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Synthesis of 4-(1Н-1,2,3-Triazol-4-Yl)-1,3-Thiazole-2-Amine Derivatives

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Chemistry of Heterocyclic Compounds Aims and scope

A series of previously unreported thiazole derivatives, 4-(1H-1,2,3-triazol-4-yl)-1,3-thiazole-2-amines, was prepared by the Hantzsch reaction between the respective 1,2,3-triazole α-bromo ketones and (het)arylthioureas.

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The authors would like to express their gratitude to the Ministry of Education and Science of the Russian Federation for the financial support (state assignment No. 426).

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Authors and Affiliations

  1. Togliatti State University, 14 Belorusskaya St., Togliatti, 445667, Russia

    A. S. Bunev, Yu. O. Trushkova, G. I. Ostapenko & V. E. Statsyuk

  2. A. N. Nesmeyanov Institute of Organoelement Compounds of Russian Academy of Sciences, 8 Vavilova St., Moscow, 119991, Russia

    A. S. Peregudov

Authors
  1. A. S. Bunev
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  2. Yu. O. Trushkova
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  3. G. I. Ostapenko
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  4. V. E. Statsyuk
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  5. A. S. Peregudov
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Correspondence to A. S. Bunev.

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Dedicated to Academician O. N. Chupakhin on the occasion of his 80th birthday.

Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 7, pp. 1114-1118, July, 2014.

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Bunev, A.S., Trushkova, Y.O., Ostapenko, G.I. et al. Synthesis of 4-(1Н-1,2,3-Triazol-4-Yl)-1,3-Thiazole-2-Amine Derivatives. Chem Heterocycl Comp 50, 1027–1031 (2014). https://doi.org/10.1007/s10593-014-1559-3

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  • DOI: https://doi.org/10.1007/s10593-014-1559-3

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