Novel quinazolinone derivatives: synthesis and antimicrobial activity Osman M. O. HabibHussein M. HassanAhmed El-Mekabaty Symposium Paper 04 May 2012 Pages: 507 - 519
Action of benzimidazolo-piperazinyl derivatives on dopamine receptors Zenish J. JainRani S. KankateRohini D. Kakad Review Article 24 April 2012 Pages: 520 - 530
Colchicine and its various physicochemical and biological aspects Sameer SapraYashika BhallaKanaya L. Dhar Review Article 13 May 2012 Pages: 531 - 547
In vitro antiproliferative effect of β-phenylethylamine derivatives and doxorubicin combinations on MCF/ADR cell lines Wanda P. AlmeidaPaula C. HuberJoão E. de Carvalho Original Research 11 April 2012 Pages: 548 - 557
Discovery of novel DPP IV inhibitors: application of pharmacophore-based virtual screening Jyoti SharmaDivya YadavSarvesh Paliwal Original Research 13 April 2012 Pages: 558 - 572
Immunomodulatory active steroidal saponins from Asparagus racemosus Upendra SharmaNeeraj KumarSupriya Bhalerao Original Research 13 April 2012 Pages: 573 - 579
Spectroscopic characterization of novel d-amino acid-Schiff bases and their Cr(III) and Ni(II) complexes as antimicrobial agents Nurşen SarıNihat PişkinNurdan Kurnaz Original Research 15 April 2012 Pages: 580 - 587
A comprehensive structure–activity analysis 2,3,5-trisubstituted 4,5-dihydro-4-oxo-3H-imidazo [4,5-c] pyridine derivatives as angiotensin II receptor antagonists: using 2D- and 3D-QSAR approach Mukesh C. SharmaD. V. Kohli Original Research 20 April 2012 Pages: 588 - 605
Binding site analysis, 3D-QSAR studies, and molecular design of flavonoids derivatives as potent neuraminidase inhibitors Jiaying SunHu Mei Original Research 20 April 2012 Pages: 606 - 614
Atom-based 3D QSAR studies on novel N-β-d-xylosylindole derivatives as SGLT2 inhibitors Venkatesan SuryanarayananArumugam SudhaPappu Srinivasan Original Research 21 April 2012 Pages: 615 - 624
From peptides to peptidomimetics: rational design of potential PKC-β II inhibitors P. Sri DivyaKapil JainM. Elizabeth Sobhia Original Research 20 April 2012 Pages: 625 - 634
Synthesis and in vitro antimicrobial and anti-tubercular evaluation of some quinoline-based azitidinone and thiazolidinone analogues Bhupendra M. MistrySmita Jauhari Original Research 22 April 2012 Pages: 635 - 646
Quinoline-based azetidinone and thiazolidinone analogues as antimicrobial and antituberculosis agents Bhupendra M. MistrySmita Jauhari Original Research 22 April 2012 Pages: 647 - 658
Novel 2-thiopyrimidine derivatives as CDK2 inhibitors: molecular modeling, synthesis, and anti-tumor activity evaluation Omar Abd El-Fattah M. FathallaMohamed A. H. IsmailAisha A. K. Ramadan Original Research 24 April 2012 Pages: 659 - 673
Synthesis and biological evaluation of gallic acid analogs Maurizio BarontiniIlaria Proietti SilvestriGiuliana Righi Original Research 24 April 2012 Pages: 674 - 680
Synthesis, structure, and estrogenic activity of 2- and 3-substituted 2,3-dihydro-4H-1-benzopyran-4-ones Yves JacquotCillian ByrneGuy Leclercq Original Research 25 April 2012 Pages: 681 - 691
Synthesis of imidazole-derived steroidal hybrids as potent aromatase inhibitors Ranju BansalSheetal GuleriaChristina Zimmer Original Research 25 April 2012 Pages: 692 - 698
Synthesis and antimicrobial screening of 4-thiazolidinone and 2-azetidinone derivatives of piperazine Sunil G. ShingadeSanjaykumar B. Bari Original Research 27 April 2012 Pages: 699 - 706
