Synthesis, characterization, and antimicrobial activity of copper(II) complexes with N,N′-propanediyl-bis-benzenesulfonamide and N,N′-ethanediyl-bis-2-methylbenzenesulfonamide Saliha AlyarNeslihan ÖzbekNurcan Karacan Original Research 14 September 2012 Pages: 2051 - 2060
Synthesis and biological evaluation of novel 4,5-dihydropyrazole derivatives as potent anticancer and antimicrobial agents Y. Rajendra PrasadG. V. Suresh KumarS. M. Chandrashekar Original Research 02 September 2012 Pages: 2061 - 2078
In vitro biological activities of new heterocyclic chalcone derivatives Chenna Govindaraju Darshan RajBalladaka Kunchanna SarojiniRamappa Ragavendra Original Research 18 September 2012 Pages: 2079 - 2087
Isolation of long-chain esters from the rhizome of Polygonatum verticillatum by potent tyrosinase inhibition Haroon KhanMuhammad SaeedRukhsana Ghaffar Original Research 02 September 2012 Pages: 2088 - 2092
Synthesis of damnacanthal, a naturally occurring 9,10-anthraquinone and its analogues, and its biological evaluation against five cancer cell lines Koushik SahaKok Wai LamNordin H. Lajis Original Research 13 September 2012 Pages: 2093 - 2104
Synthesis and antitumor studies of novel benzopyrano-1,2,3-selenadiazole and spiro[benzopyrano]-1,3,4-thiadiazoline derivatives S. I. El-DesokyF. A. BadriaA. H. Abdel-Rahman Original Research 31 August 2012 Pages: 2105 - 2114
Bioactive xanthones with effect on P-glycoprotein and prediction of intestinal absorption EmÃlia SousaAndreia PalmeiraMadalena Pinto Original Research 31 August 2012 Pages: 2115 - 2123
Comprehensive structure–activity relationship analysis of substituted 5-(biphenyl-4-ylmethyl) pyrazoles derivatives as AT1 selective angiotensin II receptor antagonists: 2D and kNNMFA QSAR approach Mukesh C. SharmaD. V. Kohli Original Research 23 September 2012 Pages: 2124 - 2138
Molecular docking studies on analogues of quercetin with d-alanine:d-alanine ligase of Helicobacter pylori Salam Pradeep SinghRocktotpal KonwarhNiranjan Karak Original Research 07 September 2012 Pages: 2139 - 2150
Structure–activity relationship study of thiosemicarbazones on an African trypanosome: Trypanosoma brucei brucei Houssou Raymond FatondjiSalomé KpoviessiGeorges Coffi Accrombessi Original Research 05 September 2012 Pages: 2151 - 2162
Synthesis, in vitro cytotoxicity, and antibacterial studies of new asymmetric bis-1,2,4-triazoles Rohit SinghGurubasavaraj V. PujarV. M. Chandrashekar Original Research 04 September 2012 Pages: 2163 - 2173
Pharmacophore model generation and 3D-QSAR analysis of N-acyl and N-aroylpyrazolines for enzymatic and cellular B-Raf kinase inhibition Omprakash TanwarAkranth MarellaMymoona Akhtar Original Research 05 September 2012 Pages: 2174 - 2187
Synthesis, characterization, and pharmacological evaluation of benzothiopyran derivatives as a novel class of calcium channel blockers Rajkumari NalwayaArvind SahaiGaurav Sarsodia Original Research 19 September 2012 Pages: 2188 - 2195
Synthesis and insect antifeedant activity of stilbene derivatives against Brontispa longissima Larvae Ying-Qian LiuXiao-Jing LiLiu Yang Original Research 06 September 2012 Pages: 2196 - 2206
Antitumor and antileishmanial evaluation of novel heterocycles derived from quinazoline scaffold: a molecular modeling approach Daisy H. FleitaRafat M. MoharebOla K. Sakka Original Research 09 September 2012 Pages: 2207 - 2221
Simultaneous determination of flavonoids in Oroxylum indicum by RP-HPLC Akhilesh K. YadavN. ManikaMadan M. Gupta Original Research 06 September 2012 Pages: 2222 - 2227
Synthesis and hypoglycemic activity evaluation of rhein amide derivatives Xiaokang ZhuXiaoli YeXuegang Li Original Research 05 September 2012 Pages: 2228 - 2234
