Chemistry of Heterocyclic Compounds

, Volume 24, Issue 12, pp 1373–1377 | Cite as

Nucleophilic substitution in hydroxyisoxazolidines

  • I. A. Motorina
  • L. A. Sviridova
  • G. A. Golubeva
  • K. N. Zelenin
  • I. P. Bezhan
  • A. Yu. Ershov
  • Yu. G. Bundel'
Article
  • 35 Downloads

Abstract

Nucleophilic substitution of the hydroxy-group in 3- (or 5-)hydroxyisoxazolidines affords the aryl(alkyl)amino-, alkoxy-, and hydrazino-compounds. 5-Dimethylhydrazinooxazolidines exist preferentially in the linear form.

Keywords

Organic Chemistry Linear Form Nucleophilic Substitution 

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Copyright information

© Plenum Publishing Corporation 1989

Authors and Affiliations

  • I. A. Motorina
    • 1
    • 2
  • L. A. Sviridova
    • 1
    • 2
  • G. A. Golubeva
    • 1
    • 2
  • K. N. Zelenin
    • 1
    • 2
  • I. P. Bezhan
    • 1
    • 2
  • A. Yu. Ershov
    • 1
    • 2
  • Yu. G. Bundel'
    • 1
    • 2
  1. 1.M. V. Lomonosov Moscow State UniversityMoscow
  2. 2.S. M. Korov Academy of Military MedicineLeningrad

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