Abstract
The Böckelheide reaction was accomplished with a number of imidazo[4,5-b]pyrazine N-oxides, and the N-oxidation of the resulting acetoxy(hydroxy)methyl derivatives of imidazo[4,5-b]pyrazine and 6-bromo-1-methylimidazo[4,5-b]pyrazine was studied. The hydrolytic cleavage of 6-bromo-1-methylimidazo[4,5-b]pyrazine and its 4-N-oxide was studied.
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Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 5, pp. 690–693, May, 1975.
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Elina, A.S., Musatova, I.S. Synthesis and transformation of N-oxides of some imidazo[4,5-b]pyrazine derivatives. Chem Heterocycl Compd 11, 600–602 (1975). https://doi.org/10.1007/BF00480488
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DOI: https://doi.org/10.1007/BF00480488