Design, synthesis, and biological evaluation of new 4-thiazolidinone derivatives substituted with benzimidazole ring as potential chemotherapeutic agents Georgina N. MasoudAmal M. YoussefAly A. B. Hazzaa Original Research 01 May 2012 Pages: 707 - 725
In vitro antimicrobial and antimycobacterial activity of some chalcones and their derivatives Divyesh PatelPremlata KumariNavin B. Patel Original Research 01 May 2012 Pages: 726 - 744
Analysis of 6-methoxy podophyllotoxin and podophyllotoxin in hairy root cultures of Linum album Kotschy ex Boiss Najmeh Ahmadian ChashmiMozafar SharifiJavier Palazon Original Research 04 May 2012 Pages: 745 - 752
Synthesis and evaluation of antioxidant activity of 2-styrylchromones Shrinivas P. PawarDasharath D. KondhareP. K. Zubaidha Original Research 04 May 2012 Pages: 753 - 757
Synthesis, characterization, anticancer, and antioxidant activity of some new thiazolidin-4-ones in MCF-7 cells Arun M. IsloorDhanya SunilNaseer Maliyakkl Original Research 04 May 2012 Pages: 758 - 767
Synthesis and antimicrobial activity of coumarin pyrazole pyrimidine 2,4,6(1H,3H,5H)triones and thioxopyrimidine4,6(1H,5H)diones S. Vijaya LaxmiB. Suresh KuarmB. Rajitha Original Research 05 May 2012 Pages: 768 - 774
Pyrazolo[3,4-d]pyrimidine analogues: synthesis, characterization and their in vitro antiamoebic activity Shadab Miyan SiddiquiAttar SalahuddinAmir Azam Original Research 06 May 2012 Pages: 775 - 781
Synthesis and evaluation of analgesic, anti-inflammatory, and anticancer activities of new pyrazole-3(5)-carboxylic acid derivatives Burcu ÇalışkanAkın YılmazErden Banoglu Original Research 06 May 2012 Pages: 782 - 793
Synthesis and antioxidant studies of novel N-substituted benzyl/phenyl-2-(3,4-dimethyl-5,5-dioxidopyrazolo[4,3-c][1,2]benzothiazin-2(4H)-yl)acetamides Matloob AhmadHamid Latif SiddiquiSana Aslam Original Research 11 May 2012 Pages: 794 - 805
Synthesis, antimicrobial and antioxidant activities of some new indole derivatives containing pyridopyrimidine and pyrazolopyridine moieties Anand R. SaundaneKatkar VijaykumarPrabhaker Walmik Original Research 11 May 2012 Pages: 806 - 817
Synthesis and antibacterial, antimycobacterial and docking studies of novel N-piperazinyl fluoroquinolones Kapil M. AgrawalGokul S. Talele Original Research 11 May 2012 Pages: 818 - 831
Essential oil composition, insecticidal and antibacterial activities of Salvia tomentosa Miller Zeynep UlukanliSalih KarabörklüMehmet Balcilar Original Research 11 May 2012 Pages: 832 - 840
Synthesis and biological evaluation of novel benzoquinones as potential antimicrobial agents Ibrahim ChaabanEl Sayeda M. El KhawassAbeer E. Abdel Wahab Original Research 13 May 2012 Pages: 841 - 851
Synthesis of new N-arylamino(2-furyl)methylphosphonic acid diesters, and in vitro evaluation of their cytotoxicity against esophageal cancer cells Anna Agnieszka KlimczakAgnieszka KuropatwaJanusz Szemraj Original Research 15 May 2012 Pages: 852 - 860
Anti-inflammatory and selective COX-2 inhibitory activities of metal complexes of Schiff bases derived from aldoses Mohammad S. IqbalSyed J. KhurshidBakhtiar Muhammad Original Research 15 May 2012 Pages: 861 - 868
Synthesis and evaluation of antibacterial and antitubercular activities of some novel imidazo[2,1-b][1,3,4]thiadiazole derivatives S. D. JoshiK. ManishAravind Badiger Original Research 19 May 2012 Pages: 869 - 878
