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Polyfunctional pyrazoles 6.* Convenient method for the synthesis of 1-aryl-1H-pyrazole-3,4-dicarboxylic acids

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Chemistry of Heterocyclic Compounds Aims and scope

A preparatively convenient method was developed for the synthesis of 1-aryl-1H-pyrazole-3,4-di-carboxylic acids based on the alkaline hydrolysis and oxidation of 1-aryl-4-formyl-1H-pyrazole-3-carboxylic esters with hydrogen peroxide in an aqueous medium.

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Authors and Affiliations

  1. Bukovinian State Medical University, Chernovtsy, 58000, Ukraine

    M. K. Bratenko & M. M. Barus

  2. Institute of Organic Chemistry, National Academy of Sciences of Ukraine, Kiev, 02094, Ukraine

    M. V. Vovk

Authors
  1. M. K. Bratenko
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  2. M. M. Barus
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  3. M. V. Vovk
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Corresponding author

Correspondence to M. K. Bratenko.

Additional information

Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 2, pp. 243-247, February, 2010.

*For Communication 5 see [1].

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Bratenko, M.K., Barus, M.M. & Vovk, M.V. Polyfunctional pyrazoles 6.* Convenient method for the synthesis of 1-aryl-1H-pyrazole-3,4-dicarboxylic acids. Chem Heterocycl Comp 46, 196–199 (2010). https://doi.org/10.1007/s10593-010-0491-4

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  • DOI: https://doi.org/10.1007/s10593-010-0491-4

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