A review of new approaches in Her-2 targeting and 1H MRI application Dorota BartusikDavid AebisherBoguslaw Tomanek Review Article 22 August 2014 Pages: 1365 - 1368
Combination therapy with p53–MDM2 binding inhibitors for malignancies Zegao JinJianfeng ShenChunqi Hu Review Article 02 September 2014 Pages: 1369 - 1379
Synthesis and anti-inflammatory evaluation of new pyrazoles bearing biodynamic thiazole and thiazolidinone scaffolds Lalit D. KhillareManisha R. BhosleRamrao A. Mane Original Research 17 August 2014 Pages: 1380 - 1386
Synthesis, characterization, and POM analysis of novel bioactive imidazolium-based ionic liquids Mouslim MessaliMohamed R. AouadBelkheir Hammouti Original Research 19 August 2014 Pages: 1387 - 1395
Indolyl linked meta-substituted benzylidene-based novel PPAR ligands: synthetic and docking studies Raman K. VermaRajiv MallAmanjot Singh Original Research 19 August 2014 Pages: 1396 - 1407
Synthesis and selected immunological properties of 10-substituted 1,8-diazaphenothiazines Beata Morak-MłodawskaKrystian PlutaMaja Kocięba Original Research Open access 19 August 2014 Pages: 1408 - 1418
Evaluation of newly synthesized quinazolinone derivatives of hydrazones as potent anti-inflammatory and antibacterial agents Bhavna KandpalJyotsna MeshramAmbareen Shaikh Original Research 19 August 2014 Pages: 1419 - 1426
Triterpenic and monoterpenic esters from stems of Ichnocarpus frutescens and their drug likeness potential Babita AggarwalRajeev K. SinglaKah Hwi Kim Original Research 19 August 2014 Pages: 1427 - 1437
Protective effect of Pelargonium graveolens against carbon tetrachloride-induced hepatotoxicity in mice and characterization of its bioactive constituents by HPLC–PDA–ESI–MS/MS analysis Eman Al-SayedOlli MartiskainenNaglaa M. El-Lakkany Original Research 20 August 2014 Pages: 1438 - 1448
Computational identification of JAK2 inhibitors: a combined pharmacophore mapping and molecular docking approach Rohit Y. SatheSeema A. KulkarniThirumurthy Madhavan Original Research 21 August 2014 Pages: 1449 - 1467
LC-MS guided isolation of antibacterial and cytotoxic constituents from Clausena anisata Simplice Joel Ndendoung TatsimoJean-De-Dieu TamokouMichael Spiteller Original Research 23 August 2014 Pages: 1468 - 1479
Synthesis and evaluation of mefway analogs as ligands for serotonin 5HT1A receptors Joanne P. ThioChristopher LiangJogeshwar Mukherjee Original Research 23 August 2014 Pages: 1480 - 1486
Microwave-assisted synthesis of substituted 4-chloro-8-methyl-2-phenyl-1,5-dioxa-2H-phenanthren-6-ones and their antimicrobial activity D. AshokB. Vijaya LakshmiA. Ganesh Original Research 24 August 2014 Pages: 1487 - 1495
Antimalarial activity of novel imidazoisoquinolinone derivatives correlates with heme binding affinity Mariela BolliniJuan J. CasalAna M. Bruno Original Research 24 August 2014 Pages: 1496 - 1503
Moisture stable heteroleptic titanium (IV) complexes derived from 8-hydroxyquinoline: synthesis, antibacterial, and antifungal studies Blassan SamuelK. R. EthirajMadhvesh Pathak Original Research 24 August 2014 Pages: 1504 - 1513
Anticancer activity of some newly synthesized pyrano[2,3-d][1,2,3]triazine derivatives using 1-(7-hydroxy-2,2-dimethylchroman-6-yl)ethanone as synthon Nabil H. OufAbd El-Galil E. AmrMohamed I. Sakran Original Research 26 August 2014 Pages: 1514 - 1526
Molecular modeling and correlation of PFI1625c-peptide models of bioactive peptides with antimalarial properties Kimjolly LhouvumKshitij Shekhar BhuyarVishal Trivedi Original Research 26 August 2014 Pages: 1527 - 1533
Hybrid pharmacophore-based drug design, synthesis, and antiproliferative activity of 1,4-dihydropyridines-linked alkylating anticancer agents Rajesh K. SinghD. N. PrasadT. R. Bhardwaj Original Research 26 August 2014 Pages: 1534 - 1545
Synthesis, X-ray characterization and biological evaluation of some new 2-(4-methy-2-oxo-2H-chromen-7yloxy) acetamide derivatives Bhagavathula S. DiwakarB. GovindhY. L. N. Murthy Original Research 28 August 2014 Pages: 1546 - 1557
Synthesis and antitumor activity of 4-cyclohexyl/aryl-5-(pyridin-4-yl)-2,4-dihydro-3H-1,2,4-triazole-3-thiones Mashooq Ahmad BhatMohamed A. Al-OmarHoong-Kun Fun Original Research 02 September 2014 Pages: 1558 - 1567
Development of 8-benzyloxy-substituted quinoline ethers and evaluation of their antimicrobial activities Po-Yee ChungRoberto GambariKim-Hung Lam Original Research 02 September 2014 Pages: 1568 - 1577
