Design, synthesis and in vitro PDE4 inhibition activity of certain quinazolinone derivatives for treatment of asthma Afaf K. ElansaryHanan H. KadryAmr Sayed Motawi Sonousi Symposium Paper 19 November 2011 Pages: 3327 - 3335
The effect of pyridazine compounds on the cardiovascular system Mohammad AsifAnita SinghAnees A. Siddiqui Review Article 19 November 2011 Pages: 3336 - 3346
Pharmacological profile of green tea and its polyphenols: a review Sumit BansalNavneet SyanShivani Choudhary Review Article 28 December 2011 Pages: 3347 - 3360
Synthesis, characterization and in vitro hydrolysis studies of ester and amide prodrugs of dexibuprofen Zaman AshrafMuhammad ImranShahid Amin Original Research 17 November 2011 Pages: 3361 - 3368
Combination of flavopiridol and embelin effectively inhibit cell growth in hepatocellular carcinoma depending on regulatory relationship between CDK6 and XIAP Yufang CheDavid Y. ZhangBo Jiang Original Research 17 November 2011 Pages: 3369 - 3375
Synthesis of 1,3,5-trisubstituted pyrazoline nucleus containing compounds and screening for antimicrobial activity Manish AgrawalPankaj Kumar SonarShailendra K. Saraf Original Research 17 November 2011 Pages: 3376 - 3381
EBHU18, a novel derivative of fatty acid bile acid conjugates, prevents cholesterol gallstone formation in experimental mice Lei YuYan-Fang JiangJun-Qi Niu Original Research 19 November 2011 Pages: 3382 - 3389
Synthesis and antimicrobial evaluation of 4,5-diaryl-2-[4-(t-amino)-2-butynyl]-2,4-dihydro-3H-1,2,4-triazol-3-ones E. N. Al-kaissiN. F. Al-GhraryZ. Muhi-eldeen Original Research 19 November 2011 Pages: 3390 - 3395
Synthesis and biological evaluation of some pyrazole derivatives as anti-inflammatory–antibacterial agents Pawan KumarNavneet ChandakPawan K. Sharma Original Research 19 November 2011 Pages: 3396 - 3405
Microwave-assisted synthesis of 3′-indolyl substituted 4H-chromenes catalyzed by DMAP and their antimicrobial activity Harshad G. KathrotiyaManish P. Patel Original Research 19 November 2011 Pages: 3406 - 3416
Pharmacophore modeling, virtual screening, and molecular docking studies for discovery of novel Carbonic anhydrase IX inhibitors Chun-Lin LuLu ZhouWei Zhang Original Research 19 November 2011 Pages: 3417 - 3427
In vivo screening of diarylimidazoles as anticonvulsant agents Mirko RivaraValentina Zuliani Original Research 19 November 2011 Pages: 3428 - 3434
Synthesis, characterization, and antibacterial activity of the ligands including thiophene/furan ring systems and their Cu(II), Zn(II) complexes Ayla Balaban GündüzalpNeslihan ÖzbekNurcan Karacan Original Research 19 November 2011 Pages: 3435 - 3444
Synthesis and leishmanicidal activity of quinoline–triclosan and quinoline–eugenol hybrids Victor ArangoJorge J. DomÃnguezJairo Sáez Original Research 19 November 2011 Pages: 3445 - 3454
Serotonin transporter activity of imidazolidine-2,4-dione and imidazo[2,1-f]purine-2,4-dione derivatives in aspect of their acid–base properties Agnieszka ZagórskaAnna CzopekGabriel Nowak Original Research Open access 19 November 2011 Pages: 3455 - 3459
Isolation and anxiolytic activity of 3,4-bis(3,4-dimethoxyphenyl)furan-2,5-dione from the ethanolic extract of heart wood of Cedrus deodara Daniel DhayabaranJeyaseeli FloranceAyarivan Puratchikody Original Research 19 November 2011 Pages: 3460 - 3464
Discovery of potent anticonvulsant ligands as dual NMDA and AMPA receptors antagonists by molecular modelling studies Shailesh V. JainKamlendra S. BhadoriyaManjunath Ghate Original Research 19 November 2011 Pages: 3465 - 3484
