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One-pot synthesis of functionalized thioureas by reaction of benzoyl isothiocyanates, secondary amines, and alkyl propiolates

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Abstract

An efficient one-pot synthesis of functionalized thioureas is described via three-component reaction of benzoyl isothiocyanates, secondary amines, and alkyl propiolates in the presence of triphenylphosphine (20 mol%).

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Authors and Affiliations

  1. Chemistry Department, Science and Research Campus, Islamic Azad University, Ponak, Tehran, Iran

    Issa Yavari, S. Zahra Sayyed-Alangi, Rahimeh Hajinasiri & Nasir Iravani

  2. Chemistry Department, Tarbiat Modares University, Tehran, Iran

    Issa Yavari & Maryam Sabbaghan

Authors
  1. Issa Yavari
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  2. S. Zahra Sayyed-Alangi
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  3. Maryam Sabbaghan
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  4. Rahimeh Hajinasiri
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  5. Nasir Iravani
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Corresponding author

Correspondence to Issa Yavari.

Additional information

Correspondence: Issa Yavari, Chemistry Department, Tarbiat Modares University, PO Box 14115-175, Tehran, Iran

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Yavari, I., Sayyed-Alangi, S., Sabbaghan, M. et al. One-pot synthesis of functionalized thioureas by reaction of benzoyl isothiocyanates, secondary amines, and alkyl propiolates. Monatsh Chem 139, 1025–1028 (2008). https://doi.org/10.1007/s00706-008-0899-z

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  • DOI: https://doi.org/10.1007/s00706-008-0899-z

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