Synthesis, spectroscopic characterization, analgesic, and antimicrobial activities of Co(II), Ni(II), and Cu(II) complexes of 2-[N,N-bis-(3,5-dimethyl-pyrazolyl-1- methyl)]aminothiazole M. KalanithiM. RajarajanS. Johnson Raja Original Research 02 September 2014 Pages: 1578 - 1585
Triarylimidazoles-synthesis of 3-(4,5-diaryl-1H-imidazol-2-yl)-2-phenyl-1H-indole derivatives as potent α-glucosidase inhibitors Sadia NaureenShazia NoreenMisbahul Ain Khan Original Research 02 September 2014 Pages: 1586 - 1595
An efficient synthesis and antimicrobial screening of new hybrid molecules containing coumarin and indenopyridine moiety Dinkar I. BrahmbhattChirag V. PatelApoorva A. Patel Original Research 03 September 2014 Pages: 1596 - 1604
Design, synthesis and antidepressant activities of some novel fatty acid analogues Selvaraj JubiePalaniswamy DhanabalRajagopal Kalirajan Original Research 03 September 2014 Pages: 1605 - 1616
A new open source data analysis python script for QSAR study and its validation Vadiraj KurdekarHemant R. Jadhav Original Research 03 September 2014 Pages: 1617 - 1625
Antibacterial potential of selected 4-phenyl hydroxycoumarins: integrated in vitro and molecular docking studies Jovana B. VeselinovićAleksandar M. VeselinovićTatjana M. Mihajilov-Krstev Original Research 03 September 2014 Pages: 1626 - 1634
Design, synthesis, and Gaussia luciferase Assay of triorganotin(IV)-based HCV inhibitors Farooq Ali ShahKaneez FatimaMohammad Ishtiaq Qadri Original Research 04 September 2014 Pages: 1635 - 1643
Antiproliferative and apoptosis inducing effect of essential oil extracted from Cyrtomium fortumei (J.) Smith leaves Shengjie YangMingchuan LiuSong Yang Original Research 04 September 2014 Pages: 1644 - 1652
Prospective study directed to the synthesis of unsymmetrical linked bis-5-arylidene rhodanine derivatives via “one-pot two steps” reactions under microwave irradiation with their antitumor activity Wacothon Karime CoulibalyLudovic PaquinJean Pierre Bazureau Original Research 05 September 2014 Pages: 1653 - 1661
Amino- and fluoro-substituted quinoline-4-carboxylic acid derivatives: MWI synthesis, cytotoxic activity, apoptotic DNA fragmentation and molecular docking studies Hardik G. BhattYadvendra K. AgrawalManish J. Patel Original Research 06 September 2014 Pages: 1662 - 1671
Biological evaluation of synthetic chalcone and flavone derivatives as anti-inflammatory agents Nelly MateevaMadhavi GangapuramKinfe K. Redda Original Research 07 September 2014 Pages: 1672 - 1680
Synthesis and biological evaluation of novel indolo[2,3-c]isoquinoline derivatives Anand R. SaundaneR. Kalpana Original Research 07 September 2014 Pages: 1681 - 1695
Two- and three-dimensional quantitative structure–permeability relationship of flavonoids in Caco-2 cells using stepwise multiple linear regression (SMLR), partial least squares regression (PLSR), and pharmacophore (GALAHAD)-based comparative molecular similarity index analysis (COMSIA) Gerard Bryan GonzalesJohn Van CampGuy Smagghe Original Research 10 September 2014 Pages: 1696 - 1706
QSAR and docking studies of some 1,2,3,4-tetrahydropyrimidines: evaluation of gp41 as possible target for anti-HIV-1 activity Saghi SepehriSajjad GharaganiAfshin Fassihi Original Research 12 September 2014 Pages: 1707 - 1724
Synthesis of quinoline/naphthalene-containing azaphenothiazines and their potent in vitro antioxidant properties Małgorzata JeleńEugenia I. BavaveaKrystian Pluta Original Research Open access 12 September 2014 Pages: 1725 - 1732
Synthesis and anti-proliferative activity evaluation of sorafenib derivatives with a 3-arylacryloyl hydrazide unit Lijing ZhangYan LiZhiqiang Feng Original Research 14 September 2014 Pages: 1733 - 1743
The SAR studies on FAP inhibitors as tumor-targeted agents Jun XuSichao HuangWeizai Shen Original Research 18 September 2014 Pages: 1744 - 1752
Modification of 3,5-bis(arylidene)-4-piperidone pharmacophore by phosphonate group using 1,2,3-triazole cycle as a linker for the synthesis of new cytostatics Mikhail V. MakarovEkaterina Yu. RybalkinaGerd-Volker Röschenthaler Original Research 20 September 2014 Pages: 1753 - 1762
Design, synthesis, and evaluation of dihydropyrimidinone (DHPM) based muscarinic receptor antagonist Badri N. AcharyaG. B. Dharma RaoMahabir P. Kaushik Original Research 21 September 2014 Pages: 1763 - 1775