Chemical composition and antibacterial activity of the essential oils from the medicinal plant Mentha cervina L. grown in Portugal Leandra RodriguesAida DuarteAna Monteiro Original Research 20 November 2011 Pages: 3485 - 3490
Acute and chronic anti-inflammatory evaluation of imidazo[1,2-a]pyridine carboxylic acid derivatives and docking analysis YazmÃn K. Márquez-FloresMa. Elena Campos-AldreteMa. Estela Meléndez-Camargo Original Research 20 November 2011 Pages: 3491 - 3498
Synthesis and biological activity of hydrazide–hydrazones and their corresponding 3-acetyl-2,5-disubstituted-2,3-dihydro-1,3,4-oxadiazoles Bedia Koçyiğit-KaymakçıoğluEmine Elçin Oruç-EmreSevim Rollas Original Research 20 November 2011 Pages: 3499 - 3508
Synthesis and antidepressant activity of di substituted-5-aryl-1,2,4-triazoles C. RadhikaA. VenkateshamManda Sarangapani Original Research 20 November 2011 Pages: 3509 - 3513
Antioxidant, cytotoxicity, and QSAR study of 1-adamantylthio derivatives of 3-picoline and phenylpyridines Apilak WorachartcheewanSupaluk PrachayasittikulVirapong Prachayasittikul Original Research 20 November 2011 Pages: 3514 - 3522
Study on single crystal structure of the antimony(III) bromide complex with 3-methyl-2-mercaptobenzothiazole and biological activity of some antimony(III) bromide complexes with thioamides I. I. OzturkA. K. MetsiosN. Hadjiliadis Original Research 20 November 2011 Pages: 3523 - 3531
Anti-inflammatory effects of two new methyl and morpholine derivatives of diphenhydramine on rats Abbas AhmadiMohsen KhaliliBabak Nahri-Niknafs Original Research 22 November 2011 Pages: 3532 - 3540
Synthesis and antimicrobial activities of some isoxazolyl thiazolyl pyrazoles Satbir MorRajni MohilMunish Ahuja Original Research 19 November 2011 Pages: 3541 - 3548
Efficient isolation of catechins from green tea and characterization of interaction property of catechins with proteins by HPLC–UV/DAD combined with ultrafiltration Jian-Min ShenXiao-Yan LiuHai-Xia Zhang Original Research 25 November 2011 Pages: 3549 - 3556
Design, synthesis, and biological activity of certain quinazolinedione derivatives as potent phosphodiestrase4 inhibitors Afaf K. ElansaryHanan H. KadryAmr Sayed Motawi Sonousi Original Research 25 November 2011 Pages: 3557 - 3567
Synthesis of new potential anticancer agents based on 4-thiazolidinone and oleanane scaffolds Danylo KaminskyyBarbara Bednarczyk-CwynarRoman Lesyk Original Research 25 November 2011 Pages: 3568 - 3580
Design, synthesis, and evaluation of anti-inflammatory and ulcerogenicity of novel pyridazinone derivatives K. A. M. AbouzidN. A. KhalilA. M. Al-Abd Original Research 25 November 2011 Pages: 3581 - 3590
Physical and chemical characterization of mefenamic acid in different pharmaceutical dosage forms and their stability studies using novel RP-HPLC method Shabana Naz ShahAgha Zeeshan MirzaMalik Asia Naz Original Research 25 November 2011 Pages: 3591 - 3597
Synthesis and biological evaluation of novel pyrimidine-2(1H)-ones/thiones as potent anti-inflammatory and anticancer agents Vachala Seekarajapuram DinakaranDivya JacobJessy Elizabeth Mathew Original Research 25 November 2011 Pages: 3598 - 3606
Diorganotin (IV) derivative of 2-thiophene acetic acid: characterizations and biological activities of {[n-Bu2SnO2C–CH2–C4H3S]2O}2 Abdelkader EttouhamiAbderrahman YahyiM. Iqbal Choudhary Original Research 25 November 2011 Pages: 3607 - 3614
1-(7-Chloroquinolin-4-yl)-2-[(1H-pyrrol-2-yl)methylene]hydrazine: a potent compound against cancer Raquel Carvalho MontenegroLetÃcia Veras LotufoMarcus VinÃcius Nora de Souza Original Research 27 November 2011 Pages: 3615 - 3619
