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Synthesis of 5H-thiazolo[3,2-a]pyrimidines

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Chemistry of Heterocyclic Compounds Aims and scope

A convenient method has been developed for preparing 5H-thiazolo[3,2-a]pyrimidines by the reaction of tetrahydropyrimidine-2-thiones with halocarboxylic acid esters or with 3-bromopentane-2,4-dione.

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Authors and Affiliations

  1. Samara State Technical University, 244 Molodogvardeiskaya St., Samara, 443100, Russia

    A. K. Shiryaev, N. S. Baranovskaya & M. S. Eremin

Authors
  1. A. K. Shiryaev
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  2. N. S. Baranovskaya
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  3. M. S. Eremin
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Corresponding author

Correspondence to A. K. Shiryaev.

Additional information

Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 10, pp. 1662-1667, October, 2012.

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Shiryaev, A.K., Baranovskaya, N.S. & Eremin, M.S. Synthesis of 5H-thiazolo[3,2-a]pyrimidines. Chem Heterocycl Comp 48, 1550–1554 (2013). https://doi.org/10.1007/s10593-013-1172-x

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  • DOI: https://doi.org/10.1007/s10593-013-1172-x

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