Identification of an antiepileptic lead compound with a more selective activity and its analogues for GABA-AT using in silico approach Hina Naz KhanSaima KulsoomHamid Rashid Original Research 22 May 2012 Pages: 879 - 889
QSAR and pharmacophore modeling of N-acetyl-2-aminobenzothiazole class of phosphoinositide-3-kinase-α inhibitors Sandip B. BharateBaljinder SinghRam A. Vishwakarma Original Research 22 May 2012 Pages: 890 - 899
Synthesis of novel benzimidazole derivatives: as potent analgesic agent Shushank DixitPramod Kumar SharmaNiranjan Kaushik Original Research 22 May 2012 Pages: 900 - 904
Microwave-assisted CAN-catalyzed solvent-free synthesis of N-allyl quinolone-based pyrano[4,3-b]chromene and benzopyrano[3,2-c]chromene derivatives and their antimicrobial activity Hardik H. JardoshManish P. Patel Original Research 22 May 2012 Pages: 905 - 915
Molecular properties prediction, synthesis, and diuretic activity of phenoxy acetic acid bearing pyrazolines Mohammed Afroz BakhtM. Shahar YarAhmed M-Alafeefy Original Research 22 May 2012 Pages: 916 - 926
Synthesis and in vitro antibacterial activity of schiff bases of N-substituted isatins as effective scaffolds Garima KumariRamendra K. Singh Original Research 26 May 2012 Pages: 927 - 933
The impact of glycerol and some carbohydrates on antibiotic production by Streptomyces hygroscopicus CH-7 Slavica B. IlićSandra S. KonstantinovićVlada B. Veljković Original Research 26 May 2012 Pages: 934 - 937
Synthesis and pharmacological evaluation of novel 4-isopropylthiazole-4-phenyl-1,2,4-triazole derivatives as potential antimicrobial and antitubercular agents G. V. Suresh KumarY. Rajendra PrasadS. M. Chandrashekar Original Research 26 May 2012 Pages: 938 - 948
In silico ligand-based pharmacophore model generation for the identification of novel Pneumocystis carinii DHFR inhibitors Yusra Sajid KianiSaima KalsoomNaveeda Riaz Original Research 30 May 2012 Pages: 949 - 963
Antibacterial, antifungal and antioxidant activity of some new water-soluble β-diketones Javed SheikhTaibi Ben Hadda Original Research 27 May 2012 Pages: 964 - 975
Application of pocket modeling and k-nearest neighbor molecular field analysis (kNN-MFA) for designing of some anticoagulants: potential factor IXa inhibitors P. B. ChoudhariM. S. BhatiaN. M. Bhatia Original Research 30 May 2012 Pages: 976 - 985
Synthesis, structure, and biological assay of cinnamic amides as potential EGFR kinase inhibitors Mao ZhangXiang LuYong-Hao Ye Original Research 29 May 2012 Pages: 986 - 994
Synthesis of kojic acid-derived copper-chelating apoptosis inducing agents Yu-Hua ChenPei-Jung LuArthur Y. Shaw Original Research 29 May 2012 Pages: 995 - 1003
In silico designing and characterization of Amiloride derivatives as ion channel modulator Ajeet Original Research 27 May 2012 Pages: 1004 - 1010
Design, synthesis, anti-inflammatory, analgesic screening, and molecular docking of some novel 2-pyridyl (3H)-quinazolin-4-one derivatives Ahmad F. EweasAhmed O. H. El-NezhawyMohamed M. Awad Original Research 27 May 2012 Pages: 1011 - 1020
Synthesis, characterization, and biological evaluation of certain 1,3-thiazolone derivatives bearing pyrazoline moiety as potential anti-breast cancer agents Nadia A. KhalilEman M. AhmedHala B. El-Nassan Original Research 27 May 2012 Pages: 1021 - 1027