3D QSAR studies on 5-(2-methylbenzimidazol-1-yl)-N-alkylthiophene-2-carboxamide derivatives as P. falciparum dihydroorotate dehydrogenase (PfDHODH) inhibitors Vivek K. VyasHarshang ParikhManjunath Ghate Original Research 06 September 2012 Pages: 2235 - 2243
Evaluation of the anti-inflammatory activity of some pyrrolo[2,3-d]pyrimidine derivatives Mosaad S. MohamedRehab KamelRania H. Abd El-hameed Original Research 06 September 2012 Pages: 2244 - 2252
Acid promoted intramolecular formation of 3,5-anhydro-1,4-furano-7-ulose derivatives via the Wittig-cyclization procedure and their antimicrobial properties Fatma Çetin TelliKadir AyYeşim Salman Original Research 18 September 2012 Pages: 2253 - 2259
Photo-activated metallotherapeutics: copper(I) or silver(I) mixed ligand complexes with 2-mercaptopyrimidine and triphenylphosphine Α. VelalopoulouG. K. BatsalaS. K. Hadjikakou Original Research 05 September 2012 Pages: 2260 - 2265
Synthesis, characterization, and antimicrobial activity of some new 2-diazo-benzimidazole derivatives and their Ni(II), Cu(II), and Ag(I) complexes Yellajyosula Lakshmi Narasimha MurthyGuduru DurgaAnjali Jha Original Research 18 October 2012 Pages: 2266 - 2272
Inhibition of pancreatic lipase by berberine and dihydroberberine: an investigation by docking simulation and experimental validation Mohammad MohammadIhab M. Al-masriYasser Bustanji Original Research 06 September 2012 Pages: 2273 - 2278
Coumarinyl pyrazole derivatives of INH: promising antimycobacterial agents Prashant AragadeMahesh PalkarDarbhamulla Satyanarayana Original Research 06 September 2012 Pages: 2279 - 2283
Integrating GUSAR and QSAR analyses for antimalarial activity of synthetic prodiginines against multi drug resistant strain Devidas T. MahajanVijay H. MasandVesna Rastija Original Research 22 September 2012 Pages: 2284 - 2292
5-Nitro-heteroarylidene analogs of 2-thiazolylimino-4-thiazolidinones as a novel series of antibacterial agents Nouraddin HosseinzadehMohammad HasaniAbbas Shafiee Original Research 13 September 2012 Pages: 2293 - 2302
Pro-apoptotic properties of parthenin analogs: a quantitative structure–activity relationship study Rukmankesh MehraAmit NargotraSurrinder Koul Original Research 04 October 2012 Pages: 2303 - 2311
Three-dimensional quantitative structure–activity relationship (3D-QSAR) analysis and molecular docking-based combined in silico rational approach to design potent and novel TRPV1 antagonists Kamlendra Singh BhadoriyaMukesh C. SharmaJyotsna R. Rananaware Original Research 04 October 2012 Pages: 2312 - 2327
New molecular scaffolds for the design of Alzheimer’s acetylcholinesterase inhibitors identified using ligand- and receptor-based virtual screening Nitin ChitranshiShipra GuptaPrahlad Kishore Seth Original Research 30 September 2012 Pages: 2328 - 2345
A new isoflavone from Blepharis ciliaris of an Egyptian origin Mohamed A. El-ShanawanyHanaa M. SayedSamir A. Ross Original Research 18 September 2012 Pages: 2346 - 2350
Synthesis, physico-chemical properties, and antimicrobial evaluation of a new series of iron(III) hexadentate chelators Yuan-Yuan XieMu-Song LiuTao Zhou Original Research 22 September 2012 Pages: 2351 - 2359
Synthesis, molecular modeling study, preliminary antibacterial, and antitumor evaluation of N-substituted naphthalimides and their structural analogues Adel S. El-AzabAmer M. AlanaziAlaa A.-M. Abdel-Aziz Original Research 04 October 2012 Pages: 2360 - 2375
Synthesis and anticancer evaluation of novel 3,5-diaryl-thiazolo[4,5-d]pyrimidin-2-one derivatives Lilianna BecanEdwin Wagner Original Research Open access 04 October 2012 Pages: 2376 - 2384
Structure–activity relationship study of growth inhibitory 2-styrylchromones against carcinoma cells Chen LinPei-Jung LuArthur Y. Shaw Original Research 23 September 2012 Pages: 2385 - 2394
