A method has been developed for the synthesis of 3-S-hetaryl-substituted pyridin-2(1H)-ones and 5,6-dihydropyridin-2(1H)-ones based on the base catalyzed cyclization of N-(3-oxoalkyl)- and N-(3-oxoalkenyl)amides which contain a divalent sulfur atom in an α-position to a carbamoyl group and bound to the heterocycle.
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* Dedicated to the memory of the prominent scientist and wise teacher, Reva S. Sagitullin.
Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 7, pp. 1044-1049, July, 2010.
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Fisyuk, A.S., Bogza, Y.P., Poendaev, N.V. et al. Synthesis of 3-S-hetaryl-substituted pyridin-2(1H)-ones and 5,6-dihydropyridin-2(1H)-ones*. Chem Heterocycl Comp 46, 844–849 (2010). https://doi.org/10.1007/s10593-010-0592-0
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DOI: https://doi.org/10.1007/s10593-010-0592-0