Abstract
A synthetic route has been proposed to 3-phenyl-1H-[1,4]oxazino[4,3-a]benzimidazol-1-one, which is the first representative of a new heterocyclic system. The transformation of the title compound to 4-phenyl-2,5-dihydro-1H-[1,2,5]triazepino[5,4-a]benzimidazol-1-one via reaction with hydrazine hydrate has been studied.
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Translated from Zhurnal Organicheskoi Khimii, 2021, Vol. 57, No. 3, pp. 426–432 https://doi.org/10.31857/S0514749221030113.
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Kharaneko, A.O., Pekhtereva, T.M. & Kharaneko, O.I. Synthesis of 3-Phenyl-1H-[1,4]oxazino[4,3-a]benzimidazol-1-one and Its Transformation into 4-Phenyl-2,5-dihydro-1H-[1,2,5]triazepino[5,4-a]benzimidazol-1-one. Russ J Org Chem 57, 396–401 (2021). https://doi.org/10.1134/S1070428021030118
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DOI: https://doi.org/10.1134/S1070428021030118