Abstract
Reaction of 2,4,6-trimethylaniline with acrylic and itaconic acids gives the corresponding N-substituted β=alanines which can be converted to derivatives of tetrahydropyridone, dihydropyrimidinedione, and 4-carboxy-2-pyrrolidinone. Bromination of the aromatic substituent in the synthesized heterocycles has been carried out.
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Kaunas Technological University, Kaunas 3028, Lithuania Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 7, pp. 951–954, July, 2000
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Mickevicius, V., Patupaite, A. Cyclization of N-(2,4,6-trimethylphenyl)-β-alanines. Chem Heterocycl Compd 36, 837–840 (2000). https://doi.org/10.1007/BF02256919
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DOI: https://doi.org/10.1007/BF02256919