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Chelate method for the synthesis of 3-amidino-substituted 4-pyridones

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Abstract

An efficient synthetic procedure to obtain 3-(N-benzoylamidino)-substituted 4-pyridones has been developed based on the reaction of difluoroboron complex of N-benzoyl-substituted diacylketene aminal with primary amines.

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References

  1. R. Gompper, R. Kunz, Chem. Ber., 1965, 98, 1391.

    Article  CAS  Google Scholar 

  2. V. A. Makarov, V. G. Granik, Russ. Chem. Rev., 1998, 67, 923.

    Article  Google Scholar 

  3. M. F. Gordeev, A. V. Komkov, V. A. Dorokhov, Chem. Heterocycl. Compd. (Engl. Transl.), 1990, 1286.

  4. V. A. Dorokhov, M. F. Gordeev, A. V. Komkov, V. S. Bogdanov, Bull. Acad. Sci. USSR, Div. Chem. Sci. (Engl. Transl.), 1991, 40, 2267.

    Article  Google Scholar 

  5. V. A. Dorokhov, V. S. Bogdanov, M. F. Gordeev, Russ. Chem. Bull. (Engl. Transl.), 1995, 44, 1276.

    Article  Google Scholar 

  6. V. A. Dorokhov, A. V. Komkov, Russ. Chem. Bull. (Int. Ed.), 2004, 53, 676.

    Article  CAS  Google Scholar 

  7. M. A. Prezent, V. A. Dorokhov, Russ. Chem. Bull. (Int. Ed.), 2005, 54, 1343.

    Article  CAS  Google Scholar 

  8. S. V. Ruban, T. V. Potapova, S. V. Baranin, V. A. Dorokhov, Russ. Chem. Bull. (Int. Ed.), 2014, 63, 2260.

    Article  CAS  Google Scholar 

  9. L. S. Vasil’ev, S. V. Baranin, I. V. Zavarzin, Russ. Chem. Bull. (Int. Ed.), 2017, 66, 1398.

    Article  Google Scholar 

  10. D. S. Khachatryan, I. I. Boyko, A. V. Kolotaev, K. R. Matevosyan, Russ. Chem. Bull. (Int. Ed.), 2020, 69, 325.

    Article  CAS  Google Scholar 

  11. M. I. Zuev, A. A. Sukhanova, A. G. Smola, M. A. Prezent, A. N. Proshin, S. V. Baranin, Yu. N. Bubnov, Mendeleev Commun., 2018, 28, 612.

    Article  CAS  Google Scholar 

  12. A. A. Sukhanova, M. I. Zuev, M. A. Prezent, A. N. Proshin, S. V. Baranin, Yu. N. Bubnov, Mendeleev Commun., 2019, 29, 196.

    Article  CAS  Google Scholar 

  13. V. A. Dorokhov, M. F. Gordeev, Bull. Acad. Sci. USSR, Div. Chem. Sci. (Engl. Transl.), 1989, 38, 2638.

    Article  Google Scholar 

  14. V. A. Dorokhov, M. A. Prezent, Russ. Chem. Bull. (Engl. Transl.), 1993, 42, 1442.

    Article  Google Scholar 

  15. V. A. Dorokhov, M. A. Prezent, Russ. Chem. Bull. (Engl. Transl.), 1994, 43, 832.

    Article  Google Scholar 

  16. V. A. Dorokhov, M. A. Prezent, V. S. Bogdanov, Russ. Chem. Bull. (Engl. Transl.), 1994, 43, 1550.

    Article  Google Scholar 

  17. V. A. Dorokhov, M. A. Prezent, V. S. Bogdanov, Russ. Chem. Bull. (Engl. Transl.), 1994, 43, 2091.

    Article  Google Scholar 

  18. V. A. Dorokhov, M. A. Prezent, M. F. Gordeev, V. S. Bogdanov, J. Org. Chem. Russia (Engl. Transl.), 1995, 31.

  19. V. A. Dorokhov, A. V. Komkov, A. M. Sakharov, V. S. Bogdanov, Russ. Chem. Bull. (Engl. Transl.), 1996, 45, 168.

    Article  Google Scholar 

  20. V. A. Dorokhov, Z. K. Dem’yanets, Russ. Chem. Bull. (Engl. Transl.), 1993, 42, 384.

    Article  Google Scholar 

  21. V. A. Dorokhov, M. F. Gordeev, Z. K. Dem’yanets, M. N. Bochkareva, V. S. Bogdanov, Bull. Acad. Sci. USSR, Div. Chem. Sci. (Engl. Transl.), 1989, 38, 1654.

    Article  Google Scholar 

  22. V. A. Dorokhov, M. F. Gordeev, E. M. Shashkova, A. M. Konkov, V. S. Bogdanov, Bull. Acad. Sci. USSR, Div. Chem. Sci. (Engl. Transl.), 1991, 40, 2274.

    Article  Google Scholar 

  23. V. A. Dorokhov, L. G. Vorontsova, M. G. Kurella, Russ. Chem. Bull. (Engl. Transl.), 1996, 45, 2411.

    Article  Google Scholar 

  24. M. Clare, S. C. Houdek, X. Xu, R. M. Weier, P. J. Lennon, T. J. Hagen, Pat. WO2005/40133, 2005, A1.

  25. A. A. Farahat, A. Kumar, M. Say, A. D. M. Barghash, F. E. Goda, H. M. Eisa, T. Wenzler, R. Brun, Y. Liu, L. Mickelson, W. D. Wilson, D. W. Boykin, Bioorg. Med. Chem., 2010, 18, 557.

    Article  CAS  Google Scholar 

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Authors and Affiliations

  1. N. D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, 47 Leninsky prosp., 119991, Moscow, Russian Federation

    M. A. Present, S. V. Baranin & Yu. N. Bubnov

Authors
  1. M. A. Present
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  2. S. V. Baranin
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  3. Yu. N. Bubnov
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Correspondence to S. V. Baranin.

Additional information

Published in Russian in Izvestiya Akademii Nauk. Seriya Khimicheskaya, No. 4, pp. 763–766, April, 2021.

The study was carried out as a part of the program for the development of scientific schools of ZIOC RAS.

This article does not contain a description of the researches carried out by the authors with the participation of humans or the use of animals as objects.

We have no conflict of interest in financial or other areas to declare.

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Present, M.A., Baranin, S.V. & Bubnov, Y.N. Chelate method for the synthesis of 3-amidino-substituted 4-pyridones. Russ Chem Bull 70, 763–766 (2021). https://doi.org/10.1007/s11172-021-3148-9

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  • DOI: https://doi.org/10.1007/s11172-021-3148-9

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