide libraries of fenamates and profens Bini MathewJudith V. HobrathRobert C. Reynolds Original Research Open access 05 August 2017 Pages: 3038 - 3045
Synthesis, in vitro evaluation of antibacterial, antifungal and larvicidal activities of pyrazole/pyridine based compounds and their nanocrystalline MS (M = Cu and Cd) derivatives Gopinath MondalHarekrishna JanaPulakesh Bera Original Research 24 August 2017 Pages: 3046 - 3056
Synthesis and neuroprotective activity of novel 1,2,4-triazine derivatives with ethyl acetate moiety against H 2 O2 and Aβ-induced neurotoxicity Tuba Tuylu KucukkilincKamaledin Safari YanghaghHamid Irannejad Original Research 04 August 2017 Pages: 3057 - 3071
Erratum to: Synthesis and characterization of new s-triazine bearing benzimidazole and benzothiazole derivatives as anticancer agents G. Jagadeesh KumarS. Naveen KumarV. Jayathirtha Rao Erratum 17 July 2017 Pages: 3072 - 3075