Polyalkylcyanoacrylate Nanoparticles as Polymeric Carriers for Antisense Oligonucleotides Christine ChavanyTrung Le DoanClaude Hélèna OriginalPaper Pages: 441 - 449
Correlation of in Vitro Release Rate and in Vivo Absorption Characteristics of Four Chlorpheniramine Maleate Extended-Release Formulations Parviz MojaverianElaine RadwanskiJack M. Rosen OriginalPaper Pages: 450 - 456
Pharmacokinetic and Pharmacodynamic Comparison of Immediate-Release and Sustained-Release Adinazolam Mesylate Tablets After Single- and Multiple-Dose Administration Joseph C. FleishakerC. Eugene Wright OriginalPaper Pages: 457 - 463
The Pharmacokinetics of Trilostane and Ketotrilostane in an Interconverting System in the Rat J. Paul McGeeP. Nicholas Shaw OriginalPaper Pages: 464 - 468
Saturable Tissue Binding and Imirestat Pharmacokinetics in Rats Jenny Y. ChienChristopher R. BanfieldJohn T. Slattery OriginalPaper Pages: 469 - 473
Significance of Binding to Na,K-ATPase in the Tissue Distribution of Ouabain in Guinea Pigs Hideyoshi HarashimaMichio MamiyaManabu Hanano OriginalPaper Pages: 474 - 479
The in Situ Acetylation of an Immobilized Human Serum Albumin Chiral Stationary Phase for High-Performance Liquid Chromatography in the Examination of Drug–Protein Binding Phenomena Terence A. G. NoctorIrving W. Wainer OriginalPaper Pages: 480 - 484
An Air-Gap Enzyme Electrode: Development and Applications Ravi M. ShankerNashed E. NashedSiegfried Lindenbaum OriginalPaper Pages: 485 - 491
Stereoselective Enzymatic Hydrolysis of Various Ester Prodrugs of Ibuprofen and Flurbiprofen in Human Plasma Niels MørkHans Bundgaard OriginalPaper Pages: 492 - 496
The in Vitro Enzymic Labilities of Chemically Distinct Phosphomonoester Prodrugs Albert S. KearneyValentine J. Stella OriginalPaper Pages: 497 - 503
Amino Acid Side-Chain Contributions to Free Energy of Transfer of Tripeptides from Water to Octanol Aeri KimFrancis C. Szoka Jr OriginalPaper Pages: 504 - 514
Nebulization of Liposomes. III. The Effects of Operating Conditions and Local Environment Ralph W. NivenTeresa M. CarvajalHans Schreier OriginalPaper Pages: 515 - 520
Infrared Imaging of Pharmaceutical Materials Undergoing Compaction Simon R. BechardG. R. B. Down OriginalPaper Pages: 521 - 528
Absorptive-Mediated Endocytosis of an Adrenocorticotropic Hormone (ACTH) Analogue, Ebiratide, into the Blood–Brain Barrier: Studies with Monolayers of Primary Cultured Bovine Brain Capillary Endothelial Cells Tetsuya TerasakiSusumu TakakuwaAkira Tsuji OriginalPaper Pages: 529 - 534
Aminopeptidase Activity in the Jejunal and Heal Peyer's Patches of the Albino Rabbit Eiji HayakawaVincent H. L. Lee OriginalPaper Pages: 535 - 540
Phagocytosis of Nanoparticles by Human Immunodeficiency Virus (HlV)-Infected Macrophages: A Possibility for Antiviral Drug Targeting Volker SchäferHagen von BriesenHelga Rübsamen-Waigmann OriginalPaper Pages: 541 - 546
Bioadhesion by Means of Specific Binding of Tomato Lectin Claus-Michael LehrJoke A. BouwstraHans E. Junginger OriginalPaper Pages: 547 - 553
Influence of Supersaturation on the Pharmacodynamic Effect of Bupranolol After Dermal Administration Using Microemulsions as Vehicle Jens KemkenAlbrecht ZieglerBernd W. Müller OriginalPaper Pages: 554 - 558
Sonophoresis. I. The Use of High-Frequency Ultrasound to Enhance Transdermal Drug Delivery D. BommannanHirohisa OkuyamaRichard H. Guy OriginalPaper Pages: 559 - 564
Characteristics of Association of Oleoyl Derivatives of 5-Fluorodeoxyuridine and Methotrexate with Low-Density Lipoproteins (LDL) P. Chris de SmidtTheo J. C. van Berkel OriginalPaper Pages: 565 - 569
Physicochemical Properties of the Novel Heteropolyanion Antiviral Hexapotassium-α-vanado-11-tungstoborate (DuP 925) Michael B. MaurinRodney D. VickeryMunir A. Hussain OriginalPaper Pages: 570 - 574
1H-Nuclear Magnetic Resonance (NMR) Studies on the Inclusion Complex of Prostaglandin El (PGE1 with α-Cyclodextrin Bert SteffanWilfried FischerRobert Müller OriginalPaper Pages: 575 - 577
A Flexible Automated Dissolution Testing System for Use with Either USP Apparatus 1 or USP Apparatus 2 Jeanette D. DunkleDaniel J. GleasonGerard C. Hokanson Note Pages: 578 - 581
Determination of Dissociation Constants of Selected Cyclodextrin–Benzaldehyde Inclusion Complexes Using Pulse Polarography1 Hee-Sook ChoiChing-jer ChangAdelbert M. Knevel Note Pages: 582 - 584
Analytical Methods Validation: Bioavailability, Bioequivalence and Pharmacokinetic Studies Vinod P. ShahKamal K. MidhaSidney Spector Conference Report Pages: 588 - 592