Abstract
5-Aryl-2,3-dihydrofuran-2,3-diones react with five-membered hetarylaminonitriles to give N-aroytpyruvoyl and N-aroylacetyt derivatives of the latter. The reaction of 2,2-dimethyl-6-aryl-1,3dioxin-4-ones with these hetarylaminonitriles leads solety to the N-aroylacetyl derivatives.
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Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 1, pp. 173–178, February, 1994. Original article submitted June 28, 1993.
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Nekrasov, D.D., Kol'tsova, S.V. & Andreichikov, Y.S. Synthesis of N-aroylpyruvoyl- and N-aroylacetyl-hetarylaminonitriles. Chem Heterocycl Compd 30, 154–159 (1994). https://doi.org/10.1007/BF01165003
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DOI: https://doi.org/10.1007/BF01165003