Copper(II) complexes with derivatives of pyrazole as potential antioxidant enzyme mimics Bogumiła KupcewiczKrzysztof SobiesiakElżbieta Budzisz Original Research Open access 26 September 2012 Pages: 2395 - 2402
Evidence of stereoselective and segmental-dependant transport of chiral antidiabetic drug nateglinide along the rat small intestine: possible role of efflux transporters Srinivas MaddiShravan Kumar YamsaniMadhusudan Rao Yamsani Original Research 28 September 2012 Pages: 2403 - 2410
Design and synthesis of niflumic acid-based N-acylhydrazone derivatives as novel anti-inflammatory and analgesic agents Amin KheradmandLatifeh NavidpourAbbas Shafiee Original Research 27 September 2012 Pages: 2411 - 2420
Synthesis and in vitro anticancer activity of novel thiazacridine derivatives Marina Galdino da Rocha PittaÉrika Silva SouzaIvan da Rocha Pitta Original Research 28 September 2012 Pages: 2421 - 2429
In vivo antidiabetic activity and in silico studies on adenosine monophosphate-activated protein kinase (AMPK) of (2E,5E)-2,5-bis(4-hydroxy-3-methoxybenzylidene) cyclopentanone Chenna Govindaraju Darshan RajBalladka Kunhanna SarojiniRamappa Raghavendra Original Research 06 October 2012 Pages: 2430 - 2436
POM analyses of antitrypanosomal activity of 2-iminobenzimidazoles: favorable and unfavorable parameters for drugs optimization Taibi Ben HaddaRahima MouhoubIsmail Warad Original Research 26 September 2012 Pages: 2437 - 2445
Synthesis, cytotoxic, and DNA binding studies of novel fluorinated condensed pyrano pyrazoles S. BhavanarushiV. KanakaiahJ. Vatsala Rani Original Research 28 September 2012 Pages: 2446 - 2454
Synthesis and anticancer activity of para-xylyl linked bis-benzimidazolium salts and respective Ag(I) N-heterocyclic carbene complexes Muhammad Adnan IqbalRosenani A. HaqueSawsan S. Al-Rawi Original Research 09 October 2012 Pages: 2455 - 2466
Synthesis, biological evaluation, and molecular modeling studies of new 1,3,4-oxadiazole- and 1,3,4-thiadiazole-substituted 4-oxo-4H-pyrido[1,2-a]pyrimidines as anti-HIV-1 agents Z. HajimahdiA. ZarghiM. R. Aghasadeghi Original Research 28 September 2012 Pages: 2467 - 2475
Synthesis and QSAR modeling 1-[3-methyl-2-(aryldiazenyl)-2H-aziren-2-yl]ethanones as potential antibacterial agents Vinita SahuPratibha SharmaAshok Kumar Original Research 27 September 2012 Pages: 2476 - 2485
Synthesis of novel 2-phenyl-3-[2-(substituted amino) ethylamino] quinazolin-4(3H)-ones as a new class of H1-antihistaminic agents V. AlagarsamyP. Shyam SundarV. Raja Solomon Original Research 26 September 2012 Pages: 2486 - 2492
Computer simulation of the in vitro and in vivo anti-inflammatory activities of dihydropyrimidines acid derivatives through the inhibition of cyclooxygenase-2 Raksha DhankarAnjali M. RahatgaonkarAshutosh Tiwari Original Research 27 September 2012 Pages: 2493 - 2504
Synthesis and bioevaluation of novel arylnaphthalene lignans as anticancer agents Yu ZhaoJie HuiLi Zhu Original Research 25 September 2012 Pages: 2505 - 2510
Enhancement of P-gylcoprotein modulators of arylmethylamine-phenyl derivatives: an integrative modeling approach Thirumurthy MadhavanChangdev G. GadheSeung Joo Cho Original Research 26 September 2012 Pages: 2511 - 2523
Free radical scavenging and hepatoprotective effects of salidroside analogs on CCl4-induced cytotoxicity in LO2 cells Yibing GuoCheng ZhengYumin Yang Original Research 26 September 2012 Pages: 2524 - 2530
Microbiologically active Mannich bases derived from 1,2,4-triazoles. The effect of C-5 substituent on antibacterial activity Tomasz PlechMonika WujecAnna Malm Original Research Open access 29 September 2012 Pages: 2531 - 2537