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Synthesis of New Amides of Isoxazole- and Isothiazole-Substituted Carboxylic Acids Containing an Arylaminopyrimidine Fragment

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Abstract

By acylation of substituted 2-aminoarylpyrimidines with 5-phenyl(p-tolyl)isoxazole- and 4,5-dichloroisothiazole-3-carbonyl chlorides new amides of pyrimidine series were obtained.

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Authors and Affiliations

  1. Institute of Chemistry of New Materials, National Academy of Sciences of Belarus, ul. F. Skoriny 36, Minsk, 220141, Belarus

    Zh. V. Ignatovich, A. L. Ermolinskaya & E. V. Koroleva

  2. Institute of Physical Organic Chemistry, National Academy of Sciences of Belarus, Minsk, 220072, Belarus

    A. V. Kletskov & V. I. Potkin

Authors
  1. Zh. V. Ignatovich
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  2. A. L. Ermolinskaya
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  3. A. V. Kletskov
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  4. V. I. Potkin
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  5. E. V. Koroleva
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Corresponding author

Correspondence to E. V. Koroleva.

Additional information

Original Russian Text © Zh.V. Ignatovich, A.L. Ermolinskaya, A.V. Kletskov, V.I. Potkin, E.V. Koroleva, 2018, published in Zhurnal Organicheskoi Khimii, 2018, Vol. 54, No. 8, pp. 1207–1210.

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Ignatovich, Z.V., Ermolinskaya, A.L., Kletskov, A.V. et al. Synthesis of New Amides of Isoxazole- and Isothiazole-Substituted Carboxylic Acids Containing an Arylaminopyrimidine Fragment. Russ J Org Chem 54, 1218–1222 (2018). https://doi.org/10.1134/S107042801808016X

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  • DOI: https://doi.org/10.1134/S107042801808016X

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