Synthesis, anti-inflammatory and anticancer activity evaluation of some mono- and bis-Schiff’s bases Sham M. SondhiSurbhi AryaPartha Roy Original Research 27 November 2011 Pages: 3620 - 3628
Microwave assisted synthesis of novel pyrimidine derivatives and investigation of their analgesic and ulcerogenic activity Anshu ChaudharyPramod Kumar SharmaRupesh Dudhe Original Research 27 November 2011 Pages: 3629 - 3645
Pharmacological screening for anti-inflammatory, analgesic activity of pyrazolyl derivatives along with molecular docking studies Darpan KaushikRajnish KumarGita Chawla Original Research 29 November 2011 Pages: 3646 - 3655
Pharmacopore hypothesis generation of BACE-1 inhibitors and pharmacophore-driven identification of potent multi-target neuroprotective agents Wen-Ting ZhangFeng-Chao JiangGuang Du Original Research 30 November 2011 Pages: 3656 - 3668
Design, synthesis, and biological evaluation of sulfonic acid ester and benzenesulfonamide derivatives as potential CETP inhibitors Reema Abu KhalafGhassan Abu SheikhaMutasem Taha Original Research 30 November 2011 Pages: 3669 - 3680
Development of QSAR model for prediction of fold selectivity of phenyl benzoxazole as estrogen receptor inhibitors Laxman M. PrajapatiVijay K. ParmarJimish R. Patel Original Research 30 November 2011 Pages: 3681 - 3686
Synthesis and antimicrobial screening of novel 2,6-ditertiarybutylpiperidin-4-ones C. GovindarajuR. ValliappanV. Sundari Original Research 01 December 2011 Pages: 3687 - 3691
Synthesis and study of the antidepressant activity of novel 4,5-dihydro-7-alkoxy(phenoxy)-tetrazolo[1,5-a]quinoline derivatives Xian-Yu SunXian-Jing HeYun-Peng Zou Original Research 01 December 2011 Pages: 3692 - 3698
Synthesis and anticonvulsant activity of some new series of pyrrole derivatives A. IdhayadhullaR. Surendra KumarS. Indumathy Original Research 02 December 2011 Pages: 3699 - 3708
Synthetic utility of sydnones: synthesis of pyrazolines derivatized with 1,2,4-triazoles as antihyperglymic, antioxidant agents and their DNA cleavage study Tasneem TajRavindra R. KambleBharati V. Badami Original Research 02 December 2011 Pages: 3709 - 3719
Synthesis of combretastatin analogs: evaluation of in vitro anticancer activity and molecular docking studies Sunil KumarSameer SapraKanahya Lal Dhar Original Research 03 December 2011 Pages: 3720 - 3729
Synthesis, biological activity and docking study of some new isatin Schiff base derivatives Javad AzizianMohammad K. MohammadiRamin Miri Original Research 03 December 2011 Pages: 3730 - 3740
Anti-HIV-1 and cytotoxicity studies of piperidyl-thienyl chalcones and their 2-pyrazoline derivatives Syed Umar Farooq RizviHamid Latif SiddiquiRaymond F. Schinazi Original Research 04 December 2011 Pages: 3741 - 3749
Synthesis and antimicrobial activity of some new 4-triazolylmethoxy-2H-chromen-2-one derivatives Siva S. PandaRitu MalikSubhash C. Jain Original Research 06 December 2011 Pages: 3750 - 3756
Heteroaromatic analogues of 1,5-diarylpyrazole class as anti-inflammatory agents Pawan K. SharmaNisha ChandnaDhirender Kaushik Original Research 06 December 2011 Pages: 3757 - 3766
Molecular modeling and protection against pentylenetetrazole-induced seizure of new 1,4-dihydropyridines containing 5(4)-imidazolyl substituent Asghar DavoodHamed ShafaroodiAbbas Shafiee Original Research 06 December 2011 Pages: 3767 - 3776
Computation of pharmacophore models for the prediction of mitogen-activated protein kinase activated protein kinase-2 inhibitory activity of pyrrolopyridines Upasna KaushikVikas SharmaVipin Kumar Original Research 06 December 2011 Pages: 3777 - 3784