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A new method for the synthesis of n-(2-aminoethyl)azoles by alkylation of azoles with 2-alkyl-4,5-dihydrooxazoles

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Abstract

Ring opening in 2-alkyl-4,5-dihydrooxazoles by the action of azoles gave intermediate N-(2-azolylethyl)alkanamides, whose hydrolysis afforded N-(2-aminoethyl)azoles.

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Authors and Affiliations

  1. D. I. Mendeleev Russian University for Chemical Technology, 9 Miusskaya pl., 125047, Moscow, Russian Federation

    S. V. Popkov & M. N. Skvortsova

Authors
  1. S. V. Popkov
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  2. M. N. Skvortsova
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Published in Russian in Izvestiya Akademii Nauk. Seriya Khimicheskaya, No. 10, pp. 1781–1784, October, 2006.

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Popkov, S.V., Skvortsova, M.N. A new method for the synthesis of n-(2-aminoethyl)azoles by alkylation of azoles with 2-alkyl-4,5-dihydrooxazoles. Russ Chem Bull 55, 1848–1851 (2006). https://doi.org/10.1007/s11172-006-0496-4

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  • DOI: https://doi.org/10.1007/s11172-006-0496-4

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