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Reactivity of Substituted 2-Spiropyrimidin-4-Ones Under Vilsmeier–Haack Conditions

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Chemistry of Heterocyclic Compounds Aims and scope

Substituted 2-spiropyrimidin-4-ones are formylated at room temperature under the conditions of the Vilsmeier–Haack reaction. When cautiously heated they undergo electrophilic rearrangement.

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Authors and Affiliations

  1. Ukrainian State Chemical-Technology University, 8 Gagarine Ave., Dnepropetrovsk, 49005, Ukraine

    S. A. Varenichenko, O. K. Farat & V. I. Markov

Authors
  1. S. A. Varenichenko
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  2. O. K. Farat
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  3. V. I. Markov
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Correspondence to S. A. Varenichenko.

Additional information

Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 11, pp. 1743–1748, November, 2014.

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Varenichenko, S.A., Farat, O.K. & Markov, V.I. Reactivity of Substituted 2-Spiropyrimidin-4-Ones Under Vilsmeier–Haack Conditions. Chem Heterocycl Comp 50, 1602–1607 (2015). https://doi.org/10.1007/s10593-014-1626-9

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  • DOI: https://doi.org/10.1007/s10593-014-1626-9

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